Sfoglia per Autore
Versatile stereoselective oxidative alkoxycarbonylation of styrenes at room-temperature
2024 Olivieri, Diego; Verboni, Michele; Tarroni, Riccardo; Zacchini, Stefano; Lucarini, Simone; Della Ca', Nicola; Mancuso, Raffaella; Gabriele, Bartolo; Carfagna, Carla
Easy one-pot synthesis of multifunctionalized indole–pyrrole hybrids as a new class of antileishmanial agents
2024 Ciccone, Vittorio; Diotallevi, Aurora; Gómez-Benmansour, Miriam; Maestrini, Sara; Mantellini, Fabio; Mari, Giacomo; Galluzzi, Luca; Lucarini, Simone; Favi, Gianfranco
Exploring hydrophilic 2,2-di(indol-3-yl)ethanamine derivatives against Leishmania infantum
2024 Centanni, Alessia; Diotallevi, Aurora; Buffi, Gloria; Olivieri, Diego; Santarém, Nuno; Lehtinen, Antti; Yli-Kauhaluoma, Jari; Cordeiro-da-Silva, Anabela; Kiuru, Paula; Lucarini, Simone; Galluzzi, Luca
Synthetic Methodologies and Therapeutic Potential of Indole-3-Carbinol (I3C) and Its Derivatives
2023 Centofanti, Federica; Buono, Alessandro; Verboni, Michele; Tomino, Carlo; Lucarini, Simone; Duranti, Andrea; Pandolfi, Pier Paolo; Novelli, Giuseppe
Synthesis and Properties of Sucrose- and Lactose-Based Aromatic Ester Surfactants as Potential Drugs Permeability Enhancers
2023 Verboni, Michele; Perinelli, Diego Romano; Qiu, Carol Yingshan; Tiboni, Mattia; Aluigi, Annalisa; Lucarini, Simone; Lam, Jenny K. W.; Duranti, Andrea
Synthesis and Biological Evaluation of 6-O-Sucrose Monoester Glycolipids as Possible New Antifungal Agents
2023 Verboni, Michele; Sisti, Maurizio; Campana, Raffaella; Benedetti, Serena; Palma, Francesco; Potenza, Lucia; Lucarini, Simone; Duranti, Andrea
Sugar-Based Monoester Surfactants: Synthetic Methodologies, Properties, and Biological Activities
2023 Verboni, Michele; Romano Perinelli, Diego; Buono, Alessandro; Campana, Raffaella; Sisti, Maurizio; Duranti, Andrea; Lucarini, Simone
The influence of mannose-based esters on the mesophase behaviour of lyotropic liquid crystalline nanosystems as drug delivery vectors
2023 Tiboni, Mattia; Astolfi, Paola; Verboni, Michele; Benedetti, Serena; Giorgini, Elisabetta; Notarstefano, Valentina; Vita, Francesco; Ranieri, Simone; Duranti, Andrea; Lucarini, Simone; Casettari, Luca; Pisani, Michela
Synthesis and Biological Characterization of the New Glycolipid Lactose Undecylenate (URB1418)
2022 Verboni, Michele; Benedetti, Serena; Campana, Raffaella; Palma, Francesco; Potenza, Lucia; Sisti, Maurizio; Duranti, Andrea; Lucarini, Simone
A combination of sugar esters and chitosan to promote in vivo wound care
2022 Tiboni, Mattia; Elmowafy, Enas; El-Derany, Marwa O; Benedetti, Serena; Campana, Raffaella; Verboni, Michele; Potenza, Lucia; Palma, Francesco; Citterio, Barbara; Sisti, Maurizio; Duranti, Andrea; Lucarini, Simone; Soliman, Mahmoud E; Casettari, Luca
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors
2022 Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
Morpho-functional analyses reveal that changes in the chemical structure of a marine bisindole alkaloid alter the cytotoxic effect of its derivatives
2022 Burattini, Sabrina; Battistelli, Michela; Verboni, Michele; Falcieri, Elisabetta; Faenza, Irene; Lucarini, Simone; Salucci, Sara
Special issue: Chirality in pharmaceutical research and development
2022 Collina, Simona; Lucarini, Simone; Benet-Buchholz, Jordi; Trapp, Oliver; Pescitelli, Gennaro; Berova, Nina
A recent update on new synthetic chiral compounds with antileishmanial activity
2022 Verboni, Michele; Olivieri, Diego; Lucarini, Simone
Phenotype screening of a bisindole chemical library identifies URB1483 as a new Antileishmanial agent with Topoisomerase IB as possible molecular target
