Sfoglia per Autore
Industrial and academic approaches to the search for alternative melatonin receptor ligands: An historical survey.
2024 Bedini, Annalida; Boutin, Jean A.; Legros, Céline; Zlotos, Darius P.; Spadoni, Gilberto
Binding and unbinding of potent melatonin receptor ligands: Mechanistic simulations and experimental evidence
2024 Bedini, Annalida; Elisi, Gian Marco; Fanini, Fabiola; Retini, Michele; Scalvini, Laura; Pasquini, Silvia; Contri, Chiara; Varani, Katia; Spadoni, Gilberto; Mor, Marco; Vincenzi, Fabrizio; Rivara, Silvia
Combined targeting of fatty acid amide hydrolase and melatonin receptors promotes neuroprotection and stimulates inflammation resolution in rats
2023 Cammarota, Mariarosaria; Ferlenghi, Francesca; Vacondio, Federica; Vincenzi, Fabrizio; Varani, Katia; Bedini, Annalida; Rivara, Silvia; Mor, Marco; Boscia, Francesca
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors
2022 Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
Radiosynthesis and In Vivo Evaluation of Four Positron Emission Tomography Tracer Candidates for Imaging of Melatonin Receptors
2022 Bdair, Hussein; Singleton, Thomas A; Ross, Karen; Jolly, Dean; Kang, Min Su; Aliaga, Arturo; Tuznik, Marius; Kaur, Tanpreet; Yous, Saïd; Soucy, Jean-Paul; Massarweh, Gassan; Scott, Peter J H; Koeppe, Robert; Spadoni, Gilberto; Bedini, Annalida; Rudko, David A; Gobbi, Gabriella; Benkelfat, Chawki; Rosa-Neto, Pedro; Brooks, Allen F; Kostikov, Alexey
In silico drug discovery of melatonin receptor ligands with therapeutic potential
2022 Elisi, Gian Marco; Scalvini, Laura; Lodola, Alessio; Bedini, Annalida; Spadoni, Gilberto; Rivara, Silvia
Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma
2021 Castelli, Riccardo; Taranto, Sara; Furiassi, Lucia; Bozza, Nicole; Marseglia, Giuseppe; Ferlenghi, Francesca; Rivara, Silvia; Retini, Michele; Bedini, Annalida; Spadoni, Gilberto; Matarazzo, Sara; Ronca, Roberto; Presta, Marco; Mor, Marco; Giacomini, Arianna
N-(Anilinoethyl)amide Melatonergic Ligands with Improved Water Solubility and Metabolic Stability
2021 Ferlenghi, Francesca; Mari, Michele; Gobbi, Gabriella; Elisi, Gian Marco; Mor, Marco; Rivara, Silvia; Vacondio, Federica; Bartolucci, Silvia; Bedini, Annalida; Fanini, Fabiola; Spadoni, Gilberto
Dysfunction of serotonergic activity and emotional responses across the light-dark cycle in mice lacking melatonin MT2 receptors
2020 Comai, Stefano; De Gregorio, Danilo; Posa, Luca; Ochoa-Sanchez, Rafael; Bedini, Annalida; Gobbi, Gabriella
Chiral Recognition of Flexible Melatonin Receptor Ligands Induced by Conformational Equilibria
2020 Elisi, Gian Marco; Bedini, Annalida; Scalvini, Laura; Carmi, Caterina; Bartolucci, Silvia; Lucini, Valeria; Scaglione, Francesco; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
Design, synthesis and biological activity of hydrogen peroxide responsive arylboronate melatonin hybrids
2019 Bedini, Annalida; Fraternale, Alessandra; Crinelli, Rita; Mari, Michele; Bartolucci, Silvia; Chiarantini, Laura; Spadoni, Gilberto
Melatonin MT1 and MT2 Receptors Exhibit Distinct Effects in the Modulation of Body Temperature across the Light/Dark Cycle
2019 López-Canul, Martha; Min, Seung Hyun; Posa, Luca; De Gregorio, Danilo; Bedini, Annalida; Spadoni, Gilberto; Gobbi, Gabriella; Comai, Stefano
Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands
2018 Rivara, Silvia; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Caignard, Daniel-Henri; Delagrange, Philippe; Collina, Simona; Lucini, Valeria; Scaglione, Francesco; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto
Identification of Bivalent Ligands with Melatonin Receptor Agonist and Fatty Acid Amide Hydrolase (FAAH) Inhibitory Activity That Exhibit Ocular Hypotensive Effect in the Rabbit
2018 Spadoni, G; Bedini, A; Furiassi, L; Mari, M; Mor, M; Scalvini, L; Lodola, A; Ghidini, A; Lucini, V; Dugnani, S; Scaglione, F; Piomelli, D; Jung, Km; Supuran, Ct; Lucarini, L; Durante, M; Sgambellone, S; Masini, E; Rivara, S.
