Sfoglia per Autore
Switchable reactivity of acylated alpha, beta-dehydroamino ester in the Friedel-Crafts alkylation of indoles by changing the Lewis acid.
2008 Angelini, E; Balsamini, Cesarino; Bartoccini, Francesca; Lucarini, Simone; Piersanti, Giovanni
Improved Synthesis of gamma-nitro-alfa-Amino ester and Acid Derivatives
2005 Ballini, R; Balsamini, Cesarino; Bartoccini, Francesca; Gianotti, M.; Martinelli, C.; Savoretti, N.
A Convenient and Easy Synthesis of γ-Nitro-α-Acetamido Esters
2005 Roberto, Ballini; Balsamini, Cesarino; Diamantini, Giuseppe; Nicoletta, Savoretti
Synthesis and biological evaluation of 6-bromo-6-substituted penicillanic acid derivatives as beta-lactamase inhibitors.
2002 Bedini, Annalida; Balsamini, Cesarino; DI GIACOMO, Barbara; Tontini, Andrea; Citterio, Barbara; Giorgi, Luca; DI MODUGNO, E.; Tarzia, Giorgio
Synthesis of new C-6 alkylidene penicillin derivatives as beta-lactamase inhibitors
2002 DI GIACOMO, Barbara; Tarzia, Giorgio; Bedini, Annalida; Gatti, G.; Bartoccini, Francesca; Balsamini, Cesarino; Tontini, Andrea; Baffone, Wally; DI MODUGNO, E.; Felici, A.
2-N-Acylaminoalkylindoles: Design and Quantitative Structure-Activity Relationship Studies Leading to MT2-Selective Antagonists.
2001 Spadoni, Gilberto; Balsamini, Cesarino; Diamantini, Giuseppe; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Rivara, S; Plazzi, P. V.; Nonno, R; Lucini, V; Pannacci, M; Fraschini, F; Stankov, Bm
A new melatonin receptor ligand with mt1-agonist and MT2-antagonist properties
2000 Nonno, R; Lucini, V; Spadoni, Gilberto; Pannacci, M; Croce, A; Esposti, D; Balsamini, Cesarino; Tarzia, Giorgio; Fraschini, F; Stankov, Bm
Synthesis of new 6-alkyliden penicillin derivatives as potential beta-lactamase inhibitors.
2000 DI GIACOMO, Barbara; Tarzia, Giorgio; Bedini, Annalida; Gatti, G; Balsamini, Cesarino; Baffone, Wally; Bartoccini, Francesca
Synthesis of new 6-bromopenicillanic acid derivatives as potential β-lactamase inhibitors.
2000 Bedini, Annalida; Tarzia, Giorgio; DI GIACOMO, Barbara; Gatti, G; Balsamini, Cesarino; Citterio, Barbara; Giorgi, Luca
3-(2-Carbamoylvinyl)-4,5-dimethylpyrrole-2-carboxylic acids as ligands at the NMDA glycine-binding site: a study on the 2-carbamoylvinyl chain modification
1999 Balsamini, Cesarino; Bedini, Annalida; Diamantini, Giuseppe; Spadoni, Gilberto; Tarzia, Giorgio; Tontini, Andrea; DI FABIO, R.; Donati, D.
(E)-3-(2-(N-phenylcarbamoyl)vinyl)pyrrole-2-carboxylic acid derivatives. A novel class of glycine site antagonists.
1998 Balsamini, Cesarino; Bedini, Annalida; Diamantini, Giuseppe; Spadoni, Gilberto; Tontini, Andrea; Tarzia, Giorgio; DI FABIO, R; Feriani, A; Reggiani, A; Tedesco, G; Valigi, R.
Melatonin receptor ligands: synthesis of new melatonin derivatives and comprehensive comparative molecular field analysis (CoMFA) study.
1998 Mor, M; Rivara, S; Silva, C; Bordi, F; Plazzi, P. V.; Spadoni, Gilberto; Diamantini, Giuseppe; Balsamini, Cesarino; Tarzia, Giorgio; Fraschini, F; Lucini, V; Nonno, R; Stankov, B. M.
1-Aminocylopropane-1-carboxylic acid derivatives as ligands at the glycine-binding site of the N-methyl-D-aspartate receptor
1998 Balsamini, C.; Bedini, A.; Spadoni, G.; Tarzia, G.; Tontini, A.; Balduini, W.; Cimino, M.
1-AMINOCYCLOPROPANE-1-CARBOXYLIC ACID DERIVATIVES AS LIGANDS AT THE GLYCINE-BINDING SITE OF THE N-METHYL-D-ASPARTATE RECEPTOR
1998 Balsamini, Cesarino; Bedini, Annalida; Spadoni, Gilberto; Tarzia, Giorgio; Tontini, Andrea; Balduini, Walter; Cimino, Mauro
2-[N-Acylamino(C1-C3)alkyl]indoles as MT1 melatonin receptor partial agonists, antagonists, and putative inverse agonists
1998 Spadoni, Gilberto; Balsamini, Cesarino; Bedini, Annalida; Diamantini, Giuseppe; DI GIACOMO, Barbara; Tontini, Andrea; Tarzia, Giorgio; Mor, M.; Plazzi, P. V.; Rivara, S.; Nonno, R.; Pannacci, M.; Lucini, V.; Fraschini, F.; Stankov, B. M.