2021 Lucarini, Simone; Diotallevi, Aurora; Buffi, Gloria; Scalvini, Laura; Lodola, Alessio; Favi, Gianfranco; Castelli, Silvia; Desideri and Luca Galluzzi, Alessandro
6'-O-Lactose Ester Surfactants as an Innovative Opportunity in the Pharmaceutical Field: From Synthetic Methods to Biological Applications
2021 Verboni, Michele; Lucarini, Simone; Duranti, Andrea
A comprehensive UHPLC-MS/MS screening method for the analysis of 98 New Psychoactive Substances and related compounds in human hair
2021 Nzekoue, Franks Kamgang; Agostini, Marco; Verboni, Michele; Renzoni, Caterina; Alfieri, Lucia; Barocci, Simone; Ricciutelli, Massimo; Caprioli, Giovanni; Lucarini, Simone
Phenotype Screening of an Azole-bisindole Chemical Library Identifies URB1483 as a New Antileishmanial Agent Devoid of Toxicity on Human Cells
2021 Diotallevi, Aurora; Scalvini, Laura; Buffi, Gloria; Pérez-Pertejo, Yolanda; De Santi, Mauro; Verboni, Michele; Favi, Gianfranco; Magnani, Mauro; Lodola, Alessio; Lucarini, Simone; Galluzzi, Luca
Permeability-enhancing effects of three laurate-disaccharide monoesters across isolated rat intestinal mucosae
2021 Mccartney, Fiona; Perinelli, Diego R; Tiboni, Mattia; Cavanagh, Robert; Lucarini, Simone; Filippo Palmieri, Giovanni; Casettari, Luca; Brayden, David J
A Fluorinated Analogue of Marine Bisindole Alkaloid 2,2-Bis(6-bromo-1H-indol-3-yl)ethanamine as Potential Anti-Biofilm Agent and Antibiotic Adjuvant Against Staphylococcus aureus
2020 Campana, Raffaella; Mangiaterra, Gianmarco; Tiboni, Mattia; Frangipani, Emanuela; Biavasco, Francesca; Lucarini, Simone; Citterio, Barbara
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Versatile stereoselective oxidative alkoxycarbonylation of styrenes at room-temperature | 1-gen-2024 | Olivieri, Diego; Verboni, Michele; Tarroni, Riccardo; Zacchini, Stefano; Lucarini, Simone; Della Ca', Nicola; Mancuso, Raffaella; Gabriele, Bartolo; Carfagna, Carla | |
Easy one-pot synthesis of multifunctionalized indole–pyrrole hybrids as a new class of antileishmanial agents | 1-gen-2024 | Ciccone, Vittorio; Diotallevi, Aurora; Gómez-Benmansour, Miriam; Maestrini, Sara; Mantellini, Fabio; Mari, Giacomo; Galluzzi, Luca; Lucarini, Simone; Favi, Gianfranco | |
Exploring hydrophilic 2,2-di(indol-3-yl)ethanamine derivatives against Leishmania infantum | 1-gen-2024 | Centanni, Alessia; Diotallevi, Aurora; Buffi, Gloria; Olivieri, Diego; Santarém, Nuno; Lehtinen, Antti; Yli-Kauhaluoma, Jari; Cordeiro-da-Silva, Anabela; Kiuru, Paula; Lucarini, Simone; Galluzzi, Luca | |
Synthetic Methodologies and Therapeutic Potential of Indole-3-Carbinol (I3C) and Its Derivatives | 1-gen-2023 | Centofanti, Federica; Buono, Alessandro; Verboni, Michele; Tomino, Carlo; Lucarini, Simone; Duranti, Andrea; Pandolfi, Pier Paolo; Novelli, Giuseppe | |
Synthesis and Properties of Sucrose- and Lactose-Based Aromatic Ester Surfactants as Potential Drugs Permeability Enhancers | 1-gen-2023 | Verboni, Michele; Perinelli, Diego Romano; Qiu, Carol Yingshan; Tiboni, Mattia; Aluigi, Annalisa; Lucarini, Simone; Lam, Jenny K. W.; Duranti, Andrea | |
Synthesis and Biological Evaluation of 6-O-Sucrose Monoester Glycolipids as Possible New Antifungal Agents | 1-gen-2023 | Verboni, Michele; Sisti, Maurizio; Campana, Raffaella; Benedetti, Serena; Palma, Francesco; Potenza, Lucia; Lucarini, Simone; Duranti, Andrea | |
Sugar-Based Monoester Surfactants: Synthetic Methodologies, Properties, and Biological Activities | 1-gen-2023 | Verboni, Michele; Romano Perinelli, Diego; Buono, Alessandro; Campana, Raffaella; Sisti, Maurizio; Duranti, Andrea; Lucarini, Simone | |
