Sfoglia per Autore
Asymmetric Synthesis and Biological Evaluation of Both Enantiomers of 5- and 6-Boronotryptophan as Potential Boron Delivery Agents for Boron Neutron Capture Therapy
2024 Retini, Michele; Järvinen, Juulia; Bahrami, Katayun; Tampio, Janne; Bartoccini, Francesca; Riihelä, Petri; Pehkonen, Henna; Värä, Arina; Laitinen, Tuomo; Huttunen, Kristiina M.; Rautio, Jarkko; Piersanti, Giovanni; Timonen, Juri M.
Practical and Selective Syntheses of S‐Acyl and N‐Acyl Glutathiones with N‐Acyl Imidazoles in Water
2024 Retini, Michele; Sisti, Andrea; Olivieri, Diego; Mari, Michele; Bartoccini, Francesca; Piersanti, Giovanni
Binding and unbinding of potent melatonin receptor ligands: Mechanistic simulations and experimental evidence
2024 Bedini, Annalida; Elisi, Gian Marco; Fanini, Fabiola; Retini, Michele; Scalvini, Laura; Pasquini, Silvia; Contri, Chiara; Varani, Katia; Spadoni, Gilberto; Mor, Marco; Vincenzi, Fabrizio; Rivara, Silvia
Inhibition of myeloid-derived suppressor cell (MDSC) activity by redox-modulating agents restores T and B cell proliferative responses in murine AIDS
2023 Fraternale, Alessandra; Green, Kathy A.; Schiavano, Giuditta F.; Bruschi, Michela; Retini, Michele; Magnani, Mauro; Green, William R.
Targeting SARS-CoV-2 by synthetic dual-acting thiol compounds that inhibit Spike/ACE2 interaction and viral protein production
2023 Fraternale, Alessandra; De Angelis, Marta; De Santis, Riccardo; Amatore, Donatella; Masini, Sofia; Monittola, Francesca; Menotta, Michele; Biancucci, Federica; Bartoccini, Francesca; Retini, Michele; Fiori, Valentina; Fioravanti, Raoul; Magurano, Fabio; Chiarantini, Laura; Lista, Romano F; Piersanti, Giovanni; Palamara, Anna T; Nencioni, Lucia; Magnani, Mauro; Crinelli, Rita
Synthesis and Fluorescence Properties of 4-Cyano and 4-Formyl Melatonin as Putative Melatoninergic Ligands
2023 Bartolucci, Silvia; Retini, Michele; Fanini, Fabiola; Paderni, Daniele; Piersanti, Giovanni
Paradigm Shift in Gastric Cancer Prevention: Harnessing the Potential of Aristolochia olivieri Extract
2023 Micucci, Matteo; Stella Bartoletti, Anna; Abdullah, Fuad O; Burattini, Sabrina; Versari, Ilaria; Canale, Matteo; D'Agostino, Federico; Roncarati, Davide; Piatti, Diletta; Sagratini, Gianni; Caprioli, Giovanni; Mari, Michele; Retini, Michele; Faenza, Irene; Battistelli, Michela; Salucci, Sara
A potential host and virus targeting tool against COVID-19: Chemical characterization, antiviral, cytoprotective, antioxidant, respiratory smooth muscle relaxant effects of Paulownia tomentosa Steud
2023 Magurano, Fabio; Micucci, Matteo; Nuzzo, Domenico; Baggieri, Melissa; Picone, Pasquale; Gioacchini, Silvia; Fioravanti, Raoul; Bucci, Paola; Kojouri, Maedeh; Mari, Michele; Retini, Michele; Budriesi, Roberta; Mattioli, Laura Beatrice; Corazza, Ivan; Di Liberto, Valentina; Todaro, Luigi; Giuseppetti, Roberto; D'Ugo, Emilio; Marchi, Antonella; Mecca, Marisabel; D'Auria, Maurizio
Dithiol Based on L-Cysteine and Cysteamine as a Disulfide-Reducing Agent
2022 Bartoccini, Francesca; Retini, Michele; Crinelli, Rita; Menotta, Michele; Fraternale, Alessandra; Piersanti, Giovanni
Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties
2022 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Asymmetric Alkylation of Cyclic Ketones with Dehydroalanine via H-Bond-Directing Enamine Catalysis: Straightforward Access to Enantiopure Unnatural α-Amino Acids
2022 Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors
2022 Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
Intracellular Redox-Modulated Pathways as Targets for Effective Approaches in the Treatment of Viral Infection
2021 Fraternale, Alessandra; Zara, Carolina; De Angelis, Marta; Nencioni, Lucia; Palamara, Anna Teresa; Retini, Michele; Di Mambro, Tomas; Magnani, Mauro; Crinelli, Rita
