Sfoglia per Autore
Anandamide suppressess pain initiation through a peripheral endocannabinoid mechanism
2010 Clapper, Jr; MORENO SANZ, G; Russo, R; Guijarro, A; Vacondio, F; Duranti, Andrea; Tontini, Andrea; Sanchini, Silvano; Sciolino, Nr; Spradley, Jm; Hohmann, Ag; Calignano, A; Mor, M; Tarzia, Giorgio; Piomelli, D.
α-Acylamino-β-lactones as a new class of N-acylethanolamine-hydrolyzing acid amidase (NAAA) inhibitors: synthesis and structure–activity relationships
2009 Antonietti, Francesca; Battista, N; Duranti, Andrea; Lodola, A; Mor, M; Piomelli, D; Rivara, S; Solorzano, C; Tarzia, Giorgio; Tontini, Andrea; Zhu, C.
Antinociceptive effects of the brain-impermeant fatty-acid amide hydrolase inhibitor URB937
2009 Clapper, Jr; MORENO SANZ, G; Russo, R; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Calignano, A; Piomelli, D.
Composition and Methods of Inhibiting N-Acylethanolamine-hydrolyzing Acid Amidase
2009 Piomelli, D; Tarzia, Giorgio; Mor, M; Duranti, Andrea; Tontini, Andrea
Synthesis and Structure-Activity/Stability Relationships of Carbamate Inhibitors of the FAAH Enzyme
2009 Sanchini, Silvano; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Vacondio, F; Fioni, A; Lodola, A; Rivara, S; Mor, M; Clapper, J; Piomelli, D.
Synthesis and characterization of a peripherally restricted CB1 cannabinoid antagonist, URB447, that reduces feeding and body-weight gain in mice
2009 Loverme, J; Duranti, Andrea; Tontini, Andrea; Spadoni, Gilberto; Mor, M; Rivara, S; Stella, N; Xu, C; Tarzia, Giorgio; Piomelli, D.
Endocannabinoids in the Treatment of Mood Disorders: Evidence from Animal Models
2009 Bambico, Fr; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Gobbi, G.
Selective N-acylethanolamine-hydrolyzing acid amidase inhibition reveals a key role for endogenous palmitoylethanolamide in inflammation
2009 Solorzano, C; Zhu, C; Battista, N; Astarita, G; Lodola, A; Rivara, S; Mor, M; Russo, R; Maccarrone, M; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Cuzzocrea, S; Tarzia, Giorgio; Piomelli, D.
A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo
2009 Clapper, Jr; Vacondio, F; King, Ar; Duranti, Andrea; Tontini, Andrea; Silva, C; Sanchini, Silvano; Tarzia, Giorgio; Mor, M; Piomelli, D.
Structure–Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors: Chemical and Biological Stability
2009 Vacondio, F; Silva, C; Lodola, A; Fioni, A; Rivara, S; Duranti, Andrea; Tontini, Andrea; Sanchini, Silvano; Clapper, J; Piomelli, D; Mor, M; Tarzia, Giorgio
The collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity
2009 Valitutti, G; Duranti, Andrea; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P.
Synthesis and pharmacological characterization of URB447, a new cannabinoid receptor neutral antagonist
2008 Tontini, Andrea; Duranti, Andrea; Spadoni, Gilberto; Tarzia, Giorgio; Mor, M; Rivara, S; Loverme, J; Piomelli, D.
Inibitori dell’enzima NAAA (N-Acylethanolamine-Hydrolizing Acid Amidase) come nuovi agenti antinfiammatori
2008 Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Lodola, A; Rivara, S; Mor, M; Zhu, C; Solorzano, C; Piomelli, D.
Synthesis, QSAR and Pharmacological Evaluation of Alkylcarbamic Acid Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: A Novel Approach to Antianxiety and Analgesic Agents
2008 Tarzia, Giorgio; Duranti, Andrea; Tontini, Andrea; Rivara, S; Mor, M; Piomelli, D.
Sintesi e studi di relazione struttura-attività/stabilità di carbammati inibitori dell’enzima FAAH
2008 Sanchini, Silvano; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Vacondio, F; Fioni, A; Lodola, A; Rivara, S; Mor, M; Clapper, J; Piomelli, D.
Novel carbamate-based fatty-acid amide hydrolase inhibitors with enhanced stability and selectivity
2008 Clapper, Jr; Vacondio, F; King, Ar; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Piomelli, D.
Inhibitors of lysosomal lipid amidase NAAA
2008 Zhu, C; Solorzano, C; Battista, N; Lodola, A; Rivara, S; Mor, M; Russo, R; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Cuzzocrea, S; Tarzia, Giorgio; Piomelli, D.
The Collisional Behavior of ESI-Generated Protonated Molecules of Some Carbamate Bioisosters and its Relationship with their Biological Activity
2008 Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P.
