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Industrial and academic approaches to the search for alternative melatonin receptor ligands: An historical survey. 1-gen-2024 Bedini, Annalida; Boutin, Jean A.; Legros, Céline; Zlotos, Darius P.; Spadoni, Gilberto
Binding and unbinding of potent melatonin receptor ligands: Mechanistic simulations and experimental evidence 1-gen-2024 Bedini, Annalida; Elisi, Gian Marco; Fanini, Fabiola; Retini, Michele; Scalvini, Laura; Pasquini, Silvia; Contri, Chiara; Varani, Katia; Spadoni, Gilberto; Mor, Marco; Vincenzi, Fabrizio; Rivara, Silvia
Combined targeting of fatty acid amide hydrolase and melatonin receptors promotes neuroprotection and stimulates inflammation resolution in rats 1-gen-2023 Cammarota, Mariarosaria; Ferlenghi, Francesca; Vacondio, Federica; Vincenzi, Fabrizio; Varani, Katia; Bedini, Annalida; Rivara, Silvia; Mor, Marco; Boscia, Francesca
Radiosynthesis and In Vivo Evaluation of Four Positron Emission Tomography Tracer Candidates for Imaging of Melatonin Receptors 1-gen-2022 Bdair, Hussein; Singleton, Thomas A; Ross, Karen; Jolly, Dean; Kang, Min Su; Aliaga, Arturo; Tuznik, Marius; Kaur, Tanpreet; Yous, Saïd; Soucy, Jean-Paul; Massarweh, Gassan; Scott, Peter J H; Koeppe, Robert; Spadoni, Gilberto; Bedini, Annalida; Rudko, David A; Gobbi, Gabriella; Benkelfat, Chawki; Rosa-Neto, Pedro; Brooks, Allen F; Kostikov, Alexey
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors 1-gen-2022 Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
In silico drug discovery of melatonin receptor ligands with therapeutic potential 1-gen-2022 Elisi, Gian Marco; Scalvini, Laura; Lodola, Alessio; Bedini, Annalida; Spadoni, Gilberto; Rivara, Silvia
N-(Anilinoethyl)amide Melatonergic Ligands with Improved Water Solubility and Metabolic Stability 1-gen-2021 Ferlenghi, Francesca; Mari, Michele; Gobbi, Gabriella; Elisi, Gian Marco; Mor, Marco; Rivara, Silvia; Vacondio, Federica; Bartolucci, Silvia; Bedini, Annalida; Fanini, Fabiola; Spadoni, Gilberto
Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma 1-gen-2021 Castelli, Riccardo; Taranto, Sara; Furiassi, Lucia; Bozza, Nicole; Marseglia, Giuseppe; Ferlenghi, Francesca; Rivara, Silvia; Retini, Michele; Bedini, Annalida; Spadoni, Gilberto; Matarazzo, Sara; Ronca, Roberto; Presta, Marco; Mor, Marco; Giacomini, Arianna
Dysfunction of serotonergic activity and emotional responses across the light-dark cycle in mice lacking melatonin  MT2 receptors 1-gen-2020 Comai, Stefano; De Gregorio, Danilo; Posa, Luca; Ochoa-Sanchez, Rafael; Bedini, Annalida; Gobbi, Gabriella
Chiral Recognition of Flexible Melatonin Receptor Ligands Induced by Conformational Equilibria 1-gen-2020 Elisi, Gian Marco; Bedini, Annalida; Scalvini, Laura; Carmi, Caterina; Bartolucci, Silvia; Lucini, Valeria; Scaglione, Francesco; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
Melatonin MT1 and MT2 Receptors Exhibit Distinct Effects in the Modulation of Body Temperature across the Light/Dark Cycle 1-gen-2019 López-Canul, Martha; Min, Seung Hyun; Posa, Luca; De Gregorio, Danilo; Bedini, Annalida; Spadoni, Gilberto; Gobbi, Gabriella; Comai, Stefano
Design, synthesis and biological activity of hydrogen peroxide responsive arylboronate melatonin hybrids 1-gen-2019 Bedini, Annalida; Fraternale, Alessandra; Crinelli, Rita; Mari, Michele; Bartolucci, Silvia; Chiarantini, Laura; Spadoni, Gilberto
Identification of Bivalent Ligands with Melatonin Receptor Agonist and Fatty Acid Amide Hydrolase (FAAH) Inhibitory Activity That Exhibit Ocular Hypotensive Effect in the Rabbit 1-gen-2018 Spadoni, G; Bedini, A; Furiassi, L; Mari, M; Mor, M; Scalvini, L; Lodola, A; Ghidini, A; Lucini, V; Dugnani, S; Scaglione, F; Piomelli, D; Jung, Km; Supuran, Ct; Lucarini, L; Durante, M; Sgambellone, S; Masini, E; Rivara, S.
Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands 1-gen-2018 Rivara, Silvia; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Caignard, Daniel-Henri; Delagrange, Philippe; Collina, Simona; Lucini, Valeria; Scaglione, Francesco; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto
Antiproliferative and pro-apoptotic activity of melatonin analogues on melanoma and breast cancer cells 1-gen-2017 Gatti, Giuliana; Lucini, Valeria; Dugnani, Silvana; Calastretti, Angela; Spadoni, Gilberto; Bedini, Annalida; Rivara, Silvia; Mor, Marco; Canti, Gianfranco; Scaglione, Francesco; Bevilacqua, Annamaria
Cardioprotective effects of fatty acid amide hydrolase inhibitor URB694, in a rodent model of trait anxiety 1-gen-2015 Carnevali, L.; Vacondio, F.; Rossi, S.; Macchi, E.; Spadoni, Gilberto; Bedini, Annalida; Neumann, I.; Rivara, S.; Mor, M; Sgoifo, A.
Antidepressant-like activity and cardioprotective effects of fatty acid amide hydrolase inhibitor URB694 in socially stressed Wistar Kyoto rats 1-gen-2015 Sgoifo, A.; Carnevali, L.; Vacondio, F.; Rossi, S.; Callegari, S.; Macchi, E.; Spadoni, Gilberto; Bedini, Annalida; Rivara, S.; Mor, M.
Selective Melatonin MT2 receptor ligands relieve neuropathic pain through modulation of brainstem descending antinociceptive pathways 1-gen-2015 M., Lopez Canul; E., Palazzo; S., Dominguez Lopez; L., Luongo; B., Lacoste; S., Comai; D., Angeloni; F., Fraschini; S., Boccella; Spadoni, Gilberto; Bedini, Annalida; G., Tarzia; S., Maione; V., Granado Sotos; G., Gobbi
Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents 1-gen-2015 Bartolucci, Silvia; Mari, Michele; Bedini, Annalida; Piersanti, Giovanni; Spadoni, Gilberto
Therapeutic uses of melatonin and melatonin derivatives: a patent review (2012-2014) 1-gen-2015 S., Rivara; D., Pala; Bedini, Annalida; Spadoni, Gilberto
Mostrati risultati da 1 a 20 di 112
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