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Anandamide suppressess pain initiation through a peripheral endocannabinoid mechanism
2010 Clapper, Jr; MORENO SANZ, G; Russo, R; Guijarro, A; Vacondio, F; Duranti, Andrea; Tontini, Andrea; Sanchini, Silvano; Sciolino, Nr; Spradley, Jm; Hohmann, Ag; Calignano, A; Mor, M; Tarzia, Giorgio; Piomelli, D.
"Hot spots" in Medicinal Chemistry
2010 Metternich, R.; Tarzia, Giorgio
Recent advances in the development of melatonin MT1 and MT2 receptor agonists
2010 Mor, M; Rivara, S; Pala, D; Bedini, Annalida; Spadoni, Gilberto; Tarzia, Giorgio
Synthesis and Structure–Activity Relationships of N-(2-Oxo-3-oxetanyl)amides as N-Acylethanolamine-hydrolyzing Acid Amidase Inhibitors
2010 Solorzano, C; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Rivara, S; Lodola, A; Vacondio, F; Tarzia, Giorgio; Piomelli, D; Mor, M.
Understanding he Role of Carbamate Reactivity in Fatty Acid Amide Hydrolase Inhibition by OM/MM Mechanistic Modelling
2011 Lodola, A.; Capoferri, L.; Rivara, S.; Chudyk, E.; Sirrak, J.; Dyguda Kazimierowicz, E.; Andrzej Sokalski, W.; Mileni, M.; Tarzia, Giorgio; Piomelli, D.; Mor, M.; Mulholland, A. J.
Promotion of non-rapid eye movement sleep and activation of reticular thalamic neurons by a novel MT2 melatonin receptor ligand
2011 Ochoa Sanchez, R; Comai, S; Lacoste, B; Bambico, Fr; Dominguez Lopez, S; Spadoni, Gilberto; Rivara, S; Bedini, Annalida; Angeloni, D; Fraschini, F; Mor, M; Tarzia, Giorgio; Descarries, L; Gobbi, G.
Bivalent Ligand Approach on N-[2-[(3-methoxyphenyl)methylamino]ethyl]acetamide. Synthesis, Binding Affinity and Intrinsic Acivity for MT(1) and MT(2) melatonin Receptors.
2011 Spadoni, Gilberto; Bedini, Annalida; Orlando, Pierfrancesco; Lucarini, Simone; Tarzia, Giorgio; Mor, M.; Rivara, S.; Lucini, V.; Pannacci, M.; Scaglione, F.
Biphenyl-3-yl alkylcarbamates as fatty acid amide hydrolase (FAAH) inhibitors: Steric effects of N-alkyl chain on rat plasma and liver stability
2011 Vacondio, F; Silva, C; Lodola, A; Carmi, C; Rivara, S; Duranti, Andrea; Tontini, Andrea; Sanchini, Silvano; Clapper, Jr; Piomelli, D; Tarzia, Giorgio; Mor, M.
Toward the Definition of Stereochemical Requirements for MT(2)-Selective Antagonists and Partial Agonists by Studying 4-Phenyl-2-propionamidotetralin Derivatives
2011 Bedini, Annalida; Lucarini, Simone; Spadoni, Gilberto; Tarzia, Giorgio; Scaglione, F; Dugnani, S; Pannacci, M; Lucini, V; Carmi, C; Pala, D; Rivara, S; Mor, M.