Antiproliferative and pro-apoptotic activity of melatonin analogues on melanoma and breast cancer cells
2017 Gatti, Giuliana; Lucini, Valeria; Dugnani, Silvana; Calastretti, Angela; Spadoni, Gilberto; Bedini, Annalida; Rivara, Silvia; Mor, Marco; Canti, Gianfranco; Scaglione, Francesco; Bevilacqua, Annamaria
Selective Melatonin MT2 receptor ligands relieve neuropathic pain through modulation of brainstem descending antinociceptive pathways
2015 M., Lopez Canul; E., Palazzo; S., Dominguez Lopez; L., Luongo; B., Lacoste; S., Comai; D., Angeloni; F., Fraschini; S., Boccella; Spadoni, Gilberto; Bedini, Annalida; G., Tarzia; S., Maione; V., Granado Sotos; G., Gobbi
Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents
2015 Bartolucci, Silvia; Mari, Michele; Bedini, Annalida; Piersanti, Giovanni; Spadoni, Gilberto
Pharmacokinetic and pharmacodynamic evaluation of ramelteon : an insomnia therapy
2015 Spadoni, Gilberto; Bedini, Annalida; Lucarini, Simone; Mor, Marco; Rivara, Silvia
Cardioprotective effects of fatty acid amide hydrolase inhibitor URB694, in a rodent model of trait anxiety
2015 Carnevali, L.; Vacondio, F.; Rossi, S.; Macchi, E.; Spadoni, Gilberto; Bedini, Annalida; Neumann, I.; Rivara, S.; Mor, M; Sgoifo, A.
Antidepressant-like activity and cardioprotective effects of fatty acid amide hydrolase inhibitor URB694 in socially stressed Wistar Kyoto rats
2015 Sgoifo, A.; Carnevali, L.; Vacondio, F.; Rossi, S.; Callegari, S.; Macchi, E.; Spadoni, Gilberto; Bedini, Annalida; Rivara, S.; Mor, M.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Industrial and academic approaches to the search for alternative melatonin receptor ligands: An historical survey. | 1-gen-2024 | Bedini, Annalida; Boutin, Jean A.; Legros, Céline; Zlotos, Darius P.; Spadoni, Gilberto | |
Binding and unbinding of potent melatonin receptor ligands: Mechanistic simulations and experimental evidence | 1-gen-2024 | Bedini, Annalida; Elisi, Gian Marco; Fanini, Fabiola; Retini, Michele; Scalvini, Laura; Pasquini, Silvia; Contri, Chiara; Varani, Katia; Spadoni, Gilberto; Mor, Marco; Vincenzi, Fabrizio; Rivara, Silvia | |
Combined targeting of fatty acid amide hydrolase and melatonin receptors promotes neuroprotection and stimulates inflammation resolution in rats | 1-gen-2023 | Cammarota, Mariarosaria; Ferlenghi, Francesca; Vacondio, Federica; Vincenzi, Fabrizio; Varani, Katia; Bedini, Annalida; Rivara, Silvia; Mor, Marco; Boscia, Francesca | |
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors | 1-gen-2022 | Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto | |
Radiosynthesis and In Vivo Evaluation of Four Positron Emission Tomography Tracer Candidates for Imaging of Melatonin Receptors | 1-gen-2022 | Bdair, Hussein; Singleton, Thomas A; Ross, Karen; Jolly, Dean; Kang, Min Su; Aliaga, Arturo; Tuznik, Marius; Kaur, Tanpreet; Yous, Saïd; Soucy, Jean-Paul; Massarweh, Gassan; Scott, Peter J H; Koeppe, Robert; Spadoni, Gilberto; Bedini, Annalida; Rudko, David A; Gobbi, Gabriella; Benkelfat, Chawki; Rosa-Neto, Pedro; Brooks, Allen F; Kostikov, Alexey | |
In silico drug discovery of melatonin receptor ligands with therapeutic potential | 1-gen-2022 | Elisi, Gian Marco; Scalvini, Laura; Lodola, Alessio; Bedini, Annalida; Spadoni, Gilberto; Rivara, Silvia | |
Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma | 1-gen-2021 | Castelli, Riccardo; Taranto, Sara; Furiassi, Lucia; Bozza, Nicole; Marseglia, Giuseppe; Ferlenghi, Francesca; Rivara, Silvia; Retini, Michele; Bedini, Annalida; Spadoni, Gilberto; Matarazzo, Sara; Ronca, Roberto; Presta, Marco; Mor, Marco; Giacomini, Arianna | |
