PIERSANTI, GIOVANNI

PIERSANTI, GIOVANNI  

Dipartimento di Scienze Biomolecolari (DISB)  

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Risultati 1 - 20 di 102 (tempo di esecuzione: 0.023 secondi).
Titolo Data di pubblicazione Autore(i) File
2-n-Butyl- 9-methyl-8-(1,2,3)triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological Characterization 1-gen-2005 Minetti, P; Tinti, M. O.; Carminati, P; Castorina, M; DI CESARE, M. A.; DI SERIO, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, Luca; Piersanti, Giovanni; Bartoccini, Francesca; Tarzia, Giorgio
2-n-butyl-9-methyl-8-(1,2,3)triazol-2yl-9H-purin-6-yl-amine (ST 1535) and analogs as A2a Adenosine receptor antagonists. Design, synthesis and pharmacological characterization 1-gen-2003 Bartoccini, Francesca; Castorina, M.; DI CESARE, M. A.; Gallo, G; Ghirardi, O.; Giorgi, F. GIORGI L.; Minetti, P.; Piersanti, Giovanni; Tarzia, Giorgio; Tinti, M. O.
5-(2-Ethyl-phenyl)-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole (DL-111-IT ) and related compounds induce morphological apoptotic patterns in cultures of human tumor cell lines 1-gen-2003 Burattini, Sabrina; Luchetti, Francesca; Battistelli, Michela; DELLA FELICE, Massimo; Papa, Stefano; Piersanti, Giovanni; Tarzia, Giorgio; Falcieri, Elisabetta
A Novel One-Pot Approach of Hexahydropyrrolo[2,3-b]indole Nucleus by a cascade addition/cyclization strategy: Synthesis of (±)-Esermethole 1-gen-2010 Lucarini, Simone; Bartoccini, Francesca; Battistoni, F; Diamantini, Giuseppe; Piersanti, Giovanni; Righi, M; Spadoni, Gilberto
A Short Synthesis of (−)‐6,7‐Secoagroclavine via Metal‐Free Reductive Coupling 1-gen-2024 Diotallevi, Francesca; Bartoccini, Francesca; Piersanti, Giovanni
A simple, modular synthesis of C4-substituted tryptophan derivatives 1-gen-2016 Bartoccini, Francesca; Bartolucci, Silvia; Mari, Michele; Piersanti, Giovanni
A Trans-Stereoselective Synthesis of 3-Halo-4-alkyl(aryl)-NH-azetidin-2-ones. 1-gen-2000 Bandini, Elisa; Favi, Gianfranco; Martelli, Giorgio; Panunzio, Mauro; Piersanti, Giovanni
A Versatile Biomimetic Approach to Diindolylmethane Derivatives as Potential Anticancer Agents 1-gen-2012 Lucarini, Simone; Piersanti, Giovanni; Duranti, Andrea; Spadoni, Gilberto
An efficient synthesis of the cyclic form of scalemic 2,4-di-epi-polyoxamic acid exploiting the hetero Diels-Alder approach. 1-gen-1997 Bandini, Elisa; Martelli, Giorgio; Spunta, Giuseppe; Bongini, Alessandro; Panunzio, Mauro; Piersanti, Giovanni
An efficient, economical synthesis of hydroxytyrosol and its protected forms via Baeyer–Villiger oxidation 1-gen-2011 Piersanti, G; Retini, M; Espartero, J; Madrona, A; Zappia, G
An improved synthesis of cis-4-phenyl-2-propionamidotetralin (4-P-PDOT): a selective MT2 melatonin receptor antagonist. 1-gen-2008 Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto; Piersanti, Giovanni
Asymmetric Alkylation of Cyclic Ketones with Dehydroalanine via H-Bond-Directing Enamine Catalysis: Straightforward Access to Enantiopure Unnatural α-Amino Acids 1-gen-2022 Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni
Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties 1-gen-2022 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Brønsted Acid-Catalyzed Bisindolization of α-amido acetals: Synthesis and Anticancer activity of bis(indolyl)ethanamino derivatives 1-gen-2014 Mari, Michele; Aurora, Tassoni; Lucarini, Simone; Fanelli, Mirco; Piersanti, Giovanni; Spadoni, Gilberto
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology 1-gen-2020 Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni
Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin 1-gen-2019 Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Mari, Michele; Piersanti, Giovanni
Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone 1-gen-2021 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Conformation by NMR of two tetralin-based receptor ligands 1-gen-2003 Gatti, G.; Piersanti, Giovanni; Spadoni, Gilberto
Correlation between energetics of collisionally activated decompositions, interaction energy and biological potency of carbamates FAAH inhibitors 1-gen-2007 Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P.
Cyclohexylcarbamic Acid 3’-or 4’-Substituted Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: Synthesis Quantitative Structure–Activity Relationships, and Molecular Modeling Studies 1-gen-2004 Mor, M; Rivara, S; Lodola, A; Plazzi, Pv; Tarzia, Giorgio; Duranti, Andrea; Tontini, Andrea; Piersanti, Giovanni; Kathuria, S; Piomelli, D.