An improved route to cycloalka[b]pyrrole 2-carboxylates
1997 Balsamini, Cesarino; Bedini, Annalida; Tarzia, Giorgio; Tontini, Andrea
1-Aminocyclopropane-1-carboxylic acid derivatives as ligands at the glicine-site of the NMDA receptor.
1997 Tarzia, Giorgio; Balsamini, Cesarino; Bedini, Annalida; Diamantini, Giuseppe; Tontini, Andrea; Cimino, Mauro; Balduini, Walter
Conformationally Restrained Melatonin Analogs: Synthesis, Binding Affinity for the Melatonin Receptor, Evaluation of the Biological Activity, and Molecular Modeling Study
1997 Spadoni, Gilberto; Balsamini, Cesarino; Diamantini, Giuseppe; DI GIACOMO, Barbara; Tarzia, Giorgio; Mor, Marco; PLAZZI PIER, Vincenzo; Rivara, Silvia; Lucini, Valeria; Nonno, Romolo; Pannacci, Marilou; Fraschini, Franco; STANKOV BOJIDAR, Michaylov
(E)-3-[2-(Carbamoylvinyl)]pyrrol-2-carboxylic acid derivatives: A novel Class of glycine site Antagonists.
1997 Balsamini, Cesarino; Bedini, Annalida; Diamantini, Giuseppe; Spadoni, Gilberto; Tontini, Andrea; Tarzia, Giorgio; DI FABIO, R.; Feriani, A.; Reggiani, A.; Tedesco, G.; Valigi, R.
Synthesis of 1-(isoxazol-3-yl)triazene derivatives. Antimetastatic activity of 3,3-dimethyl-1-(5-methylisoxazol-3-yl)triazene. European Journal of Medicinal Chemistry (1996), 31(9), 735-740.
1996 Tontini, Andrea; Diamantini, Giuseppe; Balsamini, Cesarino; Tarzia, Giorgio; Perissin, L.; Rapozzi, V.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Switchable reactivity of acylated alpha, beta-dehydroamino ester in the Friedel-Crafts alkylation of indoles by changing the Lewis acid. | 1-gen-2008 | Angelini, E; Balsamini, Cesarino; Bartoccini, Francesca; Lucarini, Simone; Piersanti, Giovanni | |
Improved Synthesis of gamma-nitro-alfa-Amino ester and Acid Derivatives | 1-gen-2005 | Ballini, R; Balsamini, Cesarino; Bartoccini, Francesca; Gianotti, M.; Martinelli, C.; Savoretti, N. | |
A Convenient and Easy Synthesis of γ-Nitro-α-Acetamido Esters | 1-gen-2005 | Roberto, Ballini; Balsamini, Cesarino; Diamantini, Giuseppe; Nicoletta, Savoretti | |
Synthesis and biological evaluation of 6-bromo-6-substituted penicillanic acid derivatives as beta-lactamase inhibitors. | 1-gen-2002 | Bedini, Annalida; Balsamini, Cesarino; DI GIACOMO, Barbara; Tontini, Andrea; Citterio, Barbara; Giorgi, Luca; DI MODUGNO, E.; Tarzia, Giorgio | |
Synthesis of new C-6 alkylidene penicillin derivatives as beta-lactamase inhibitors | 1-gen-2002 | DI GIACOMO, Barbara; Tarzia, Giorgio; Bedini, Annalida; Gatti, G.; Bartoccini, Francesca; Balsamini, Cesarino; Tontini, Andrea; Baffone, Wally; DI MODUGNO, E.; Felici, A. | |
2-N-Acylaminoalkylindoles: Design and Quantitative Structure-Activity Relationship Studies Leading to MT2-Selective Antagonists. | 1-gen-2001 | Spadoni, Gilberto; Balsamini, Cesarino; Diamantini, Giuseppe; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Rivara, S; Plazzi, P. V.; Nonno, R; Lucini, V; Pannacci, M; Fraschini, F; Stankov, Bm | |
A new melatonin receptor ligand with mt1-agonist and MT2-antagonist properties | 1-gen-2000 | Nonno, R; Lucini, V; Spadoni, Gilberto; Pannacci, M; Croce, A; Esposti, D; Balsamini, Cesarino; Tarzia, Giorgio; Fraschini, F; Stankov, Bm | |
Synthesis of new 6-alkyliden penicillin derivatives as potential beta-lactamase inhibitors. | 1-gen-2000 | DI GIACOMO, Barbara; Tarzia, Giorgio; Bedini, Annalida; Gatti, G; Balsamini, Cesarino; Baffone, Wally; Bartoccini, Francesca | |
