PIERSANTI, GIOVANNI
PIERSANTI, GIOVANNI
Dipartimento di Scienze Biomolecolari (DISB)
2-n-Butyl- 9-methyl-8-(1,2,3)triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological Characterization
2005-01-01 Minetti, P; TINTI M., O; Carminati, P; Castorina, M; DI CESARE M., A; DI SERIO, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, Luca; Piersanti, Giovanni; Bartoccini, Francesca; Tarzia, Giorgio
2-n-butyl-9-methyl-8-(1,2,3)triazol-2yl-9H-purin-6-yl-amine (ST 1535) and analogs as A2a Adenosine receptor antagonists. Design, synthesis and pharmacological characterization
2003-01-01 Bartoccini, Francesca; Castorina, M.; DI CESARE, M. A.; Gallo, G; Ghirardi, O.; Giorgi, F. GIORGI L.; Minetti, P.; Piersanti, Giovanni; Tarzia, Giorgio; Tinti, M. O.
5-(2-Ethyl-phenyl)-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole (DL-111-IT ) and related compounds induce morphological apoptotic patterns in cultures of human tumor cell lines
2003-01-01 Burattini, Sabrina; Luchetti, Francesca; Battistelli, Michela; DELLA FELICE, Massimo; Papa, Stefano; Piersanti, Giovanni; Tarzia, Giorgio; Falcieri, Elisabetta
A Versatile Biomimetic Approach to Diindolylmethane Derivatives as Potential Anticancer Agents
2012-01-01 Lucarini, Simone; Piersanti, Giovanni; Duranti, Andrea; Spadoni, Gilberto
An efficient, economical synthesis of hydroxytyrosol and its protected forms via Baeyer–Villiger oxidation
2011-01-01 Piersanti, Giovanni; Retini, M; ESPARTERO J., L; Madrona, A; Zappia, Giovanni
Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties
2022-01-01 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Brønsted Acid-Catalyzed Bisindolization of α-amido acetals: Synthesis and Anticancer activity of bis(indolyl)ethanamino derivatives
2014-01-01 Mari, Michele; Aurora, Tassoni; Lucarini, Simone; Fanelli, Mirco; Piersanti, Giovanni; Spadoni, Gilberto
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology
2020-01-01 Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni
The collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity
2009-01-01 Valitutti, G; Duranti, Andrea; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P.
Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin
2019-01-01 Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Mari, Michele; Piersanti, Giovanni
Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone
2021-01-01 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Conformation by NMR of two tetralin-based receptor ligands
2003-01-01 Gatti, G.; Piersanti, Giovanni; Spadoni, Gilberto
Correlation between energetics of collisionally activated decompositions, interaction energy and biological potency of carbamates FAAH inhibitors
2007-01-01 Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P.
Cyclohexylcarbamic Acid 3’-or 4’-Substituted Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: Synthesis Quantitative Structure–Activity Relationships, and Molecular Modeling Studies
2004-01-01 Mor, M; Rivara, S; Lodola, A; Plazzi, Pv; Tarzia, Giorgio; Duranti, Andrea; Tontini, Andrea; Piersanti, Giovanni; Kathuria, S; Piomelli, D.
Derivatives of triazoly-imidazopyridine useful as ligands of the adenosine A2a receptor ant their use as medicaments
2009-01-01 Tarzia, Giorgio; Piersanti, Giovanni; Giorgi, Luca; Patrizia, Minetti; MARIA A., DI CESARE; Grazia, Gallo; Fabrizio, Giorgi
DERIVATIVES OF TRIAZOLYL-IMIDAZOPYRIDINE AND OF THE TRIAZOLYLPURINES USEFUL AS LIGANDS OF THE ADENOSINE A2a RECEPTOR AND THEIR USE AS MEDICAMENTS.
2003-01-01 Tarzia, Giorgio; Piersanti, Giovanni; P., Minetti; A., DI CESARE; G., Gallo; F., Giorgi; Giorgi, Luca
Derivatizzazione one-pot di indoli per la sintesi di triptofani, pirroloindoline, bis-indoli & co
2014-01-01 Lucarini, Simone; Piersanti, Giovanni; Duranti, Andrea; Spadoni, Gilberto
Design, SAR and Biological Activity of a New Class of FAAH Inhibitors: Cyclohexyl Carbamic Acid Biphenyl-3-yl Esters
2003-01-01 Mor, M; Duranti, Andrea; Tontini, Andrea; Piersanti, Giovanni; Tarzia, Giorgio; Rivara, S; Lodola, A; Plazzi, Pv; Calignano, A; Cuomo, V; Kathuria, S; Piomelli, D.
Design, Synthesis and SAR of Alkylcarbamic Acid Aryl Esters, a New Class of Fatty Acids Amide Hydrolase Inhibitors
2003-01-01 Tarzia, Giorgio; Mor, M; Duranti, Andrea; Tontini, Andrea; Piersanti, Giovanni; Piomelli, D.