Novel, Chiral, and Enantiopure C2‐Symmetric Thioureas Promote Asymmetric Protio‐Pictet‐Spengler Reactions by Anion‐Binding Catalysis
2021 Retini, Michele; Bartoccini, Francesca; Zappia, Giovanni; Piersanti, Giovanni
Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma
2021 Castelli, Riccardo; Taranto, Sara; Furiassi, Lucia; Bozza, Nicole; Marseglia, Giuseppe; Ferlenghi, Francesca; Rivara, Silvia; Retini, Michele; Bedini, Annalida; Spadoni, Gilberto; Matarazzo, Sara; Ronca, Roberto; Presta, Marco; Mor, Marco; Giacomini, Arianna
Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone
2021 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign
2020 Linciano, Pasquale; Cullia, Gregorio; Borsari, Chiara; Santucci, Matteo; Ferrari, Stefania; Witt, Gesa; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Santarém, Nuno; Cordeiro da Silva, Anabela; Conti, Paola; Bolognesi, Maria Laura; Roberti, Marinella; Prati, Federica; Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni; Cavalli, Andrea; Goldoni, Luca; Bertozzi, Sine Mandrup; Bertozzi, Fabio; Brambilla, Enzo; Rizzo, Vincenzo; Piomelli, Daniele; Pinto, Andrea; Bandiera, Tiziano; Costi, Maria Paola
Single‐Step Synthesis of Dehydroalanine Derivatives via a Brønsted Acid‐Catalyzed Multicomponent Reaction
2020 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Galarini, Roberta; Bartolucci, Silvia; Piersanti, Giovanni
General synthesis of unnatural 4-, 5-, 6-, and 7-bromo-d-tryptophans by means of a regioselective indole alkylation
2020 Bartoccini, Francesca; Fanini, Fabiola; Retini, Michele; Piersanti, Giovanni
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology
2020 Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Asymmetric Synthesis and Biological Evaluation of Both Enantiomers of 5- and 6-Boronotryptophan as Potential Boron Delivery Agents for Boron Neutron Capture Therapy | 1-gen-2024 | Retini, Michele; Järvinen, Juulia; Bahrami, Katayun; Tampio, Janne; Bartoccini, Francesca; Riihelä, Petri; Pehkonen, Henna; Värä, Arina; Laitinen, Tuomo; Huttunen, Kristiina M.; Rautio, Jarkko; Piersanti, Giovanni; Timonen, Juri M. | |
Practical and Selective Syntheses of S‐Acyl and N‐Acyl Glutathiones with N‐Acyl Imidazoles in Water | 1-gen-2024 | Retini, Michele; Sisti, Andrea; Olivieri, Diego; Mari, Michele; Bartoccini, Francesca; Piersanti, Giovanni | |
Binding and unbinding of potent melatonin receptor ligands: Mechanistic simulations and experimental evidence | 1-gen-2024 | Bedini, Annalida; Elisi, Gian Marco; Fanini, Fabiola; Retini, Michele; Scalvini, Laura; Pasquini, Silvia; Contri, Chiara; Varani, Katia; Spadoni, Gilberto; Mor, Marco; Vincenzi, Fabrizio; Rivara, Silvia | |
Inhibition of myeloid-derived suppressor cell (MDSC) activity by redox-modulating agents restores T and B cell proliferative responses in murine AIDS | 1-gen-2023 | Fraternale, Alessandra; Green, Kathy A.; Schiavano, Giuditta F.; Bruschi, Michela; Retini, Michele; Magnani, Mauro; Green, William R. | |
Targeting SARS-CoV-2 by synthetic dual-acting thiol compounds that inhibit Spike/ACE2 interaction and viral protein production | 1-gen-2023 | Fraternale, Alessandra; De Angelis, Marta; De Santis, Riccardo; Amatore, Donatella; Masini, Sofia; Monittola, Francesca; Menotta, Michele; Biancucci, Federica; Bartoccini, Francesca; Retini, Michele; Fiori, Valentina; Fioravanti, Raoul; Magurano, Fabio; Chiarantini, Laura; Lista, Romano F; Piersanti, Giovanni; Palamara, Anna T; Nencioni, Lucia; Magnani, Mauro; Crinelli, Rita | |
Synthesis and Fluorescence Properties of 4-Cyano and 4-Formyl Melatonin as Putative Melatoninergic Ligands | 1-gen-2023 | Bartolucci, Silvia; Retini, Michele; Fanini, Fabiola; Paderni, Daniele; Piersanti, Giovanni | |
