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Quantification of 2- and 3-isopropylmalic acids in forty Italian wines by UHPLC-MS/MS triple quadrupole and evaluation of their antimicrobial, antioxidant activities and biocompatibility 1-gen-2020 Ricciutelli, Massimo; Bartolucci, Gianluca; Campana, Raffaella; Salucci, Sara; Benedetti, Serena; Caprioli, Giovanni; Maggi, Filippo; Sagratini, Gianni; Vittori, Sauro; Lucarini, Simone
SYNTHESIS AND EVALUATION OF SUGAR-BASED ALIPHATIC AND AROMATIC FATTY ACID ESTERS AS ANTIMICROBIAL AND ANTIBIOFILM AGENTS 1-gen-2019 Lucarini, Simone; Campana, Raffaella; Duranti, Andrea
Lactose-based Fatty Acid Monoesters: Synthesis, antimicrobial activity and permeability enhancement studies 1-gen-2019 Lucarini, Simone
Marine Alkaloid 2,2-Bis(6-bromo-3-indolyl) Ethylamine and Its Synthetic Derivatives Inhibit Microbial Biofilms Formation and Disaggregate Developed Biofilms 1-gen-2019 Campana, Raffaella; Favi, Gianfranco; Baffone, Wally; Lucarini, Simone
Synthesis and Evaluation of Saccharide-Based Aliphatic and Aromatic Esters as Antimicrobial and Antibiofilm Agents 1-gen-2019 Campana, Raffaella; Merli, Alessio; Verboni, Michele; Biondo, Francesca; Favi, Gianfranco; Duranti, Andrea; Lucarini, Simone
Marine bisindole alkaloid 2,2-bis(6-bromo-3-indolyl)ethylamine to control and prevent fungal growth on building material: a potential antifungal agent 1-gen-2019 Campana, Raffaella; Sisti, Maurizio; Sabatini, Luigia; Lucarini, Simone
Identification and quantification of new isomers of isopropyl-malic acid in wine by LC-IT and LC-Q-Orbitrap 1-gen-2019 Ricciutelli, Massimo; Moretti, Simone; Galarini, Roberta; Sagratini, Gianni; Mari, Michele; Lucarini, Simone; Vittori, Sauro; Caprioli, Giovanni
Synthesis, Structure-Activity Relationships and In Vitro Toxicity Profile of Lactose-Based Fatty Acid Monoesters as Possible Drug Permeability Enhancers 1-gen-2018 Lucarini, Simone; Fagioli, Laura; Cavanagh, Robert; Liang, Wanling; Perinelli, Diego Romano; Campana, Mario; Stolnik, Snjezana; Lam, Jenny K W; Casettari, Luca; Duranti, Andrea
Lactose oleate as new biocompatible surfactant for pharmaceutical applications 1-gen-2018 Perinelli, D. R; Lucarini, S; Fagioli, L; Campana, R; Vllasaliu, D; Duranti, A; Casettari, L.
Marine bisindole alkaloid: A potential apoptotic inducer in human cancer cells 1-gen-2018 Salucci, Sara; Burattini, Sabrina; Buontempo, Francesca; Orsini, E; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Martelli, Alberto Maria; Falcieri, Elisabetta
Polycyclic Indolines by Acid-Mediated Intramolecular Dearomative Strategy: Reversing Indole Reactivity in the Pictet‒Spengler-Type Reaction 1-gen-2018 Ciccolini, Cecilia; Mari, Michele; Lucarini, Simone; Mantellini, Fabio; Piersanti, Giovanni; Favi, Gianfranco
Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands 1-gen-2018 Rivara, Silvia; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Caignard, Daniel-Henri; Delagrange, Philippe; Collina, Simona; Lucini, Valeria; Scaglione, Francesco; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto
Further Highlighting on the Prevention of Oxidative Damage by Polyphenol-Rich Wine Extracts 1-gen-2017 Salucci, Sara; Burattini, Sabrina; Giordano, FRANCESCO MARIA; Lucarini, Simone; Diamantini, Giuseppe; Falcieri, Elisabetta
Palladium(II)-Catalyzed Intramolecular Oxidative C−H/C−H Cross-Coupling Reaction of C3,N-linked Biheterocycles: Rapid Access to Polycyclic Nitrogen Heterocycles 1-gen-2017 Mantenuto, Serena; Ciccolini, Cecilia; Lucarini, Simone; Piersanti, Giovanni; Favi, Gianfranco; Mantellini, Fabio
One-Pot Synthesis of Biheterocycles Based on Indole and Azole Scaffolds Using Tryptamines and 1,2-Diaza-1,3-dienes as Building Blocks 1-gen-2016 Mantenuto, Serena; Lucarini, Simone; DE SANTI, Mauro; Piersanti, Giovanni; Brandi, Giorgio; Favi, Gianfranco; Mantellini, Fabio
Unsaturated fatty acids lactose esters: cytotoxicity, permeability enhancement and antimicrobial activity 1-gen-2016 Lucarini, Simone; Fagioli, Laura; Campana, Raffaella; Cole, Hannah; Duranti, Andrea; Baffone, Wally; Vllasaliu, Driton; Casettari, Luca
Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands 1-gen-2015 Pace, Silvia; Brogin, Giandomenico; Stasi, Maria Antonietta; Riccioni, Teresa; Borsini, Franco; Capocasa, Francesca; Manera, Francesco; Tallarico, Carlo; Grossi, Pietro; Vacondio, Federica; Bassi, Michele; Bartoccini, Francesca; Lucarini, Simone; Piersanti, Giovanni; Tarzia, Giorgio; Cabri, Walter; Minetti, Patrizia
Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives 1-gen-2015 Bartoccini, Francesca; Bartolucci, Silvia; Lucarini, Simone; Piersanti, Giovanni
Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines 1-gen-2015 Spadoni, Gilberto; Bedini, Annalida; Lucarini, Simone; Mari, Michele; Caignard, D; Boutin, J; Delagrange, P; Lucini, V; Scaglione, F; Lodola, A; Zanardi, F; Pala, D; Mor, M; Rivara, S.
Pharmacokinetic and pharmacodynamic evaluation of ramelteon : an insomnia therapy 1-gen-2015 Spadoni, Gilberto; Bedini, Annalida; Lucarini, Simone; Mor, Marco; Rivara, Silvia
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