Design, Synthesis and Structure–Activity Relationships of Alkylcarbamic Acid Aryl Esters, a New Class of Fatty Acid Amide Hydrolase Inhibitors
2003-01-01 Tarzia, Giorgio; Duranti, Andrea; Tontini, Andrea; Piersanti, Giovanni; Mor, M; Rivara, S; Plazzi, Pv; Park, C; Kathuria, S; Piomelli, D.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
2-n-Butyl- 9-methyl-8-(1,2,3)triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological Characterization | 1-gen-2005 | Minetti, P; TINTI M., O; Carminati, P; Castorina, M; DI CESARE M., A; DI SERIO, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, Luca; Piersanti, Giovanni; Bartoccini, Francesca; Tarzia, Giorgio | |
2-n-butyl-9-methyl-8-(1,2,3)triazol-2yl-9H-purin-6-yl-amine (ST 1535) and analogs as A2a Adenosine receptor antagonists. Design, synthesis and pharmacological characterization | 1-gen-2003 | Bartoccini, Francesca; Castorina, M.; DI CESARE, M. A.; Gallo, G; Ghirardi, O.; Giorgi, F. GIORGI L.; Minetti, P.; Piersanti, Giovanni; Tarzia, Giorgio; Tinti, M. O. | |
5-(2-Ethyl-phenyl)-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole (DL-111-IT ) and related compounds induce morphological apoptotic patterns in cultures of human tumor cell lines | 1-gen-2003 | Burattini, Sabrina; Luchetti, Francesca; Battistelli, Michela; DELLA FELICE, Massimo; Papa, Stefano; Piersanti, Giovanni; Tarzia, Giorgio; Falcieri, Elisabetta | |
A Versatile Biomimetic Approach to Diindolylmethane Derivatives as Potential Anticancer Agents | 1-gen-2012 | Lucarini, Simone; Piersanti, Giovanni; Duranti, Andrea; Spadoni, Gilberto | |
An efficient, economical synthesis of hydroxytyrosol and its protected forms via Baeyer–Villiger oxidation | 1-gen-2011 | Piersanti, Giovanni; Retini, M; ESPARTERO J., L; Madrona, A; Zappia, Giovanni | |
Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties | 1-gen-2022 | Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni | |
Brønsted Acid-Catalyzed Bisindolization of α-amido acetals: Synthesis and Anticancer activity of bis(indolyl)ethanamino derivatives | 1-gen-2014 | Mari, Michele; Aurora, Tassoni; Lucarini, Simone; Fanelli, Mirco; Piersanti, Giovanni; Spadoni, Gilberto | |
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology | 1-gen-2020 | Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni | |
The collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity | 1-gen-2009 | Valitutti, G; Duranti, Andrea; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P. | |
Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin | 1-gen-2019 | Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Mari, Michele; Piersanti, Giovanni | |
Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone | 1-gen-2021 | Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni | |
Conformation by NMR of two tetralin-based receptor ligands | 1-gen-2003 | Gatti, G.; Piersanti, Giovanni; Spadoni, Gilberto | |
Correlation between energetics of collisionally activated decompositions, interaction energy and biological potency of carbamates FAAH inhibitors | 1-gen-2007 | Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P. | |
Cyclohexylcarbamic Acid 3’-or 4’-Substituted Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: Synthesis Quantitative Structure–Activity Relationships, and Molecular Modeling Studies | 1-gen-2004 | Mor, M; Rivara, S; Lodola, A; Plazzi, Pv; Tarzia, Giorgio; Duranti, Andrea; Tontini, Andrea; Piersanti, Giovanni; Kathuria, S; Piomelli, D. | |
Derivatives of triazoly-imidazopyridine useful as ligands of the adenosine A2a receptor ant their use as medicaments | 1-gen-2009 | Tarzia, Giorgio; Piersanti, Giovanni; Giorgi, Luca; Patrizia, Minetti; MARIA A., DI CESARE; Grazia, Gallo; Fabrizio, Giorgi | |
DERIVATIVES OF TRIAZOLYL-IMIDAZOPYRIDINE AND OF THE TRIAZOLYLPURINES USEFUL AS LIGANDS OF THE ADENOSINE A2a RECEPTOR AND THEIR USE AS MEDICAMENTS. | 1-gen-2003 | Tarzia, Giorgio; Piersanti, Giovanni; P., Minetti; A., DI CESARE; G., Gallo; F., Giorgi; Giorgi, Luca | |
Derivatizzazione one-pot di indoli per la sintesi di triptofani, pirroloindoline, bis-indoli & co | 1-gen-2014 | Lucarini, Simone; Piersanti, Giovanni; Duranti, Andrea; Spadoni, Gilberto | |
Design, SAR and Biological Activity of a New Class of FAAH Inhibitors: Cyclohexyl Carbamic Acid Biphenyl-3-yl Esters | 1-gen-2003 | Mor, M; Duranti, Andrea; Tontini, Andrea; Piersanti, Giovanni; Tarzia, Giorgio; Rivara, S; Lodola, A; Plazzi, Pv; Calignano, A; Cuomo, V; Kathuria, S; Piomelli, D. | |
Design, Synthesis and SAR of Alkylcarbamic Acid Aryl Esters, a New Class of Fatty Acids Amide Hydrolase Inhibitors | 1-gen-2003 | Tarzia, Giorgio; Mor, M; Duranti, Andrea; Tontini, Andrea; Piersanti, Giovanni; Piomelli, D. | |
Design, Synthesis and Structure–Activity Relationships of Alkylcarbamic Acid Aryl Esters, a New Class of Fatty Acid Amide Hydrolase Inhibitors | 1-gen-2003 | Tarzia, Giorgio; Duranti, Andrea; Tontini, Andrea; Piersanti, Giovanni; Mor, M; Rivara, S; Plazzi, Pv; Park, C; Kathuria, S; Piomelli, D. |