Cannabinoids Modify Hippocampal Serotonergic Transmission
2008 Hattan, P; Bambico, F; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Walker, Cd; Gobbi, G.
Application of computational models to the design of new inhibitors of fatty acid amide hydrolase
2008 Lodola, A; Mulholland, Aj; Rivara, S; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Piomelli, D; Mor, M.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Anandamide suppressess pain initiation through a peripheral endocannabinoid mechanism | 1-gen-2010 | Clapper, Jr; MORENO SANZ, G; Russo, R; Guijarro, A; Vacondio, F; Duranti, Andrea; Tontini, Andrea; Sanchini, Silvano; Sciolino, Nr; Spradley, Jm; Hohmann, Ag; Calignano, A; Mor, M; Tarzia, Giorgio; Piomelli, D. | |
α-Acylamino-β-lactones as a new class of N-acylethanolamine-hydrolyzing acid amidase (NAAA) inhibitors: synthesis and structure–activity relationships | 1-gen-2009 | Antonietti, Francesca; Battista, N; Duranti, Andrea; Lodola, A; Mor, M; Piomelli, D; Rivara, S; Solorzano, C; Tarzia, Giorgio; Tontini, Andrea; Zhu, C. | |
Antinociceptive effects of the brain-impermeant fatty-acid amide hydrolase inhibitor URB937 | 1-gen-2009 | Clapper, Jr; MORENO SANZ, G; Russo, R; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Calignano, A; Piomelli, D. | |
Composition and Methods of Inhibiting N-Acylethanolamine-hydrolyzing Acid Amidase | 1-gen-2009 | Piomelli, D; Tarzia, Giorgio; Mor, M; Duranti, Andrea; Tontini, Andrea | |
Synthesis and Structure-Activity/Stability Relationships of Carbamate Inhibitors of the FAAH Enzyme | 1-gen-2009 | Sanchini, Silvano; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Vacondio, F; Fioni, A; Lodola, A; Rivara, S; Mor, M; Clapper, J; Piomelli, D. | |
Synthesis and characterization of a peripherally restricted CB1 cannabinoid antagonist, URB447, that reduces feeding and body-weight gain in mice | 1-gen-2009 | Loverme, J; Duranti, Andrea; Tontini, Andrea; Spadoni, Gilberto; Mor, M; Rivara, S; Stella, N; Xu, C; Tarzia, Giorgio; Piomelli, D. | |
Endocannabinoids in the Treatment of Mood Disorders: Evidence from Animal Models | 1-gen-2009 | Bambico, Fr; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Gobbi, G. | |
Selective N-acylethanolamine-hydrolyzing acid amidase inhibition reveals a key role for endogenous palmitoylethanolamide in inflammation | 1-gen-2009 | Solorzano, C; Zhu, C; Battista, N; Astarita, G; Lodola, A; Rivara, S; Mor, M; Russo, R; Maccarrone, M; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Cuzzocrea, S; Tarzia, Giorgio; Piomelli, D. | |
A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo | 1-gen-2009 | Clapper, Jr; Vacondio, F; King, Ar; Duranti, Andrea; Tontini, Andrea; Silva, C; Sanchini, Silvano; Tarzia, Giorgio; Mor, M; Piomelli, D. | |
Structure–Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors: Chemical and Biological Stability | 1-gen-2009 | Vacondio, F; Silva, C; Lodola, A; Fioni, A; Rivara, S; Duranti, Andrea; Tontini, Andrea; Sanchini, Silvano; Clapper, J; Piomelli, D; Mor, M; Tarzia, Giorgio | |
The collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity | 1-gen-2009 | Valitutti, G; Duranti, Andrea; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P. | |
Synthesis and pharmacological characterization of URB447, a new cannabinoid receptor neutral antagonist | 1-gen-2008 | Tontini, Andrea; Duranti, Andrea; Spadoni, Gilberto; Tarzia, Giorgio; Mor, M; Rivara, S; Loverme, J; Piomelli, D. | |
Inibitori dell’enzima NAAA (N-Acylethanolamine-Hydrolizing Acid Amidase) come nuovi agenti antinfiammatori | 1-gen-2008 | Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Lodola, A; Rivara, S; Mor, M; Zhu, C; Solorzano, C; Piomelli, D. | |
Synthesis, QSAR and Pharmacological Evaluation of Alkylcarbamic Acid Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: A Novel Approach to Antianxiety and Analgesic Agents | 1-gen-2008 | Tarzia, Giorgio; Duranti, Andrea; Tontini, Andrea; Rivara, S; Mor, M; Piomelli, D. | |
Sintesi e studi di relazione struttura-attività/stabilità di carbammati inibitori dell’enzima FAAH | 1-gen-2008 | Sanchini, Silvano; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Vacondio, F; Fioni, A; Lodola, A; Rivara, S; Mor, M; Clapper, J; Piomelli, D. | |
Novel carbamate-based fatty-acid amide hydrolase inhibitors with enhanced stability and selectivity | 1-gen-2008 | Clapper, Jr; Vacondio, F; King, Ar; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Piomelli, D. | |
Inhibitors of lysosomal lipid amidase NAAA | 1-gen-2008 | Zhu, C; Solorzano, C; Battista, N; Lodola, A; Rivara, S; Mor, M; Russo, R; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Cuzzocrea, S; Tarzia, Giorgio; Piomelli, D. | |
The Collisional Behavior of ESI-Generated Protonated Molecules of Some Carbamate Bioisosters and its Relationship with their Biological Activity | 1-gen-2008 | Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P. | |
Cannabinoids Modify Hippocampal Serotonergic Transmission | 1-gen-2008 | Hattan, P; Bambico, F; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Walker, Cd; Gobbi, G. | |
Application of computational models to the design of new inhibitors of fatty acid amide hydrolase | 1-gen-2008 | Lodola, A; Mulholland, Aj; Rivara, S; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Piomelli, D; Mor, M. |
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