Sfoglia per Autore
Quantification of 2- and 3-isopropylmalic acids in forty Italian wines by UHPLC-MS/MS triple quadrupole and evaluation of their antimicrobial, antioxidant activities and biocompatibility
2020 Ricciutelli, Massimo; Bartolucci, Gianluca; Campana, Raffaella; Salucci, Sara; Benedetti, Serena; Caprioli, Giovanni; Maggi, Filippo; Sagratini, Gianni; Vittori, Sauro; Lucarini, Simone
SYNTHESIS AND EVALUATION OF SUGAR-BASED ALIPHATIC AND AROMATIC FATTY ACID ESTERS AS ANTIMICROBIAL AND ANTIBIOFILM AGENTS
2019 Lucarini, Simone; Campana, Raffaella; Duranti, Andrea
Lactose-based Fatty Acid Monoesters: Synthesis, antimicrobial activity and permeability enhancement studies
2019 Lucarini, Simone
Marine Alkaloid 2,2-Bis(6-bromo-3-indolyl) Ethylamine and Its Synthetic Derivatives Inhibit Microbial Biofilms Formation and Disaggregate Developed Biofilms
2019 Campana, Raffaella; Favi, Gianfranco; Baffone, Wally; Lucarini, Simone
Synthesis and Evaluation of Saccharide-Based Aliphatic and Aromatic Esters as Antimicrobial and Antibiofilm Agents
2019 Campana, Raffaella; Merli, Alessio; Verboni, Michele; Biondo, Francesca; Favi, Gianfranco; Duranti, Andrea; Lucarini, Simone
Marine bisindole alkaloid 2,2-bis(6-bromo-3-indolyl)ethylamine to control and prevent fungal growth on building material: a potential antifungal agent
2019 Campana, Raffaella; Sisti, Maurizio; Sabatini, Luigia; Lucarini, Simone
Identification and quantification of new isomers of isopropyl-malic acid in wine by LC-IT and LC-Q-Orbitrap
2019 Ricciutelli, Massimo; Moretti, Simone; Galarini, Roberta; Sagratini, Gianni; Mari, Michele; Lucarini, Simone; Vittori, Sauro; Caprioli, Giovanni
Synthesis, Structure-Activity Relationships and In Vitro Toxicity Profile of Lactose-Based Fatty Acid Monoesters as Possible Drug Permeability Enhancers
2018 Lucarini, Simone; Fagioli, Laura; Cavanagh, Robert; Liang, Wanling; Perinelli, Diego Romano; Campana, Mario; Stolnik, Snjezana; Lam, Jenny K W; Casettari, Luca; Duranti, Andrea
Lactose oleate as new biocompatible surfactant for pharmaceutical applications
2018 Perinelli, D. R; Lucarini, S; Fagioli, L; Campana, R; Vllasaliu, D; Duranti, A; Casettari, L.
Marine bisindole alkaloid: A potential apoptotic inducer in human cancer cells
2018 Salucci, Sara; Burattini, Sabrina; Buontempo, Francesca; Orsini, E; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Martelli, Alberto Maria; Falcieri, Elisabetta
Polycyclic Indolines by Acid-Mediated Intramolecular Dearomative Strategy: Reversing Indole Reactivity in the Pictet‒Spengler-Type Reaction
2018 Ciccolini, Cecilia; Mari, Michele; Lucarini, Simone; Mantellini, Fabio; Piersanti, Giovanni; Favi, Gianfranco
Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands
2018 Rivara, Silvia; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Caignard, Daniel-Henri; Delagrange, Philippe; Collina, Simona; Lucini, Valeria; Scaglione, Francesco; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto
Further Highlighting on the Prevention of Oxidative Damage by Polyphenol-Rich Wine Extracts
2017 Salucci, Sara; Burattini, Sabrina; Giordano, FRANCESCO MARIA; Lucarini, Simone; Diamantini, Giuseppe; Falcieri, Elisabetta
Palladium(II)-Catalyzed Intramolecular Oxidative C−H/C−H Cross-Coupling Reaction of C3,N-linked Biheterocycles: Rapid Access to Polycyclic Nitrogen Heterocycles