Synthesis of new 6-bromopenicillanic acid derivatives as potential β-lactamase inhibitors. | 1-gen-2000 | Bedini, Annalida; Tarzia, Giorgio; DI GIACOMO, Barbara; Gatti, G; Balsamini, Cesarino; Citterio, Barbara; Giorgi, Luca | |
3-(2-Carbamoylvinyl)-4,5-dimethylpyrrole-2-carboxylic acids as ligands at the NMDA glycine-binding site: a study on the 2-carbamoylvinyl chain modification | 1-gen-1999 | Balsamini, Cesarino; Bedini, Annalida; Diamantini, Giuseppe; Spadoni, Gilberto; Tarzia, Giorgio; Tontini, Andrea; DI FABIO, R.; Donati, D. | |
(E)-3-(2-(N-phenylcarbamoyl)vinyl)pyrrole-2-carboxylic acid derivatives. A novel class of glycine site antagonists. | 1-gen-1998 | Balsamini, Cesarino; Bedini, Annalida; Diamantini, Giuseppe; Spadoni, Gilberto; Tontini, Andrea; Tarzia, Giorgio; DI FABIO, R; Feriani, A; Reggiani, A; Tedesco, G; Valigi, R. | |
Melatonin receptor ligands: synthesis of new melatonin derivatives and comprehensive comparative molecular field analysis (CoMFA) study. | 1-gen-1998 | Mor, M; Rivara, S; Silva, C; Bordi, F; Plazzi, P. V.; Spadoni, Gilberto; Diamantini, Giuseppe; Balsamini, Cesarino; Tarzia, Giorgio; Fraschini, F; Lucini, V; Nonno, R; Stankov, B. M. | |
1-Aminocylopropane-1-carboxylic acid derivatives as ligands at the glycine-binding site of the N-methyl-D-aspartate receptor | 1-gen-1998 | Balsamini, C.; Bedini, A.; Spadoni, G.; Tarzia, G.; Tontini, A.; Balduini, W.; Cimino, M. | |
1-AMINOCYCLOPROPANE-1-CARBOXYLIC ACID DERIVATIVES AS LIGANDS AT THE GLYCINE-BINDING SITE OF THE N-METHYL-D-ASPARTATE RECEPTOR | 1-gen-1998 | Balsamini, Cesarino; Bedini, Annalida; Spadoni, Gilberto; Tarzia, Giorgio; Tontini, Andrea; Balduini, Walter; Cimino, Mauro | |
2-[N-Acylamino(C1-C3)alkyl]indoles as MT1 melatonin receptor partial agonists, antagonists, and putative inverse agonists | 1-gen-1998 | Spadoni, Gilberto; Balsamini, Cesarino; Bedini, Annalida; Diamantini, Giuseppe; DI GIACOMO, Barbara; Tontini, Andrea; Tarzia, Giorgio; Mor, M.; Plazzi, P. V.; Rivara, S.; Nonno, R.; Pannacci, M.; Lucini, V.; Fraschini, F.; Stankov, B. M. | |
An improved route to cycloalka[b]pyrrole 2-carboxylates | 1-gen-1997 | Balsamini, Cesarino; Bedini, Annalida; Tarzia, Giorgio; Tontini, Andrea | |
1-Aminocyclopropane-1-carboxylic acid derivatives as ligands at the glicine-site of the NMDA receptor. | 1-gen-1997 | Tarzia, Giorgio; Balsamini, Cesarino; Bedini, Annalida; Diamantini, Giuseppe; Tontini, Andrea; Cimino, Mauro; Balduini, Walter | |
Conformationally Restrained Melatonin Analogs: Synthesis, Binding Affinity for the Melatonin Receptor, Evaluation of the Biological Activity, and Molecular Modeling Study | 1-gen-1997 | Spadoni, Gilberto; Balsamini, Cesarino; Diamantini, Giuseppe; DI GIACOMO, Barbara; Tarzia, Giorgio; Mor, Marco; PLAZZI PIER, Vincenzo; Rivara, Silvia; Lucini, Valeria; Nonno, Romolo; Pannacci, Marilou; Fraschini, Franco; STANKOV BOJIDAR, Michaylov | |
(E)-3-[2-(Carbamoylvinyl)]pyrrol-2-carboxylic acid derivatives: A novel Class of glycine site Antagonists. | 1-gen-1997 | Balsamini, Cesarino; Bedini, Annalida; Diamantini, Giuseppe; Spadoni, Gilberto; Tontini, Andrea; Tarzia, Giorgio; DI FABIO, R.; Feriani, A.; Reggiani, A.; Tedesco, G.; Valigi, R. | |
Synthesis of 1-(isoxazol-3-yl)triazene derivatives. Antimetastatic activity of 3,3-dimethyl-1-(5-methylisoxazol-3-yl)triazene. European Journal of Medicinal Chemistry (1996), 31(9), 735-740. | 1-gen-1996 | Tontini, Andrea; Diamantini, Giuseppe; Balsamini, Cesarino; Tarzia, Giorgio; Perissin, L.; Rapozzi, V. |
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