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Synthesis and Fluorescence Properties of 4-Cyano and 4-Formyl Melatonin as Putative Melatoninergic Ligands 1-gen-2023 Bartolucci, Silvia; Retini, Michele; Fanini, Fabiola; Paderni, Daniele; Piersanti, Giovanni
Asymmetric Alkylation of Cyclic Ketones with Dehydroalanine via H-Bond-Directing Enamine Catalysis: Straightforward Access to Enantiopure Unnatural α-Amino Acids 1-gen-2022 Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni
N-(Anilinoethyl)amide Melatonergic Ligands with Improved Water Solubility and Metabolic Stability 1-gen-2021 Ferlenghi, Francesca; Mari, Michele; Gobbi, Gabriella; Elisi, Gian Marco; Mor, Marco; Rivara, Silvia; Vacondio, Federica; Bartolucci, Silvia; Bedini, Annalida; Fanini, Fabiola; Spadoni, Gilberto
Single‐Step Synthesis of Dehydroalanine Derivatives via a Brønsted Acid‐Catalyzed Multicomponent Reaction 1-gen-2020 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Galarini, Roberta; Bartolucci, Silvia; Piersanti, Giovanni
Chiral Recognition of Flexible Melatonin Receptor Ligands Induced by Conformational Equilibria 1-gen-2020 Elisi, Gian Marco; Bedini, Annalida; Scalvini, Laura; Carmi, Caterina; Bartolucci, Silvia; Lucini, Valeria; Scaglione, Francesco; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
Design, synthesis and biological activity of hydrogen peroxide responsive arylboronate melatonin hybrids 1-gen-2019 Bedini, Annalida; Fraternale, Alessandra; Crinelli, Rita; Mari, Michele; Bartolucci, Silvia; Chiarantini, Laura; Spadoni, Gilberto
Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin 1-gen-2019 Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Mari, Michele; Piersanti, Giovanni
Divergent reactions of oxindoles with amino alcohols via the borrowing hydrogen process: oxindole ring opening vs. C3 alkylation 1-gen-2018 Di Gregorio, Giovanni; Mari, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni
Organocatalytic Aza-Friedel-Crafts/Lactonization Domino Reaction of Naphthols and Phenols with 2-Acetamidoacrylate to Naphtho- and Benzofuranones Bearing a Quaternary Center at the C3 Position 1-gen-2018 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Bartolucci, Silvia; Piersanti, Giovanni
Observations concerning the synthesis of tryptamine homologues and branched tryptamine derivatives via the borrowing hydrogen process: synthesis of psilocin, bufotenin, and serotonin 1-gen-2016 Bartolucci, Silvia; Mari, Michele; DI GREGORIO, Giovanni; Piersanti, Giovanni
A simple, modular synthesis of C4-substituted tryptophan derivatives 1-gen-2016 Bartoccini, Francesca; Bartolucci, Silvia; Mari, Michele; Piersanti, Giovanni
Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives 1-gen-2015 Bartoccini, Francesca; Bartolucci, Silvia; Lucarini, Simone; Piersanti, Giovanni
Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents 1-gen-2015 Bartolucci, Silvia; Mari, Michele; Bedini, Annalida; Piersanti, Giovanni; Spadoni, Gilberto
Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moieties 1-gen-2014 Spadoni, Gilberto; Bedini, Annalida; Bartolucci, Silvia; Pala, D.; Mor, M.; Riccioni, T.; Borsini, F.; Cabri, W.; Celona, D.; Marzi, M.; Tarzia, Giorgio; Rivara, S.; Minetti, P.
Synthesis and Characterization of New Bivalent Agents as Melatonin- and Histamine H3-Ligands 1-gen-2014 Pala, D.; Scalvini, L.; Lodola, A.; Mor, M.; Flammini, L.; Barocelli, E.; Lucini, V.; Scaglione, F.; Bartolucci, Silvia; Bedini, Annalida; Rivara, S.; Spadoni, Gilberto
Direct, Regioselective, and Chemoselective Preparation of Novel Boronated Tryptophans by Friedel–Crafts Alkylation 1-gen-2012 Bartolucci, Silvia; Bartoccini, Francesca; Righi, M.; Piersanti, Giovanni
Synthesis of Tryptamine Derivatives via a Direct, One-Pot Reductive Alkylation of Indoles 1-gen-2012 Marika, Righi; Francesca, Topi; Bartolucci, Silvia; Bedini, Annalida; Piersanti, Giovanni; Spadoni, Gilberto
Synthesis and Configuration Determination of All Enantiopure Stereoisomers of the Melatonin Receptor Ligand 4-Phenyl-2-propionamidotetralin using an Expedient Optical Resolution of 4-Phenyl-2-tetralone 1-gen-2012 Lucarini, Simone; Bartolucci, Silvia; Bedini, Annalida; Gatti, G.; Orlando, Pierfrancesco; Piersanti, Giovanni; Spadoni, Gilberto
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