Paradigm Shift in Gastric Cancer Prevention: Harnessing the Potential of Aristolochia olivieri Extract | 1-gen-2023 | Micucci, Matteo; Stella Bartoletti, Anna; Abdullah, Fuad O; Burattini, Sabrina; Versari, Ilaria; Canale, Matteo; D'Agostino, Federico; Roncarati, Davide; Piatti, Diletta; Sagratini, Gianni; Caprioli, Giovanni; Mari, Michele; Retini, Michele; Faenza, Irene; Battistelli, Michela; Salucci, Sara | |
A potential host and virus targeting tool against COVID-19: Chemical characterization, antiviral, cytoprotective, antioxidant, respiratory smooth muscle relaxant effects of Paulownia tomentosa Steud | 1-gen-2023 | Magurano, Fabio; Micucci, Matteo; Nuzzo, Domenico; Baggieri, Melissa; Picone, Pasquale; Gioacchini, Silvia; Fioravanti, Raoul; Bucci, Paola; Kojouri, Maedeh; Mari, Michele; Retini, Michele; Budriesi, Roberta; Mattioli, Laura Beatrice; Corazza, Ivan; Di Liberto, Valentina; Todaro, Luigi; Giuseppetti, Roberto; D'Ugo, Emilio; Marchi, Antonella; Mecca, Marisabel; D'Auria, Maurizio | |
Dithiol Based on L-Cysteine and Cysteamine as a Disulfide-Reducing Agent | 1-gen-2022 | Bartoccini, Francesca; Retini, Michele; Crinelli, Rita; Menotta, Michele; Fraternale, Alessandra; Piersanti, Giovanni | |
Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties | 1-gen-2022 | Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni | |
Asymmetric Alkylation of Cyclic Ketones with Dehydroalanine via H-Bond-Directing Enamine Catalysis: Straightforward Access to Enantiopure Unnatural α-Amino Acids | 1-gen-2022 | Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni | |
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors | 1-gen-2022 | Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto | |
Intracellular Redox-Modulated Pathways as Targets for Effective Approaches in the Treatment of Viral Infection | 1-gen-2021 | Fraternale, Alessandra; Zara, Carolina; De Angelis, Marta; Nencioni, Lucia; Palamara, Anna Teresa; Retini, Michele; Di Mambro, Tomas; Magnani, Mauro; Crinelli, Rita | |
Novel, Chiral, and Enantiopure C2‐Symmetric Thioureas Promote Asymmetric Protio‐Pictet‐Spengler Reactions by Anion‐Binding Catalysis | 1-gen-2021 | Retini, Michele; Bartoccini, Francesca; Zappia, Giovanni; Piersanti, Giovanni | |
Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma | 1-gen-2021 | Castelli, Riccardo; Taranto, Sara; Furiassi, Lucia; Bozza, Nicole; Marseglia, Giuseppe; Ferlenghi, Francesca; Rivara, Silvia; Retini, Michele; Bedini, Annalida; Spadoni, Gilberto; Matarazzo, Sara; Ronca, Roberto; Presta, Marco; Mor, Marco; Giacomini, Arianna | |
Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone | 1-gen-2021 | Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni | |
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign | 1-gen-2020 | Linciano, Pasquale; Cullia, Gregorio; Borsari, Chiara; Santucci, Matteo; Ferrari, Stefania; Witt, Gesa; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Santarém, Nuno; Cordeiro da Silva, Anabela; Conti, Paola; Bolognesi, Maria Laura; Roberti, Marinella; Prati, Federica; Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni; Cavalli, Andrea; Goldoni, Luca; Bertozzi, Sine Mandrup; Bertozzi, Fabio; Brambilla, Enzo; Rizzo, Vincenzo; Piomelli, Daniele; Pinto, Andrea; Bandiera, Tiziano; Costi, Maria Paola | |
Single‐Step Synthesis of Dehydroalanine Derivatives via a Brønsted Acid‐Catalyzed Multicomponent Reaction | 1-gen-2020 | Bartoccini, Francesca; Mari, Michele; Retini, Michele; Galarini, Roberta; Bartolucci, Silvia; Piersanti, Giovanni | |
General synthesis of unnatural 4-, 5-, 6-, and 7-bromo-d-tryptophans by means of a regioselective indole alkylation | 1-gen-2020 | Bartoccini, Francesca; Fanini, Fabiola; Retini, Michele; Piersanti, Giovanni | |
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology | 1-gen-2020 | Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni |
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