Sfoglia per Autore
SYNTHESIS AND EVALUATION OF SUGAR-BASED ALIPHATIC AND AROMATIC FATTY ACID ESTERS AS ANTIMICROBIAL AND ANTIBIOFILM AGENTS
2019 Lucarini, Simone; Campana, Raffaella; Duranti, Andrea
Synthesis and Evaluation of Saccharide-Based Aliphatic and Aromatic Esters as Antimicrobial and Antibiofilm Agents
2019 Campana, Raffaella; Merli, Alessio; Verboni, Michele; Biondo, Francesca; Favi, Gianfranco; Duranti, Andrea; Lucarini, Simone
Pharmacokinetics, pharmacodynamics and safety studies on URB 937, a peripherally restricted fatty acid amide hydrolase inhibitor, in rats
2019 Vozella, Valentina; Ahmed, Faizy; Choobchian, Paoula; Merrill, Collin B.; Zibardi, Cristina; Tarzia, Giorgio; Mor, Marco; Duranti, Andrea; Tontini, Andrea; Rivara, Silvia; Piomelli, Daniele
Acute Reduction in Neonatal Brain Injury by Selective Blockage of CB1 and Activation of CB2 Receptors
2019 Alonso-Alconada, D; Carloni, S; Duranti, A; Pintor-Rial, A; Alvarez, A; Hilario, E; Balduini, W
Lactose oleate as new biocompatible surfactant for pharmaceutical applications
2018 Perinelli, D. R; Lucarini, S; Fagioli, L; Campana, R; Vllasaliu, D; Duranti, A; Casettari, L.
Synthesis, Structure-Activity Relationships and In Vitro Toxicity Profile of Lactose-Based Fatty Acid Monoesters as Possible Drug Permeability Enhancers
2018 Lucarini, Simone; Fagioli, Laura; Cavanagh, Robert; Liang, Wanling; Perinelli, Diego Romano; Campana, Mario; Stolnik, Snjezana; Lam, Jenny K W; Casettari, Luca; Duranti, Andrea
The fatty acid amide hydrolase inhibitor URB597 modulates serotonin-dependent emotional behaviour, and serotonin1A and serotonin2A/C activity in the hippocampus
2016 Bambico, Fr; Duranti, Andrea; Nobrega, Jn; Gobbi, G.
Unsaturated fatty acids lactose esters: cytotoxicity, permeability enhancement and antimicrobial activity
2016 Lucarini, Simone; Fagioli, Laura; Campana, Raffaella; Cole, Hannah; Duranti, Andrea; Baffone, Wally; Vllasaliu, Driton; Casettari, Luca
Composition and Methods of Inhibiting N-Acylethanolamine-hydrolyzing Acid Amidase
2016 Piomelli, D; Tarzia, Giorgio; Mor, M; Duranti, Andrea; Tontini, Andrea
Inhibition of anandamide hydrolysis enhances noradrenergic and GABAergic transmission in the prefrontal cortex and basolateral amygdala of rat subjected to acute swim stress
2015 Besde, G; Romano, A; Tempesta, B; Lavecchia, Ma; Pace, L; Bellomo, A; Duranti, Andrea; MICIONI DI BONAVENTURA, Mv; Cifani, C; Cassano, T; Gaetani, S.
Chronic stimulation of the endogenous anandamide tone reduces cocaine-seeking and cue-induced relapse in rats
2015 Chauvet, C; Nicolas, C; Thiriet, N; Lardeux, V; Duranti, Andrea; Solinas, M.
Anestetici locali (Cap. 14)
2015 Duranti, Andrea
Derivatizzazione one-pot di indoli per la sintesi di triptofani, pirroloindoline, bis-indoli & co
2014 Lucarini, Simone; Piersanti, Giovanni; Duranti, Andrea; Spadoni, Gilberto
Structural determinants of peripheral O-arylcarbamate FAAH inhibitors render them dual substrates for Abcb1 and Abcg2 and restrict their access to the brain
2014 MORENO SANZ, G; Barrera, B; Armirotti, A; MANDRUP BERTOZZI, S; Prieto, Jg; Scarpelli, R; Duranti, Andrea; Tarzia, Giorgio; Bandiera, T; Merino, G; Piomelli, D.
Prior stimulation of the endocannabinoid system prevents methamphetamine-induced neurotoxicity in the striatum through activation of CB2 receptors
2014 Nader, J; Rapino, C; Gennequin, B; Chavant, F; Francheteau, M; Makriyannis, A; Duranti, Andrea; Maccarrone, M; Solinas, M; Thiriet, N.