2017 Mantenuto, Serena; Ciccolini, Cecilia; Lucarini, Simone; Piersanti, Giovanni; Favi, Gianfranco; Mantellini, Fabio
One-Pot Synthesis of Biheterocycles Based on Indole and Azole Scaffolds Using Tryptamines and 1,2-Diaza-1,3-dienes as Building Blocks
2016 Mantenuto, Serena; Lucarini, Simone; DE SANTI, Mauro; Piersanti, Giovanni; Brandi, Giorgio; Favi, Gianfranco; Mantellini, Fabio
Unsaturated fatty acids lactose esters: cytotoxicity, permeability enhancement and antimicrobial activity
2016 Lucarini, Simone; Fagioli, Laura; Campana, Raffaella; Cole, Hannah; Duranti, Andrea; Baffone, Wally; Vllasaliu, Driton; Casettari, Luca
Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands
2015 Pace, Silvia; Brogin, Giandomenico; Stasi, Maria Antonietta; Riccioni, Teresa; Borsini, Franco; Capocasa, Francesca; Manera, Francesco; Tallarico, Carlo; Grossi, Pietro; Vacondio, Federica; Bassi, Michele; Bartoccini, Francesca; Lucarini, Simone; Piersanti, Giovanni; Tarzia, Giorgio; Cabri, Walter; Minetti, Patrizia
Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives
2015 Bartoccini, Francesca; Bartolucci, Silvia; Lucarini, Simone; Piersanti, Giovanni
Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines
2015 Spadoni, Gilberto; Bedini, Annalida; Lucarini, Simone; Mari, Michele; Caignard, D; Boutin, J; Delagrange, P; Lucini, V; Scaglione, F; Lodola, A; Zanardi, F; Pala, D; Mor, M; Rivara, S.
Pharmacokinetic and pharmacodynamic evaluation of ramelteon : an insomnia therapy
2015 Spadoni, Gilberto; Bedini, Annalida; Lucarini, Simone; Mor, Marco; Rivara, Silvia
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Quantification of 2- and 3-isopropylmalic acids in forty Italian wines by UHPLC-MS/MS triple quadrupole and evaluation of their antimicrobial, antioxidant activities and biocompatibility | 1-gen-2020 | Ricciutelli, Massimo; Bartolucci, Gianluca; Campana, Raffaella; Salucci, Sara; Benedetti, Serena; Caprioli, Giovanni; Maggi, Filippo; Sagratini, Gianni; Vittori, Sauro; Lucarini, Simone | |
SYNTHESIS AND EVALUATION OF SUGAR-BASED ALIPHATIC AND AROMATIC FATTY ACID ESTERS AS ANTIMICROBIAL AND ANTIBIOFILM AGENTS | 1-gen-2019 | Lucarini, Simone; Campana, Raffaella; Duranti, Andrea | |
Lactose-based Fatty Acid Monoesters: Synthesis, antimicrobial activity and permeability enhancement studies | 1-gen-2019 | Lucarini, Simone | |
Marine Alkaloid 2,2-Bis(6-bromo-3-indolyl) Ethylamine and Its Synthetic Derivatives Inhibit Microbial Biofilms Formation and Disaggregate Developed Biofilms | 1-gen-2019 | Campana, Raffaella; Favi, Gianfranco; Baffone, Wally; Lucarini, Simone | |
Synthesis and Evaluation of Saccharide-Based Aliphatic and Aromatic Esters as Antimicrobial and Antibiofilm Agents | 1-gen-2019 | Campana, Raffaella; Merli, Alessio; Verboni, Michele; Biondo, Francesca; Favi, Gianfranco; Duranti, Andrea; Lucarini, Simone | |
Marine bisindole alkaloid 2,2-bis(6-bromo-3-indolyl)ethylamine to control and prevent fungal growth on building material: a potential antifungal agent | 1-gen-2019 | Campana, Raffaella; Sisti, Maurizio; Sabatini, Luigia; Lucarini, Simone | |
Identification and quantification of new isomers of isopropyl-malic acid in wine by LC-IT and LC-Q-Orbitrap | 1-gen-2019 | Ricciutelli, Massimo; Moretti, Simone; Galarini, Roberta; Sagratini, Gianni; Mari, Michele; Lucarini, Simone; Vittori, Sauro; Caprioli, Giovanni | |
