PIERSANTI, GIOVANNI
PIERSANTI, GIOVANNI
Dipartimento di Scienze Biomolecolari (DISB)
2-n-Butyl- 9-methyl-8-(1,2,3)triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological Characterization
2005 Minetti, P; Tinti, M. O.; Carminati, P; Castorina, M; DI CESARE, M. A.; DI SERIO, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, Luca; Piersanti, Giovanni; Bartoccini, Francesca; Tarzia, Giorgio
2-n-butyl-9-methyl-8-(1,2,3)triazol-2yl-9H-purin-6-yl-amine (ST 1535) and analogs as A2a Adenosine receptor antagonists. Design, synthesis and pharmacological characterization
2003 Bartoccini, Francesca; Castorina, M.; DI CESARE, M. A.; Gallo, G; Ghirardi, O.; Giorgi, F. GIORGI L.; Minetti, P.; Piersanti, Giovanni; Tarzia, Giorgio; Tinti, M. O.
5-(2-Ethyl-phenyl)-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole (DL-111-IT ) and related compounds induce morphological apoptotic patterns in cultures of human tumor cell lines
2003 Burattini, Sabrina; Luchetti, Francesca; Battistelli, Michela; DELLA FELICE, Massimo; Papa, Stefano; Piersanti, Giovanni; Tarzia, Giorgio; Falcieri, Elisabetta
A Novel One-Pot Approach of Hexahydropyrrolo[2,3-b]indole Nucleus by a cascade addition/cyclization strategy: Synthesis of (±)-Esermethole
2010 Lucarini, Simone; Bartoccini, Francesca; Battistoni, F; Diamantini, Giuseppe; Piersanti, Giovanni; Righi, M; Spadoni, Gilberto
A Short Synthesis of (−)‐6,7‐Secoagroclavine via Metal‐Free Reductive Coupling
2024 Diotallevi, Francesca; Bartoccini, Francesca; Piersanti, Giovanni
A simple, modular synthesis of C4-substituted tryptophan derivatives
2016 Bartoccini, Francesca; Bartolucci, Silvia; Mari, Michele; Piersanti, Giovanni
A Trans-Stereoselective Synthesis of 3-Halo-4-alkyl(aryl)-NH-azetidin-2-ones.
2000 Bandini, Elisa; Favi, Gianfranco; Martelli, Giorgio; Panunzio, Mauro; Piersanti, Giovanni
A Versatile Biomimetic Approach to Diindolylmethane Derivatives as Potential Anticancer Agents
2012 Lucarini, Simone; Piersanti, Giovanni; Duranti, Andrea; Spadoni, Gilberto
An efficient synthesis of the cyclic form of scalemic 2,4-di-epi-polyoxamic acid exploiting the hetero Diels-Alder approach.
1997 Bandini, Elisa; Martelli, Giorgio; Spunta, Giuseppe; Bongini, Alessandro; Panunzio, Mauro; Piersanti, Giovanni
An efficient, economical synthesis of hydroxytyrosol and its protected forms via Baeyer–Villiger oxidation
2011 Piersanti, G; Retini, M; Espartero, J; Madrona, A; Zappia, G
An improved synthesis of cis-4-phenyl-2-propionamidotetralin (4-P-PDOT): a selective MT2 melatonin receptor antagonist.
2008 Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto; Piersanti, Giovanni
Asymmetric Alkylation of Cyclic Ketones with Dehydroalanine via H-Bond-Directing Enamine Catalysis: Straightforward Access to Enantiopure Unnatural α-Amino Acids
2022 Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni
Asymmetric Synthesis and Biological Evaluation of Both Enantiomers of 5- and 6-Boronotryptophan as Potential Boron Delivery Agents for Boron Neutron Capture Therapy
2024 Retini, Michele; Järvinen, Juulia; Bahrami, Katayun; Tampio, Janne; Bartoccini, Francesca; Riihelä, Petri; Pehkonen, Henna; Värä, Arina; Laitinen, Tuomo; Huttunen, Kristiina M.; Rautio, Jarkko; Piersanti, Giovanni; Timonen, Juri M.
Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties
2022 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Brønsted Acid-Catalyzed Bisindolization of α-amido acetals: Synthesis and Anticancer activity of bis(indolyl)ethanamino derivatives
2014 Mari, Michele; Aurora, Tassoni; Lucarini, Simone; Fanelli, Mirco; Piersanti, Giovanni; Spadoni, Gilberto
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology
2020 Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni
Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin
2019 Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Mari, Michele; Piersanti, Giovanni
Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone
2021 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Conformation by NMR of two tetralin-based receptor ligands
2003 Gatti, G.; Piersanti, Giovanni; Spadoni, Gilberto
Correlation between energetics of collisionally activated decompositions, interaction energy and biological potency of carbamates FAAH inhibitors
2007 Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
2-n-Butyl- 9-methyl-8-(1,2,3)triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological Characterization | 1-gen-2005 | Minetti, P; Tinti, M. O.; Carminati, P; Castorina, M; DI CESARE, M. A.; DI SERIO, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, Luca; Piersanti, Giovanni; Bartoccini, Francesca; Tarzia, Giorgio | |
2-n-butyl-9-methyl-8-(1,2,3)triazol-2yl-9H-purin-6-yl-amine (ST 1535) and analogs as A2a Adenosine receptor antagonists. Design, synthesis and pharmacological characterization | 1-gen-2003 | Bartoccini, Francesca; Castorina, M.; DI CESARE, M. A.; Gallo, G; Ghirardi, O.; Giorgi, F. GIORGI L.; Minetti, P.; Piersanti, Giovanni; Tarzia, Giorgio; Tinti, M. O. | |
5-(2-Ethyl-phenyl)-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole (DL-111-IT ) and related compounds induce morphological apoptotic patterns in cultures of human tumor cell lines | 1-gen-2003 | Burattini, Sabrina; Luchetti, Francesca; Battistelli, Michela; DELLA FELICE, Massimo; Papa, Stefano; Piersanti, Giovanni; Tarzia, Giorgio; Falcieri, Elisabetta | |
A Novel One-Pot Approach of Hexahydropyrrolo[2,3-b]indole Nucleus by a cascade addition/cyclization strategy: Synthesis of (±)-Esermethole | 1-gen-2010 | Lucarini, Simone; Bartoccini, Francesca; Battistoni, F; Diamantini, Giuseppe; Piersanti, Giovanni; Righi, M; Spadoni, Gilberto | |
A Short Synthesis of (−)‐6,7‐Secoagroclavine via Metal‐Free Reductive Coupling | 1-gen-2024 | Diotallevi, Francesca; Bartoccini, Francesca; Piersanti, Giovanni | |
A simple, modular synthesis of C4-substituted tryptophan derivatives | 1-gen-2016 | Bartoccini, Francesca; Bartolucci, Silvia; Mari, Michele; Piersanti, Giovanni | |
A Trans-Stereoselective Synthesis of 3-Halo-4-alkyl(aryl)-NH-azetidin-2-ones. | 1-gen-2000 | Bandini, Elisa; Favi, Gianfranco; Martelli, Giorgio; Panunzio, Mauro; Piersanti, Giovanni | |
A Versatile Biomimetic Approach to Diindolylmethane Derivatives as Potential Anticancer Agents | 1-gen-2012 | Lucarini, Simone; Piersanti, Giovanni; Duranti, Andrea; Spadoni, Gilberto | |
An efficient synthesis of the cyclic form of scalemic 2,4-di-epi-polyoxamic acid exploiting the hetero Diels-Alder approach. | 1-gen-1997 | Bandini, Elisa; Martelli, Giorgio; Spunta, Giuseppe; Bongini, Alessandro; Panunzio, Mauro; Piersanti, Giovanni | |
An efficient, economical synthesis of hydroxytyrosol and its protected forms via Baeyer–Villiger oxidation | 1-gen-2011 | Piersanti, G; Retini, M; Espartero, J; Madrona, A; Zappia, G | |
An improved synthesis of cis-4-phenyl-2-propionamidotetralin (4-P-PDOT): a selective MT2 melatonin receptor antagonist. | 1-gen-2008 | Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto; Piersanti, Giovanni | |
Asymmetric Alkylation of Cyclic Ketones with Dehydroalanine via H-Bond-Directing Enamine Catalysis: Straightforward Access to Enantiopure Unnatural α-Amino Acids | 1-gen-2022 | Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni | |
Asymmetric Synthesis and Biological Evaluation of Both Enantiomers of 5- and 6-Boronotryptophan as Potential Boron Delivery Agents for Boron Neutron Capture Therapy | 1-gen-2024 | Retini, Michele; Järvinen, Juulia; Bahrami, Katayun; Tampio, Janne; Bartoccini, Francesca; Riihelä, Petri; Pehkonen, Henna; Värä, Arina; Laitinen, Tuomo; Huttunen, Kristiina M.; Rautio, Jarkko; Piersanti, Giovanni; Timonen, Juri M. | |
Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties | 1-gen-2022 | Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni | |
Brønsted Acid-Catalyzed Bisindolization of α-amido acetals: Synthesis and Anticancer activity of bis(indolyl)ethanamino derivatives | 1-gen-2014 | Mari, Michele; Aurora, Tassoni; Lucarini, Simone; Fanelli, Mirco; Piersanti, Giovanni; Spadoni, Gilberto | |
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology | 1-gen-2020 | Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni | |
Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin | 1-gen-2019 | Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Mari, Michele; Piersanti, Giovanni | |
Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone | 1-gen-2021 | Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni | |
Conformation by NMR of two tetralin-based receptor ligands | 1-gen-2003 | Gatti, G.; Piersanti, Giovanni; Spadoni, Gilberto | |
Correlation between energetics of collisionally activated decompositions, interaction energy and biological potency of carbamates FAAH inhibitors | 1-gen-2007 | Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P. |