ST1936 stimulates cAMP, Ca2+, ERK1/2 and Fyn Kinase through a full activation of cloned hman 5-HT6 receptors
2011 Riccioni, T.; Bordi, F.; Minetti, P.; Spadoni, Gilberto; Yun, H. M.; Im, B. H.; Tarzia, Giorgio; Rhim, H.; Borsini, F.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Anandamide suppressess pain initiation through a peripheral endocannabinoid mechanism | 1-gen-2010 | Clapper, Jr; MORENO SANZ, G; Russo, R; Guijarro, A; Vacondio, F; Duranti, Andrea; Tontini, Andrea; Sanchini, Silvano; Sciolino, Nr; Spradley, Jm; Hohmann, Ag; Calignano, A; Mor, M; Tarzia, Giorgio; Piomelli, D. | |
"Hot spots" in Medicinal Chemistry | 1-gen-2010 | Metternich, R.; Tarzia, Giorgio | |
Recent advances in the development of melatonin MT1 and MT2 receptor agonists | 1-gen-2010 | Mor, M; Rivara, S; Pala, D; Bedini, Annalida; Spadoni, Gilberto; Tarzia, Giorgio | |
Synthesis and Structure–Activity Relationships of N-(2-Oxo-3-oxetanyl)amides as N-Acylethanolamine-hydrolyzing Acid Amidase Inhibitors | 1-gen-2010 | Solorzano, C; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Rivara, S; Lodola, A; Vacondio, F; Tarzia, Giorgio; Piomelli, D; Mor, M. | |
Understanding he Role of Carbamate Reactivity in Fatty Acid Amide Hydrolase Inhibition by OM/MM Mechanistic Modelling | 1-gen-2011 | Lodola, A.; Capoferri, L.; Rivara, S.; Chudyk, E.; Sirrak, J.; Dyguda Kazimierowicz, E.; Andrzej Sokalski, W.; Mileni, M.; Tarzia, Giorgio; Piomelli, D.; Mor, M.; Mulholland, A. J. | |
Promotion of non-rapid eye movement sleep and activation of reticular thalamic neurons by a novel MT2 melatonin receptor ligand | 1-gen-2011 | Ochoa Sanchez, R; Comai, S; Lacoste, B; Bambico, Fr; Dominguez Lopez, S; Spadoni, Gilberto; Rivara, S; Bedini, Annalida; Angeloni, D; Fraschini, F; Mor, M; Tarzia, Giorgio; Descarries, L; Gobbi, G. | |
Bivalent Ligand Approach on N-[2-[(3-methoxyphenyl)methylamino]ethyl]acetamide. Synthesis, Binding Affinity and Intrinsic Acivity for MT(1) and MT(2) melatonin Receptors. | 1-gen-2011 | Spadoni, Gilberto; Bedini, Annalida; Orlando, Pierfrancesco; Lucarini, Simone; Tarzia, Giorgio; Mor, M.; Rivara, S.; Lucini, V.; Pannacci, M.; Scaglione, F. | |
Biphenyl-3-yl alkylcarbamates as fatty acid amide hydrolase (FAAH) inhibitors: Steric effects of N-alkyl chain on rat plasma and liver stability | 1-gen-2011 | Vacondio, F; Silva, C; Lodola, A; Carmi, C; Rivara, S; Duranti, Andrea; Tontini, Andrea; Sanchini, Silvano; Clapper, Jr; Piomelli, D; Tarzia, Giorgio; Mor, M. | |
Toward the Definition of Stereochemical Requirements for MT(2)-Selective Antagonists and Partial Agonists by Studying 4-Phenyl-2-propionamidotetralin Derivatives | 1-gen-2011 | Bedini, Annalida; Lucarini, Simone; Spadoni, Gilberto; Tarzia, Giorgio; Scaglione, F; Dugnani, S; Pannacci, M; Lucini, V; Carmi, C; Pala, D; Rivara, S; Mor, M. | |
ST1936 stimulates cAMP, Ca2+, ERK1/2 and Fyn Kinase through a full activation of cloned hman 5-HT6 receptors | 1-gen-2011 | Riccioni, T.; Bordi, F.; Minetti, P.; Spadoni, Gilberto; Yun, H. M.; Im, B. H.; Tarzia, Giorgio; Rhim, H.; Borsini, F. |
Legenda icone
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Opzioni
Scopri
Tipologia
- 1 Contributo su rivista 194
- 1 Contributo su rivista::1.1 Art... 194
Data di pubblicazione
- 2010 - 2020 24
- 2000 - 2009 67
- 1990 - 1999 48
- 1980 - 1989 37
- 1970 - 1979 12
- 1964 - 1969 6
Editore
- Weinheim : Wiley-VCH-Verl.. 1
- Wichtig Editore:Via Friuli 72 74,... 1
Rivista
- JOURNAL OF MEDICINAL CHEMISTRY 31
- IL FARMACO 13
- CHEMMEDCHEM 10
- IL FARMACO. EDIZIONE SCIENTIFICA 9
- RAPID COMMUNICATIONS IN MASS SPEC... 9
- EUROPEAN JOURNAL OF MEDICINAL CHE... 8
- ANNALI DI CHIMICA 6
- GAZZETTA CHIMICA ITALIANA 6
- JOURNAL OF PINEAL RESEARCH 5
- OMS, ORGANIC MASS SPECTROMETRY 5
Keyword
- Melatonin 3
- 5-HT7 1
- adenosine A2a receptors 1
- Amides 1
- Amidohydrolases 1
- Amino Acid Sequence 1
- Animals 1
- Anti-Inflammatory Agents 1
- Antioxidant 1
- Anxiety 1
Lingua
- eng 154
- ita 3
Accesso al fulltext
- no fulltext 193
- partially open 1