Synthesis, Structure-Activity Relationships and In Vitro Toxicity Profile of Lactose-Based Fatty Acid Monoesters as Possible Drug Permeability Enhancers | 1-gen-2018 | Lucarini, Simone; Fagioli, Laura; Cavanagh, Robert; Liang, Wanling; Perinelli, Diego Romano; Campana, Mario; Stolnik, Snjezana; Lam, Jenny K W; Casettari, Luca; Duranti, Andrea | |
Lactose oleate as new biocompatible surfactant for pharmaceutical applications | 1-gen-2018 | Perinelli, D. R; Lucarini, S; Fagioli, L; Campana, R; Vllasaliu, D; Duranti, A; Casettari, L. | |
Marine bisindole alkaloid: A potential apoptotic inducer in human cancer cells | 1-gen-2018 | Salucci, Sara; Burattini, Sabrina; Buontempo, Francesca; Orsini, E; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Martelli, Alberto Maria; Falcieri, Elisabetta | |
Polycyclic Indolines by Acid-Mediated Intramolecular Dearomative Strategy: Reversing Indole Reactivity in the Pictet‒Spengler-Type Reaction | 1-gen-2018 | Ciccolini, Cecilia; Mari, Michele; Lucarini, Simone; Mantellini, Fabio; Piersanti, Giovanni; Favi, Gianfranco | |
Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands | 1-gen-2018 | Rivara, Silvia; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Caignard, Daniel-Henri; Delagrange, Philippe; Collina, Simona; Lucini, Valeria; Scaglione, Francesco; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto | |
Further Highlighting on the Prevention of Oxidative Damage by Polyphenol-Rich Wine Extracts | 1-gen-2017 | Salucci, Sara; Burattini, Sabrina; Giordano, FRANCESCO MARIA; Lucarini, Simone; Diamantini, Giuseppe; Falcieri, Elisabetta | |
Palladium(II)-Catalyzed Intramolecular Oxidative C−H/C−H Cross-Coupling Reaction of C3,N-linked Biheterocycles: Rapid Access to Polycyclic Nitrogen Heterocycles | 1-gen-2017 | Mantenuto, Serena; Ciccolini, Cecilia; Lucarini, Simone; Piersanti, Giovanni; Favi, Gianfranco; Mantellini, Fabio | |
One-Pot Synthesis of Biheterocycles Based on Indole and Azole Scaffolds Using Tryptamines and 1,2-Diaza-1,3-dienes as Building Blocks | 1-gen-2016 | Mantenuto, Serena; Lucarini, Simone; DE SANTI, Mauro; Piersanti, Giovanni; Brandi, Giorgio; Favi, Gianfranco; Mantellini, Fabio | |
Unsaturated fatty acids lactose esters: cytotoxicity, permeability enhancement and antimicrobial activity | 1-gen-2016 | Lucarini, Simone; Fagioli, Laura; Campana, Raffaella; Cole, Hannah; Duranti, Andrea; Baffone, Wally; Vllasaliu, Driton; Casettari, Luca | |
Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands | 1-gen-2015 | Pace, Silvia; Brogin, Giandomenico; Stasi, Maria Antonietta; Riccioni, Teresa; Borsini, Franco; Capocasa, Francesca; Manera, Francesco; Tallarico, Carlo; Grossi, Pietro; Vacondio, Federica; Bassi, Michele; Bartoccini, Francesca; Lucarini, Simone; Piersanti, Giovanni; Tarzia, Giorgio; Cabri, Walter; Minetti, Patrizia | |
Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives | 1-gen-2015 | Bartoccini, Francesca; Bartolucci, Silvia; Lucarini, Simone; Piersanti, Giovanni | |
Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines | 1-gen-2015 | Spadoni, Gilberto; Bedini, Annalida; Lucarini, Simone; Mari, Michele; Caignard, D; Boutin, J; Delagrange, P; Lucini, V; Scaglione, F; Lodola, A; Zanardi, F; Pala, D; Mor, M; Rivara, S. | |
Pharmacokinetic and pharmacodynamic evaluation of ramelteon : an insomnia therapy | 1-gen-2015 | Spadoni, Gilberto; Bedini, Annalida; Lucarini, Simone; Mor, Marco; Rivara, Silvia |
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