Stimulation of the endocannabinoid system prevents methamphetamine-induced neurotoxicity in mice
2013 Thiriet, N; Nader, J; Rapino, C; Gennequin, B; Francheteau, M; Makryiannis, A; Duranti, Andrea; Maccarrone, M; Solinas, M.
Sintesi e studi di relazione struttura–attività/selettività su O-bifenil-3-ilcarbammati disostituiti quali inibitori periferici dell’enzima FAAH
2013 Mestichelli, Paola; MORENO SANZ, G; Duranti, Andrea; Sanchini, Silvano; Tontini, Andrea; Lodola, A; Mor, M; Bandiera, T; Piomelli, D; Tarzia, Giorgio
O-Biphenyl-3-yl Carbamates as Peripheral FAAH Inhibitors: Synthesis and Structure–Activity (SAR) Relationship Studies
2013 Mestichelli, Paola; MORENO SANZ, G; Duranti, Andrea; Sanchini, Silvano; Tontini, Andrea; Lodola, A; Mor, M; Bandiera, T; Piomelli, D; Tarzia, Giorgio
Synthesis and Structure–Activity Relationship (SAR) of 2-Methyl-4-oxo-3-oxetanyl Carbamic Acid Esters, a Class of Potent N-Acylethanolamine Acid Amidase (NAAA) Inhibitors
2013 Ponzano, S; Bertozzi, F; Mengatto, L; Dionisi, M; Armirotti, A; Romeo, E; Berteotti, A; Fiorelli, C; Tarozzo, G; Reggiani, A; Duranti, Andrea; Tarzia, Giorgio; Mor, M; Cavalli, A; Piomelli, D; Bandiera, T.
Synthesis and Structure–Activity Relationship Studies of O-Biphenyl-3-yl Carbamates as Peripherally Restricted Fatty Acid Amide Hydrolase Inhibitors
2013 MORENO SANZ, G; Duranti, Andrea; Melzig, L; Fiorelli, C; Ruda, Gf; Colombano, G; Mestichelli, Paola; Sanchini, Silvano; Tontini, Andrea; Mor, M; Bandiera, T; Scarpelli, R; Tarzia, Giorgio; Piomelli, D.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
SYNTHESIS AND EVALUATION OF SUGAR-BASED ALIPHATIC AND AROMATIC FATTY ACID ESTERS AS ANTIMICROBIAL AND ANTIBIOFILM AGENTS | 1-gen-2019 | Lucarini, Simone; Campana, Raffaella; Duranti, Andrea | |
Synthesis and Evaluation of Saccharide-Based Aliphatic and Aromatic Esters as Antimicrobial and Antibiofilm Agents | 1-gen-2019 | Campana, Raffaella; Merli, Alessio; Verboni, Michele; Biondo, Francesca; Favi, Gianfranco; Duranti, Andrea; Lucarini, Simone | |
Pharmacokinetics, pharmacodynamics and safety studies on URB 937, a peripherally restricted fatty acid amide hydrolase inhibitor, in rats | 1-gen-2019 | Vozella, Valentina; Ahmed, Faizy; Choobchian, Paoula; Merrill, Collin B.; Zibardi, Cristina; Tarzia, Giorgio; Mor, Marco; Duranti, Andrea; Tontini, Andrea; Rivara, Silvia; Piomelli, Daniele | |
Acute Reduction in Neonatal Brain Injury by Selective Blockage of CB1 and Activation of CB2 Receptors | 1-gen-2019 | Alonso-Alconada, D; Carloni, S; Duranti, A; Pintor-Rial, A; Alvarez, A; Hilario, E; Balduini, W | |
Lactose oleate as new biocompatible surfactant for pharmaceutical applications | 1-gen-2018 | Perinelli, D. R; Lucarini, S; Fagioli, L; Campana, R; Vllasaliu, D; Duranti, A; Casettari, L. | |
Synthesis, Structure-Activity Relationships and In Vitro Toxicity Profile of Lactose-Based Fatty Acid Monoesters as Possible Drug Permeability Enhancers | 1-gen-2018 | Lucarini, Simone; Fagioli, Laura; Cavanagh, Robert; Liang, Wanling; Perinelli, Diego Romano; Campana, Mario; Stolnik, Snjezana; Lam, Jenny K W; Casettari, Luca; Duranti, Andrea | |
The fatty acid amide hydrolase inhibitor URB597 modulates serotonin-dependent emotional behaviour, and serotonin1A and serotonin2A/C activity in the hippocampus | 1-gen-2016 | Bambico, Fr; Duranti, Andrea; Nobrega, Jn; Gobbi, G. | |
