Sfoglia per Autore
Synthesis and Quantitative Structure–Activity Relationship of Fatty Acid Amide Hydrolase Inhibitors: Modulation at the N-Portion of Biphenyl-3-yl Alkylcarbamates
2008 Mor, M; Lodola, A; Rivara, S; Vacondio, F; Duranti, Andrea; Tontini, Andrea; Sanchini, S; Piersanti, Giovanni; Tarzia, Giorgio; Clapper, Jr; King, Ar; Piomelli, D.
Novel carbamate-based fatty-acid amide hydrolase inhibitors with enhanced stability and selectivity
2008 Clapper, Jr; Vacondio, F; King, Ar; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Piomelli, D.
Quantitative Structure-Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors
2008 Fioni, A; Vacondio, F; Mor, M; Silva, C; Lodola, A; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Piomelli, D.
Inhibitors of lysosomal lipid amidase NAAA
2008 Zhu, C; Solorzano, C; Battista, N; Lodola, A; Rivara, S; Mor, M; Russo, R; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Cuzzocrea, S; Tarzia, Giorgio; Piomelli, D.
The Collisional Behavior of ESI-Generated Protonated Molecules of Some Carbamate Bioisosters and its Relationship with their Biological Activity
2008 Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P.
Cannabinoids Modify Hippocampal Serotonergic Transmission
2008 Hattan, P; Bambico, F; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Walker, Cd; Gobbi, G.
Synthesis and Biological Activity of Monoacylglycerol Lipase (MGL) Inhibitor URB602 and its Analogs
2007 Tontini, Andrea; King, A; Clapper, J; Duranti, Andrea; Lodola, A; Mor, M; Rivara, S; Rosengarth, A; Tarzia, Giorgio; Piomelli, D.
Effect of the Selective Fatty Acid Amide Hydrolase Inhibitor URB597 on Ethanol Abuse Related Behaviours in the Rat
2007 Braconi, S; Piomelli, D; Duranti, Andrea; Tonini, A; Tarzia, Giorgio; Cannella, N; Massi, M; Ciccocioppo, R; Cippitelli, A; Tontini, Andrea
Identification of a Bioactive Impurity in a Commercial Sample of 6-Methyl-2-p-tolylaminobenzo[d][1,3]oxazin-4-one (URB754)
2007 Tarzia, Giorgio; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Mor, M; Rivara, S; Traldi, P; Astarita, G; King, A; Clapper, J; Piomelli, D.
Correlation between energetics of collisionally activated decompositions, interaction energy and biological potency of carbamates FAAH inhibitors
2007 Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P.
URB602 Inhibits Monoacylglycerol Lipase and Selectively Blocks 2-Arachidonoylglycerol Degradation in Intact Brain Slices
2007 King, Ar; Duranti, Andrea; Tontini, Andrea; Rivara, S; Rosengarth, A; Clapper, Jr; Astarita, G; Geaga, Ja; Luecke, H; Mor, M; Tarzia, Giorgio; Piomelli, D.
The Fatty Acid Amide Hydrolase Inhibitor URB597 (Cyclohexylcarbamic Acid 3’-Carbamoylbiphenyl-3-yl Ester) Reduces Neuropathic Pain after Oral Administration in Mice
2007 Russo, R; Loverme, J; LA RANA, G; Compton, Tr; Parrott, J; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Calignano, A; Piomelli, D.
Antidepressant-like Activity of the Fatty Acid Amide Hydrolase Inhibitor URB597 in a Rat Model of Chronic Mild Stress
2007 Bortolato, M; Mangieri, R; Fu, J; Kim, Jh; Arguello, O; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Piomelli, D.
QSAR and molecular modelling investigations of a new series of alkyl carbamic acid aryl ester inhibitors of fatty acid amide hydrolase
2007 Lodola, A; Rivara, S; Mor, M; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Piomelli, D.
Mass Spectrometry and Pharmacology Activity: The Case of Carbamic Analogs
2007 Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P.
Characterization of monoacylglycerol lipase (MGL) inhibitor URB602
2007 King, Ar; Rosengarth, A; Clapper, J; Duranti, Andrea; Tontini, Andrea; Mor, M; Rivara, S; Tarzia, Giorgio; Piomelli, D.
FAAH and MGL Inhibitors. Design and Therapeutic Implications
2006 Tarzia, Giorgio; Tontini, Andrea; Piomelli, D; Mor, M; Duranti, Andrea; Antonietti, F.
Methods, Compositions, and Other Compounds for Modulation of Monoacylglycerol Lipase Pain, and Stress-related Disorders
2006 Piomelli, D; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Hohmann, A.
Interazione tra sistema cannabinoide e serotoninergico: implicazioni farmacologiche e cliniche per il trattamento della depressione
2006 Bambico, Fr; Katz, N; Nguyen, N. T.; Ciszek, A; Debonnel, G; Mor, M; Tontini, Andrea; Duranti, Andrea; Tarzia, Giorgio; Piomelli, D; Gobbi, G.
Reactivity, metabolic stability and interaction at the catalytic site for carbamate inhibitors of FAAH
2006 Mor, M; Lodola, A; Vacondio, F; Silva, C; Rivara, S; Tontini, Andrea; Duranti, Andrea; Tarzia, Giorgio; Piomelli, D.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and Quantitative Structure–Activity Relationship of Fatty Acid Amide Hydrolase Inhibitors: Modulation at the N-Portion of Biphenyl-3-yl Alkylcarbamates | 1-gen-2008 | Mor, M; Lodola, A; Rivara, S; Vacondio, F; Duranti, Andrea; Tontini, Andrea; Sanchini, S; Piersanti, Giovanni; Tarzia, Giorgio; Clapper, Jr; King, Ar; Piomelli, D. | |
Novel carbamate-based fatty-acid amide hydrolase inhibitors with enhanced stability and selectivity | 1-gen-2008 | Clapper, Jr; Vacondio, F; King, Ar; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Piomelli, D. | |
Quantitative Structure-Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors | 1-gen-2008 | Fioni, A; Vacondio, F; Mor, M; Silva, C; Lodola, A; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Piomelli, D. | |
Inhibitors of lysosomal lipid amidase NAAA | 1-gen-2008 | Zhu, C; Solorzano, C; Battista, N; Lodola, A; Rivara, S; Mor, M; Russo, R; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Cuzzocrea, S; Tarzia, Giorgio; Piomelli, D. | |
The Collisional Behavior of ESI-Generated Protonated Molecules of Some Carbamate Bioisosters and its Relationship with their Biological Activity | 1-gen-2008 | Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P. | |
Cannabinoids Modify Hippocampal Serotonergic Transmission | 1-gen-2008 | Hattan, P; Bambico, F; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Walker, Cd; Gobbi, G. | |
Synthesis and Biological Activity of Monoacylglycerol Lipase (MGL) Inhibitor URB602 and its Analogs | 1-gen-2007 | Tontini, Andrea; King, A; Clapper, J; Duranti, Andrea; Lodola, A; Mor, M; Rivara, S; Rosengarth, A; Tarzia, Giorgio; Piomelli, D. | |
Effect of the Selective Fatty Acid Amide Hydrolase Inhibitor URB597 on Ethanol Abuse Related Behaviours in the Rat | 1-gen-2007 | Braconi, S; Piomelli, D; Duranti, Andrea; Tonini, A; Tarzia, Giorgio; Cannella, N; Massi, M; Ciccocioppo, R; Cippitelli, A; Tontini, Andrea | |
Identification of a Bioactive Impurity in a Commercial Sample of 6-Methyl-2-p-tolylaminobenzo[d][1,3]oxazin-4-one (URB754) | 1-gen-2007 | Tarzia, Giorgio; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Mor, M; Rivara, S; Traldi, P; Astarita, G; King, A; Clapper, J; Piomelli, D. | |
Correlation between energetics of collisionally activated decompositions, interaction energy and biological potency of carbamates FAAH inhibitors | 1-gen-2007 | Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P. | |
URB602 Inhibits Monoacylglycerol Lipase and Selectively Blocks 2-Arachidonoylglycerol Degradation in Intact Brain Slices | 1-gen-2007 | King, Ar; Duranti, Andrea; Tontini, Andrea; Rivara, S; Rosengarth, A; Clapper, Jr; Astarita, G; Geaga, Ja; Luecke, H; Mor, M; Tarzia, Giorgio; Piomelli, D. | |
The Fatty Acid Amide Hydrolase Inhibitor URB597 (Cyclohexylcarbamic Acid 3’-Carbamoylbiphenyl-3-yl Ester) Reduces Neuropathic Pain after Oral Administration in Mice | 1-gen-2007 | Russo, R; Loverme, J; LA RANA, G; Compton, Tr; Parrott, J; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Calignano, A; Piomelli, D. | |
Antidepressant-like Activity of the Fatty Acid Amide Hydrolase Inhibitor URB597 in a Rat Model of Chronic Mild Stress | 1-gen-2007 | Bortolato, M; Mangieri, R; Fu, J; Kim, Jh; Arguello, O; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Piomelli, D. | |
QSAR and molecular modelling investigations of a new series of alkyl carbamic acid aryl ester inhibitors of fatty acid amide hydrolase | 1-gen-2007 | Lodola, A; Rivara, S; Mor, M; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Piomelli, D. | |
Mass Spectrometry and Pharmacology Activity: The Case of Carbamic Analogs | 1-gen-2007 | Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P. | |
Characterization of monoacylglycerol lipase (MGL) inhibitor URB602 | 1-gen-2007 | King, Ar; Rosengarth, A; Clapper, J; Duranti, Andrea; Tontini, Andrea; Mor, M; Rivara, S; Tarzia, Giorgio; Piomelli, D. | |
FAAH and MGL Inhibitors. Design and Therapeutic Implications | 1-gen-2006 | Tarzia, Giorgio; Tontini, Andrea; Piomelli, D; Mor, M; Duranti, Andrea; Antonietti, F. | |
Methods, Compositions, and Other Compounds for Modulation of Monoacylglycerol Lipase Pain, and Stress-related Disorders | 1-gen-2006 | Piomelli, D; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Hohmann, A. | |
Interazione tra sistema cannabinoide e serotoninergico: implicazioni farmacologiche e cliniche per il trattamento della depressione | 1-gen-2006 | Bambico, Fr; Katz, N; Nguyen, N. T.; Ciszek, A; Debonnel, G; Mor, M; Tontini, Andrea; Duranti, Andrea; Tarzia, Giorgio; Piomelli, D; Gobbi, G. | |
Reactivity, metabolic stability and interaction at the catalytic site for carbamate inhibitors of FAAH | 1-gen-2006 | Mor, M; Lodola, A; Vacondio, F; Silva, C; Rivara, S; Tontini, Andrea; Duranti, Andrea; Tarzia, Giorgio; Piomelli, D. |
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