N-(Anilinoethyl)amide Melatonergic Ligands with Improved Water Solubility and Metabolic Stability | 1-gen-2021 | Ferlenghi, Francesca; Mari, Michele; Gobbi, Gabriella; Elisi, Gian Marco; Mor, Marco; Rivara, Silvia; Vacondio, Federica; Bartolucci, Silvia; Bedini, Annalida; Fanini, Fabiola; Spadoni, Gilberto | |
Dysfunction of serotonergic activity and emotional responses across the light-dark cycle in mice lacking melatonin MT2 receptors | 1-gen-2020 | Comai, Stefano; De Gregorio, Danilo; Posa, Luca; Ochoa-Sanchez, Rafael; Bedini, Annalida; Gobbi, Gabriella | |
Chiral Recognition of Flexible Melatonin Receptor Ligands Induced by Conformational Equilibria | 1-gen-2020 | Elisi, Gian Marco; Bedini, Annalida; Scalvini, Laura; Carmi, Caterina; Bartolucci, Silvia; Lucini, Valeria; Scaglione, Francesco; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto | |
Design, synthesis and biological activity of hydrogen peroxide responsive arylboronate melatonin hybrids | 1-gen-2019 | Bedini, Annalida; Fraternale, Alessandra; Crinelli, Rita; Mari, Michele; Bartolucci, Silvia; Chiarantini, Laura; Spadoni, Gilberto | |
Melatonin MT1 and MT2 Receptors Exhibit Distinct Effects in the Modulation of Body Temperature across the Light/Dark Cycle | 1-gen-2019 | López-Canul, Martha; Min, Seung Hyun; Posa, Luca; De Gregorio, Danilo; Bedini, Annalida; Spadoni, Gilberto; Gobbi, Gabriella; Comai, Stefano | |
Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands | 1-gen-2018 | Rivara, Silvia; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Caignard, Daniel-Henri; Delagrange, Philippe; Collina, Simona; Lucini, Valeria; Scaglione, Francesco; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto | |
Identification of Bivalent Ligands with Melatonin Receptor Agonist and Fatty Acid Amide Hydrolase (FAAH) Inhibitory Activity That Exhibit Ocular Hypotensive Effect in the Rabbit | 1-gen-2018 | Spadoni, G; Bedini, A; Furiassi, L; Mari, M; Mor, M; Scalvini, L; Lodola, A; Ghidini, A; Lucini, V; Dugnani, S; Scaglione, F; Piomelli, D; Jung, Km; Supuran, Ct; Lucarini, L; Durante, M; Sgambellone, S; Masini, E; Rivara, S. | |
Antiproliferative and pro-apoptotic activity of melatonin analogues on melanoma and breast cancer cells | 1-gen-2017 | Gatti, Giuliana; Lucini, Valeria; Dugnani, Silvana; Calastretti, Angela; Spadoni, Gilberto; Bedini, Annalida; Rivara, Silvia; Mor, Marco; Canti, Gianfranco; Scaglione, Francesco; Bevilacqua, Annamaria | |
Selective Melatonin MT2 receptor ligands relieve neuropathic pain through modulation of brainstem descending antinociceptive pathways | 1-gen-2015 | M., Lopez Canul; E., Palazzo; S., Dominguez Lopez; L., Luongo; B., Lacoste; S., Comai; D., Angeloni; F., Fraschini; S., Boccella; Spadoni, Gilberto; Bedini, Annalida; G., Tarzia; S., Maione; V., Granado Sotos; G., Gobbi | |
Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents | 1-gen-2015 | Bartolucci, Silvia; Mari, Michele; Bedini, Annalida; Piersanti, Giovanni; Spadoni, Gilberto | |
Pharmacokinetic and pharmacodynamic evaluation of ramelteon : an insomnia therapy | 1-gen-2015 | Spadoni, Gilberto; Bedini, Annalida; Lucarini, Simone; Mor, Marco; Rivara, Silvia | |
Cardioprotective effects of fatty acid amide hydrolase inhibitor URB694, in a rodent model of trait anxiety | 1-gen-2015 | Carnevali, L.; Vacondio, F.; Rossi, S.; Macchi, E.; Spadoni, Gilberto; Bedini, Annalida; Neumann, I.; Rivara, S.; Mor, M; Sgoifo, A. | |
Antidepressant-like activity and cardioprotective effects of fatty acid amide hydrolase inhibitor URB694 in socially stressed Wistar Kyoto rats | 1-gen-2015 | Sgoifo, A.; Carnevali, L.; Vacondio, F.; Rossi, S.; Callegari, S.; Macchi, E.; Spadoni, Gilberto; Bedini, Annalida; Rivara, S.; Mor, M. |
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