Unsaturated fatty acids lactose esters: cytotoxicity, permeability enhancement and antimicrobial activity | 1-gen-2016 | Lucarini, Simone; Fagioli, Laura; Campana, Raffaella; Cole, Hannah; Duranti, Andrea; Baffone, Wally; Vllasaliu, Driton; Casettari, Luca | |
Composition and Methods of Inhibiting N-Acylethanolamine-hydrolyzing Acid Amidase | 1-gen-2016 | Piomelli, D; Tarzia, Giorgio; Mor, M; Duranti, Andrea; Tontini, Andrea | |
Inhibition of anandamide hydrolysis enhances noradrenergic and GABAergic transmission in the prefrontal cortex and basolateral amygdala of rat subjected to acute swim stress | 1-gen-2015 | Besde, G; Romano, A; Tempesta, B; Lavecchia, Ma; Pace, L; Bellomo, A; Duranti, Andrea; MICIONI DI BONAVENTURA, Mv; Cifani, C; Cassano, T; Gaetani, S. | |
Chronic stimulation of the endogenous anandamide tone reduces cocaine-seeking and cue-induced relapse in rats | 1-gen-2015 | Chauvet, C; Nicolas, C; Thiriet, N; Lardeux, V; Duranti, Andrea; Solinas, M. | |
Anestetici locali (Cap. 14) | 1-gen-2015 | Duranti, Andrea | |
Derivatizzazione one-pot di indoli per la sintesi di triptofani, pirroloindoline, bis-indoli & co | 1-gen-2014 | Lucarini, Simone; Piersanti, Giovanni; Duranti, Andrea; Spadoni, Gilberto | |
Structural determinants of peripheral O-arylcarbamate FAAH inhibitors render them dual substrates for Abcb1 and Abcg2 and restrict their access to the brain | 1-gen-2014 | MORENO SANZ, G; Barrera, B; Armirotti, A; MANDRUP BERTOZZI, S; Prieto, Jg; Scarpelli, R; Duranti, Andrea; Tarzia, Giorgio; Bandiera, T; Merino, G; Piomelli, D. | |
Prior stimulation of the endocannabinoid system prevents methamphetamine-induced neurotoxicity in the striatum through activation of CB2 receptors | 1-gen-2014 | Nader, J; Rapino, C; Gennequin, B; Chavant, F; Francheteau, M; Makriyannis, A; Duranti, Andrea; Maccarrone, M; Solinas, M; Thiriet, N. | |
Stimulation of the endocannabinoid system prevents methamphetamine-induced neurotoxicity in mice | 1-gen-2013 | Thiriet, N; Nader, J; Rapino, C; Gennequin, B; Francheteau, M; Makryiannis, A; Duranti, Andrea; Maccarrone, M; Solinas, M. | |
Sintesi e studi di relazione struttura–attività/selettività su O-bifenil-3-ilcarbammati disostituiti quali inibitori periferici dell’enzima FAAH | 1-gen-2013 | Mestichelli, Paola; MORENO SANZ, G; Duranti, Andrea; Sanchini, Silvano; Tontini, Andrea; Lodola, A; Mor, M; Bandiera, T; Piomelli, D; Tarzia, Giorgio | |
O-Biphenyl-3-yl Carbamates as Peripheral FAAH Inhibitors: Synthesis and Structure–Activity (SAR) Relationship Studies | 1-gen-2013 | Mestichelli, Paola; MORENO SANZ, G; Duranti, Andrea; Sanchini, Silvano; Tontini, Andrea; Lodola, A; Mor, M; Bandiera, T; Piomelli, D; Tarzia, Giorgio | |
Synthesis and Structure–Activity Relationship (SAR) of 2-Methyl-4-oxo-3-oxetanyl Carbamic Acid Esters, a Class of Potent N-Acylethanolamine Acid Amidase (NAAA) Inhibitors | 1-gen-2013 | Ponzano, S; Bertozzi, F; Mengatto, L; Dionisi, M; Armirotti, A; Romeo, E; Berteotti, A; Fiorelli, C; Tarozzo, G; Reggiani, A; Duranti, Andrea; Tarzia, Giorgio; Mor, M; Cavalli, A; Piomelli, D; Bandiera, T. | |
Synthesis and Structure–Activity Relationship Studies of O-Biphenyl-3-yl Carbamates as Peripherally Restricted Fatty Acid Amide Hydrolase Inhibitors | 1-gen-2013 | MORENO SANZ, G; Duranti, Andrea; Melzig, L; Fiorelli, C; Ruda, Gf; Colombano, G; Mestichelli, Paola; Sanchini, Silvano; Tontini, Andrea; Mor, M; Bandiera, T; Scarpelli, R; Tarzia, Giorgio; Piomelli, D. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile