Sfoglia per Autore
Large-Scale Preparation of N-Butanoyl-l-glutathione (C4-GSH)
2019 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Fraternale, Alessandra; Piersanti, Giovanni
Total Synthesis of (-)-Clavicipitic Acid via γ,γ-Dimethylallyltryptophan (DMAT) and Chemoselective C-H Hydroxylation
2019 Bartoccini, Francesca; Venturi, Silvia; Retini, Michele; Mari, Michele; Piersanti, Giovanni
Divergent reactions of oxindoles with amino alcohols via the borrowing hydrogen process: oxindole ring opening vs. C3 alkylation
2018 Di Gregorio, Giovanni; Mari, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni
Organocatalytic Aza-Friedel-Crafts/Lactonization Domino Reaction of Naphthols and Phenols with 2-Acetamidoacrylate to Naphtho- and Benzofuranones Bearing a Quaternary Center at the C3 Position
2018 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Bartolucci, Silvia; Piersanti, Giovanni
Iron-Catalyzed Direct C3-Benzylation of Indoles with Benzyl Alcohols through Borrowing Hydrogen
2017 DI GREGORIO, Giovanni; Mari, Michele; Bartoccini, Francesca; Piersanti, Giovanni
Metodo di sintesi di derivati del glutatione [Method for the synthesis of glutathione derivatives]
2017 Bartoccini, Francesca; Fraternale, Alessandra; Piersanti, Giovanni
Palladium(II)-Catalyzed Cross-Dehydrogenative Coupling (CDC) of N-Phthaloyl Dehydroalanine Esters with Simple Arenes: Stereoselective Synthesis of Z-Dehydrophenylalanine Derivatives
2016 Bartoccini, Francesca; Cannas, Diego Maria; Fini, Francesco; Piersanti, Giovanni
A simple, modular synthesis of C4-substituted tryptophan derivatives
2016 Bartoccini, Francesca; Bartolucci, Silvia; Mari, Michele; Piersanti, Giovanni
Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands
2015 Pace, Silvia; Brogin, Giandomenico; Stasi, Maria Antonietta; Riccioni, Teresa; Borsini, Franco; Capocasa, Francesca; Manera, Francesco; Tallarico, Carlo; Grossi, Pietro; Vacondio, Federica; Bassi, Michele; Bartoccini, Francesca; Lucarini, Simone; Piersanti, Giovanni; Tarzia, Giorgio; Cabri, Walter; Minetti, Patrizia
Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives
2015 Bartoccini, Francesca; Bartolucci, Silvia; Lucarini, Simone; Piersanti, Giovanni
Synthesis of (±)-cis-Clavicipitic Acid by a Rh(I)-Catalyzed Intramolecular Imine Reaction
2014 Bartoccini, Francesca; Mariangela, Casoli; Mari, Michele; Piersanti, Giovanni
Synthesis of 2-substituted tryptophans via a C3- to C2-alkyl migration
2014 Mari, Michele; Lucarini, Simone; Bartoccini, Francesca; Piersanti, Giovanni; Spadoni, Gilberto
Development of a practical and sustainable strategy for the synthesis of ST1535 by an iron-catalyzed Kumada cross-coupling reaction
2014 Bartoccini, Francesca; Piersanti, Giovanni; Silvia, Armaroli; Alberto, Cerri; Walter, Cabri
Synthesis of (−)-Epi-Indolactam V by an Intramolecular Buchwald–Hartwig C–N Coupling Cyclization Reaction
2013 Mari, Michele; Bartoccini, Francesca; Piersanti, Giovanni
Synthesis of (E)-8-(3-Chlorostyryl)caffeine Analogues Leading to 9-Deazaxanthine Derivatives as Dual A2AAntagonists/MAO-B Inhibitors
2013 Silvia, Rivara; Piersanti, Giovanni; Bartoccini, Francesca; Diamantini, Giuseppe; Daniele, Pala; Teresa, Riccioni; Maria Antonietta, Stasi; Walter, Cabri; Franco, Borsini; Marco, Mor; Tarzia, Giorgio; Patrizia, Minetti
Synthesis and Biological Evaluation of Metabolites of 2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), A Potent Antagonist of the A2AAdenosine Receptor for the Treatment of Parkinson’s Disease
2013 Piersanti, Giovanni; Bartoccini, Francesca; Lucarini, Simone; Walter, Cabri; Maria Antonietta, Stasi; Teresa, Riccioni; Franco, Borsini; Tarzia, Giorgio; Patrizia, Minetti
Direct, Regioselective, and Chemoselective Preparation of Novel Boronated Tryptophans by Friedel–Crafts Alkylation
2012 Bartolucci, Silvia; Bartoccini, Francesca; Righi, M.; Piersanti, Giovanni
Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions
2012 Bartoccini, Francesca; Piersanti, Giovanni; Marco, Mor; Tarzia, Giorgio; Patrizia, Minetti; Walter, Cabri
Organocatalytic synthesis of α-quaternary amino acid derivatives via aza-Friedel–Crafts alkylation of indoles with simple α-amidoacrylates
2011 Righi, M.; Bartoccini, Francesca; Lucarini, Simone; Piersanti, Giovanni
Direct B-alkyl Suzuki-Miyaura cross-coupling of 2-halopurines. Practical synthesis os ST1535, a potent adenosine A2A receptor antagonist
2010 Bartoccini, Francesca; Cabri, W; Celona, D; Minetti, P; Piersanti, Giovanni; G., Tarzia
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Large-Scale Preparation of N-Butanoyl-l-glutathione (C4-GSH) | 1-gen-2019 | Bartoccini, Francesca; Mari, Michele; Retini, Michele; Fraternale, Alessandra; Piersanti, Giovanni | |
