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Binding and unbinding of potent melatonin receptor ligands: Mechanistic simulations and experimental evidence 1-gen-2024 Bedini, Annalida; Elisi, Gian Marco; Fanini, Fabiola; Retini, Michele; Scalvini, Laura; Pasquini, Silvia; Contri, Chiara; Varani, Katia; Spadoni, Gilberto; Mor, Marco; Vincenzi, Fabrizio; Rivara, Silvia
Practical and Selective Syntheses of S‐Acyl and N‐Acyl Glutathiones with N‐Acyl Imidazoles in Water 1-gen-2024 Retini, Michele; Sisti, Andrea; Olivieri, Diego; Mari, Michele; Bartoccini, Francesca; Piersanti, Giovanni
Paradigm Shift in Gastric Cancer Prevention: Harnessing the Potential of Aristolochia olivieri Extract 1-gen-2023 Micucci, Matteo; Stella Bartoletti, Anna; Abdullah, Fuad O; Burattini, Sabrina; Versari, Ilaria; Canale, Matteo; D'Agostino, Federico; Roncarati, Davide; Piatti, Diletta; Sagratini, Gianni; Caprioli, Giovanni; Mari, Michele; Retini, Michele; Faenza, Irene; Battistelli, Michela; Salucci, Sara
A potential host and virus targeting tool against COVID-19: Chemical characterization, antiviral, cytoprotective, antioxidant, respiratory smooth muscle relaxant effects of Paulownia tomentosa Steud 1-gen-2023 Magurano, Fabio; Micucci, Matteo; Nuzzo, Domenico; Baggieri, Melissa; Picone, Pasquale; Gioacchini, Silvia; Fioravanti, Raoul; Bucci, Paola; Kojouri, Maedeh; Mari, Michele; Retini, Michele; Budriesi, Roberta; Mattioli, Laura Beatrice; Corazza, Ivan; Di Liberto, Valentina; Todaro, Luigi; Giuseppetti, Roberto; D'Ugo, Emilio; Marchi, Antonella; Mecca, Marisabel; D'Auria, Maurizio
Targeting SARS-CoV-2 by synthetic dual-acting thiol compounds that inhibit Spike/ACE2 interaction and viral protein production 1-gen-2023 Fraternale, Alessandra; De Angelis, Marta; De Santis, Riccardo; Amatore, Donatella; Masini, Sofia; Monittola, Francesca; Menotta, Michele; Biancucci, Federica; Bartoccini, Francesca; Retini, Michele; Fiori, Valentina; Fioravanti, Raoul; Magurano, Fabio; Chiarantini, Laura; Lista, Romano F; Piersanti, Giovanni; Palamara, Anna T; Nencioni, Lucia; Magnani, Mauro; Crinelli, Rita
Inhibition of myeloid-derived suppressor cell (MDSC) activity by redox-modulating agents restores T and B cell proliferative responses in murine AIDS 1-gen-2023 Fraternale, Alessandra; Green, Kathy A.; Schiavano, Giuditta F.; Bruschi, Michela; Retini, Michele; Magnani, Mauro; Green, William R.
Synthesis and Fluorescence Properties of 4-Cyano and 4-Formyl Melatonin as Putative Melatoninergic Ligands 1-gen-2023 Bartolucci, Silvia; Retini, Michele; Fanini, Fabiola; Paderni, Daniele; Piersanti, Giovanni
Asymmetric Alkylation of Cyclic Ketones with Dehydroalanine via H-Bond-Directing Enamine Catalysis: Straightforward Access to Enantiopure Unnatural α-Amino Acids 1-gen-2022 Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors 1-gen-2022 Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
Dithiol Based on L-Cysteine and Cysteamine as a Disulfide-Reducing Agent 1-gen-2022 Bartoccini, Francesca; Retini, Michele; Crinelli, Rita; Menotta, Michele; Fraternale, Alessandra; Piersanti, Giovanni
Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties 1-gen-2022 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Intracellular Redox-Modulated Pathways as Targets for Effective Approaches in the Treatment of Viral Infection 1-gen-2021 Fraternale, Alessandra; Zara, Carolina; De Angelis, Marta; Nencioni, Lucia; Palamara, Anna Teresa; Retini, Michele; Di Mambro, Tomas; Magnani, Mauro; Crinelli, Rita
Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma 1-gen-2021 Castelli, Riccardo; Taranto, Sara; Furiassi, Lucia; Bozza, Nicole; Marseglia, Giuseppe; Ferlenghi, Francesca; Rivara, Silvia; Retini, Michele; Bedini, Annalida; Spadoni, Gilberto; Matarazzo, Sara; Ronca, Roberto; Presta, Marco; Mor, Marco; Giacomini, Arianna
Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone 1-gen-2021 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Novel, Chiral, and Enantiopure C2‐Symmetric Thioureas Promote Asymmetric Protio‐Pictet‐Spengler Reactions by Anion‐Binding Catalysis 1-gen-2021 Retini, Michele; Bartoccini, Francesca; Zappia, Giovanni; Piersanti, Giovanni
Single‐Step Synthesis of Dehydroalanine Derivatives via a Brønsted Acid‐Catalyzed Multicomponent Reaction 1-gen-2020 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Galarini, Roberta; Bartolucci, Silvia; Piersanti, Giovanni
General synthesis of unnatural 4-, 5-, 6-, and 7-bromo-d-tryptophans by means of a regioselective indole alkylation 1-gen-2020 Bartoccini, Francesca; Fanini, Fabiola; Retini, Michele; Piersanti, Giovanni
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign 1-gen-2020 Linciano, Pasquale; Cullia, Gregorio; Borsari, Chiara; Santucci, Matteo; Ferrari, Stefania; Witt, Gesa; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Santarém, Nuno; Cordeiro da Silva, Anabela; Conti, Paola; Bolognesi, Maria Laura; Roberti, Marinella; Prati, Federica; Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni; Cavalli, Andrea; Goldoni, Luca; Bertozzi, Sine Mandrup; Bertozzi, Fabio; Brambilla, Enzo; Rizzo, Vincenzo; Piomelli, Daniele; Pinto, Andrea; Bandiera, Tiziano; Costi, Maria Paola
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology 1-gen-2020 Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni
Boosting GSH Using the Co-Drug Approach: I-152, a Conjugate of N-acetyl-cysteine and β-mercaptoethylamine 1-gen-2019 Crinelli, Rita; Zara, Carolina; Smietana, Michaël; Retini, Michele; Magnani, Mauro; Fraternale, Alessandra
Mostrati risultati da 1 a 20 di 27
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