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Mostrati risultati da 1 a 20 di 47
Titolo Data di pubblicazione Autore(i) File
A Short Synthesis of (−)‐6,7‐Secoagroclavine via Metal‐Free Reductive Coupling 1-gen-2024 Diotallevi, Francesca; Bartoccini, Francesca; Piersanti, Giovanni
General Access to Clavine Alkaloids via a Rhodium(I)‐Catalyzed Diastereoselective Hayashi‐Miyaura Reaction 1-gen-2024 Leoni, Giovanni; Bartoccini, Francesca; Piersanti, Giovanni
Enantioselective organocatalytic strategies to noncanonical α‐amino acids 1-gen-2024 Pecchini, Pietro; Fochi, Mariafrancesca; Bartoccini, Francesca; Piersanti, Giovanni; Bernardi, Luca
A synthetic thiol molecule releasing N-acetyl-l-cysteine and cysteamine drives early up-regulation of immunoproteasome subunits in the lymph nodes of mice infected with LP-BM5 leukemia retrovirus 1-gen-2024 Crinelli, Rita; Monittola, Francesca; Masini, Sofia; Diotallevi, Aurora; Bartoccini, Francesca; Smietana, Michaël; Galluzzi, Luca; Magnani, Mauro; Fraternale, Alessandra
Photoredox catalysis enabling decarboxylative radical cyclization of γ,γ-dimethylallyltryptophan (DMAT) derivatives: formal synthesis of 6,7-secoagroclavine 1-gen-2023 Regni, Alessio; Bartoccini, Francesca; Piersanti, Giovanni
The influence of redox modulation on hypoxic endothelial cell metabolic and proteomic profiles through a small thiol-based compound tuning glutathione and thioredoxin systems 1-gen-2023 Bruschi, Michela; Biancucci, Federica; Masini, Sofia; Piacente, Francesco; Ligi, Daniela; Bartoccini, Francesca; Antonelli, Antonella; Mannello, Ferdinando; Bruzzone, Santina; Menotta, Michele; Fraternale, Alessandra; Magnani, Mauro
Targeting SARS-CoV-2 by synthetic dual-acting thiol compounds that inhibit Spike/ACE2 interaction and viral protein production 1-gen-2023 Fraternale, Alessandra; De Angelis, Marta; De Santis, Riccardo; Amatore, Donatella; Masini, Sofia; Monittola, Francesca; Menotta, Michele; Biancucci, Federica; Bartoccini, Francesca; Retini, Michele; Fiori, Valentina; Fioravanti, Raoul; Magurano, Fabio; Chiarantini, Laura; Lista, Romano F; Piersanti, Giovanni; Palamara, Anna T; Nencioni, Lucia; Magnani, Mauro; Crinelli, Rita
Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties 1-gen-2022 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Asymmetric Alkylation of Cyclic Ketones with Dehydroalanine via H-Bond-Directing Enamine Catalysis: Straightforward Access to Enantiopure Unnatural α-Amino Acids 1-gen-2022 Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni
Dithiol Based on L-Cysteine and Cysteamine as a Disulfide-Reducing Agent 1-gen-2022 Bartoccini, Francesca; Retini, Michele; Crinelli, Rita; Menotta, Michele; Fraternale, Alessandra; Piersanti, Giovanni
Synthesis and Reactivity of Uhle’s Ketone and Its Derivatives 1-gen-2021 Piersanti, Giovanni; Bartoccini, Francesca
Novel, Chiral, and Enantiopure C2‐Symmetric Thioureas Promote Asymmetric Protio‐Pictet‐Spengler Reactions by Anion‐Binding Catalysis 1-gen-2021 Retini, Michele; Bartoccini, Francesca; Zappia, Giovanni; Piersanti, Giovanni
Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone 1-gen-2021 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology 1-gen-2020 Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni
Single‐Step Synthesis of Dehydroalanine Derivatives via a Brønsted Acid‐Catalyzed Multicomponent Reaction 1-gen-2020 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Galarini, Roberta; Bartolucci, Silvia; Piersanti, Giovanni
General synthesis of unnatural 4-, 5-, 6-, and 7-bromo-d-tryptophans by means of a regioselective indole alkylation 1-gen-2020 Bartoccini, Francesca; Fanini, Fabiola; Retini, Michele; Piersanti, Giovanni
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign 1-gen-2020 Linciano, Pasquale; Cullia, Gregorio; Borsari, Chiara; Santucci, Matteo; Ferrari, Stefania; Witt, Gesa; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Santarém, Nuno; Cordeiro da Silva, Anabela; Conti, Paola; Bolognesi, Maria Laura; Roberti, Marinella; Prati, Federica; Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni; Cavalli, Andrea; Goldoni, Luca; Bertozzi, Sine Mandrup; Bertozzi, Fabio; Brambilla, Enzo; Rizzo, Vincenzo; Piomelli, Daniele; Pinto, Andrea; Bandiera, Tiziano; Costi, Maria Paola
I-152, a supplier of N-acetyl-cysteine and cysteamine, inhibits immunoglobulin secretion and plasma cell maturation in LP-BM5 murine leukemia retrovirus-infected mice by affecting the unfolded protein response 1-gen-2020 Fraternale, Alessandra; Zara, Carolina; Di Mambro, Tomas; Manuali, Elisabetta; Genovese, Domenica Anna; Galluzzi, Luca; Diotallevi, Aurora; Pompa, Andrea; De Marchis, Francesca; Ambrogini, Patrizia; Cesarini, Erica; Luchetti, Francesca; Smietana, Michaël; Green, Kathy; Bartoccini, Francesca; Magnani, Mauro; Crinelli, Rita
Total Synthesis of (-)-Clavicipitic Acid via γ,γ-Dimethylallyltryptophan (DMAT) and Chemoselective C-H Hydroxylation 1-gen-2019 Bartoccini, Francesca; Venturi, Silvia; Retini, Michele; Mari, Michele; Piersanti, Giovanni
Large-Scale Preparation of N-Butanoyl-l-glutathione (C4-GSH) 1-gen-2019 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Fraternale, Alessandra; Piersanti, Giovanni
Mostrati risultati da 1 a 20 di 47
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