The influence of mannose-based esters on the mesophase behaviour of lyotropic liquid crystalline nanosystems as drug delivery vectors | 1-gen-2023 | Tiboni, Mattia; Astolfi, Paola; Verboni, Michele; Benedetti, Serena; Giorgini, Elisabetta; Notarstefano, Valentina; Vita, Francesco; Ranieri, Simone; Duranti, Andrea; Lucarini, Simone; Casettari, Luca; Pisani, Michela | |
Synthesis and Biological Characterization of the New Glycolipid Lactose Undecylenate (URB1418) | 1-gen-2022 | Verboni, Michele; Benedetti, Serena; Campana, Raffaella; Palma, Francesco; Potenza, Lucia; Sisti, Maurizio; Duranti, Andrea; Lucarini, Simone | |
A combination of sugar esters and chitosan to promote in vivo wound care | 1-gen-2022 | Tiboni, Mattia; Elmowafy, Enas; El-Derany, Marwa O; Benedetti, Serena; Campana, Raffaella; Verboni, Michele; Potenza, Lucia; Palma, Francesco; Citterio, Barbara; Sisti, Maurizio; Duranti, Andrea; Lucarini, Simone; Soliman, Mahmoud E; Casettari, Luca | |
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors | 1-gen-2022 | Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto | |
Morpho-functional analyses reveal that changes in the chemical structure of a marine bisindole alkaloid alter the cytotoxic effect of its derivatives | 1-gen-2022 | Burattini, Sabrina; Battistelli, Michela; Verboni, Michele; Falcieri, Elisabetta; Faenza, Irene; Lucarini, Simone; Salucci, Sara | |
Special issue: Chirality in pharmaceutical research and development | 1-gen-2022 | Collina, Simona; Lucarini, Simone; Benet-Buchholz, Jordi; Trapp, Oliver; Pescitelli, Gennaro; Berova, Nina | |
A recent update on new synthetic chiral compounds with antileishmanial activity | 1-gen-2022 | Verboni, Michele; Olivieri, Diego; Lucarini, Simone | |
Phenotype screening of a bisindole chemical library identifies URB1483 as a new Antileishmanial agent with Topoisomerase IB as possible molecular target | 1-gen-2021 | Lucarini, Simone; Diotallevi, Aurora; Buffi, Gloria; Scalvini, Laura; Lodola, Alessio; Favi, Gianfranco; Castelli, Silvia; Desideri and Luca Galluzzi, Alessandro | |
6'-O-Lactose Ester Surfactants as an Innovative Opportunity in the Pharmaceutical Field: From Synthetic Methods to Biological Applications | 1-gen-2021 | Verboni, Michele; Lucarini, Simone; Duranti, Andrea | |
A comprehensive UHPLC-MS/MS screening method for the analysis of 98 New Psychoactive Substances and related compounds in human hair | 1-gen-2021 | Nzekoue, Franks Kamgang; Agostini, Marco; Verboni, Michele; Renzoni, Caterina; Alfieri, Lucia; Barocci, Simone; Ricciutelli, Massimo; Caprioli, Giovanni; Lucarini, Simone | |
Phenotype Screening of an Azole-bisindole Chemical Library Identifies URB1483 as a New Antileishmanial Agent Devoid of Toxicity on Human Cells | 1-gen-2021 | Diotallevi, Aurora; Scalvini, Laura; Buffi, Gloria; Pérez-Pertejo, Yolanda; De Santi, Mauro; Verboni, Michele; Favi, Gianfranco; Magnani, Mauro; Lodola, Alessio; Lucarini, Simone; Galluzzi, Luca | |
Permeability-enhancing effects of three laurate-disaccharide monoesters across isolated rat intestinal mucosae | 1-gen-2021 | Mccartney, Fiona; Perinelli, Diego R; Tiboni, Mattia; Cavanagh, Robert; Lucarini, Simone; Filippo Palmieri, Giovanni; Casettari, Luca; Brayden, David J | |
A Fluorinated Analogue of Marine Bisindole Alkaloid 2,2-Bis(6-bromo-1H-indol-3-yl)ethanamine as Potential Anti-Biofilm Agent and Antibiotic Adjuvant Against Staphylococcus aureus | 1-gen-2020 | Campana, Raffaella; Mangiaterra, Gianmarco; Tiboni, Mattia; Frangipani, Emanuela; Biavasco, Francesca; Lucarini, Simone; Citterio, Barbara |
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