Total Synthesis of (-)-Clavicipitic Acid via γ,γ-Dimethylallyltryptophan (DMAT) and Chemoselective C-H Hydroxylation | 1-gen-2019 | Bartoccini, Francesca; Venturi, Silvia; Retini, Michele; Mari, Michele; Piersanti, Giovanni | |
Divergent reactions of oxindoles with amino alcohols via the borrowing hydrogen process: oxindole ring opening vs. C3 alkylation | 1-gen-2018 | Di Gregorio, Giovanni; Mari, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni | |
Organocatalytic Aza-Friedel-Crafts/Lactonization Domino Reaction of Naphthols and Phenols with 2-Acetamidoacrylate to Naphtho- and Benzofuranones Bearing a Quaternary Center at the C3 Position | 1-gen-2018 | Bartoccini, Francesca; Mari, Michele; Retini, Michele; Bartolucci, Silvia; Piersanti, Giovanni | |
Iron-Catalyzed Direct C3-Benzylation of Indoles with Benzyl Alcohols through Borrowing Hydrogen | 1-gen-2017 | DI GREGORIO, Giovanni; Mari, Michele; Bartoccini, Francesca; Piersanti, Giovanni | |
Metodo di sintesi di derivati del glutatione [Method for the synthesis of glutathione derivatives] | 1-gen-2017 | Bartoccini, Francesca; Fraternale, Alessandra; Piersanti, Giovanni | |
Palladium(II)-Catalyzed Cross-Dehydrogenative Coupling (CDC) of N-Phthaloyl Dehydroalanine Esters with Simple Arenes: Stereoselective Synthesis of Z-Dehydrophenylalanine Derivatives | 1-gen-2016 | Bartoccini, Francesca; Cannas, Diego Maria; Fini, Francesco; Piersanti, Giovanni | |
A simple, modular synthesis of C4-substituted tryptophan derivatives | 1-gen-2016 | Bartoccini, Francesca; Bartolucci, Silvia; Mari, Michele; Piersanti, Giovanni | |
Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands | 1-gen-2015 | Pace, Silvia; Brogin, Giandomenico; Stasi, Maria Antonietta; Riccioni, Teresa; Borsini, Franco; Capocasa, Francesca; Manera, Francesco; Tallarico, Carlo; Grossi, Pietro; Vacondio, Federica; Bassi, Michele; Bartoccini, Francesca; Lucarini, Simone; Piersanti, Giovanni; Tarzia, Giorgio; Cabri, Walter; Minetti, Patrizia | |
Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives | 1-gen-2015 | Bartoccini, Francesca; Bartolucci, Silvia; Lucarini, Simone; Piersanti, Giovanni | |
Synthesis of (±)-cis-Clavicipitic Acid by a Rh(I)-Catalyzed Intramolecular Imine Reaction | 1-gen-2014 | Bartoccini, Francesca; Mariangela, Casoli; Mari, Michele; Piersanti, Giovanni | |
Synthesis of 2-substituted tryptophans via a C3- to C2-alkyl migration | 1-gen-2014 | Mari, Michele; Lucarini, Simone; Bartoccini, Francesca; Piersanti, Giovanni; Spadoni, Gilberto | |
Development of a practical and sustainable strategy for the synthesis of ST1535 by an iron-catalyzed Kumada cross-coupling reaction | 1-gen-2014 | Bartoccini, Francesca; Piersanti, Giovanni; Silvia, Armaroli; Alberto, Cerri; Walter, Cabri | |
Synthesis of (−)-Epi-Indolactam V by an Intramolecular Buchwald–Hartwig C–N Coupling Cyclization Reaction | 1-gen-2013 | Mari, Michele; Bartoccini, Francesca; Piersanti, Giovanni | |
Synthesis of (E)-8-(3-Chlorostyryl)caffeine Analogues Leading to 9-Deazaxanthine Derivatives as Dual A2AAntagonists/MAO-B Inhibitors | 1-gen-2013 | Silvia, Rivara; Piersanti, Giovanni; Bartoccini, Francesca; Diamantini, Giuseppe; Daniele, Pala; Teresa, Riccioni; Maria Antonietta, Stasi; Walter, Cabri; Franco, Borsini; Marco, Mor; Tarzia, Giorgio; Patrizia, Minetti | |
Synthesis and Biological Evaluation of Metabolites of 2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), A Potent Antagonist of the A2AAdenosine Receptor for the Treatment of Parkinson’s Disease | 1-gen-2013 | Piersanti, Giovanni; Bartoccini, Francesca; Lucarini, Simone; Walter, Cabri; Maria Antonietta, Stasi; Teresa, Riccioni; Franco, Borsini; Tarzia, Giorgio; Patrizia, Minetti | |
Direct, Regioselective, and Chemoselective Preparation of Novel Boronated Tryptophans by Friedel–Crafts Alkylation | 1-gen-2012 | Bartolucci, Silvia; Bartoccini, Francesca; Righi, M.; Piersanti, Giovanni | |
Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions | 1-gen-2012 | Bartoccini, Francesca; Piersanti, Giovanni; Marco, Mor; Tarzia, Giorgio; Patrizia, Minetti; Walter, Cabri | |
Organocatalytic synthesis of α-quaternary amino acid derivatives via aza-Friedel–Crafts alkylation of indoles with simple α-amidoacrylates | 1-gen-2011 | Righi, M.; Bartoccini, Francesca; Lucarini, Simone; Piersanti, Giovanni | |
Direct B-alkyl Suzuki-Miyaura cross-coupling of 2-halopurines. Practical synthesis os ST1535, a potent adenosine A2A receptor antagonist | 1-gen-2010 | Bartoccini, Francesca; Cabri, W; Celona, D; Minetti, P; Piersanti, Giovanni; G., Tarzia |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile