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Selective Melatonin MT2 receptor ligands relieve neuropathic pain through modulation of brainstem descending antinociceptive pathways 1-gen-2015 M., Lopez Canul; E., Palazzo; S., Dominguez Lopez; L., Luongo; B., Lacoste; S., Comai; D., Angeloni; F., Fraschini; S., Boccella; Spadoni, Gilberto; Bedini, Annalida; G., Tarzia; S., Maione; V., Granado Sotos; G., Gobbi
Antidepressant-like activity and cardioprotective effects of fatty acid amide hydrolase inhibitor URB694 in socially stressed Wistar Kyoto rats 1-gen-2015 Sgoifo, A.; Carnevali, L.; Vacondio, F.; Rossi, S.; Callegari, S.; Macchi, E.; Spadoni, Gilberto; Bedini, Annalida; Rivara, S.; Mor, M.
Synthetic Melatonin Receptor Ligands 1-gen-2014 S., Rivara; M., Mor; Bedini, Annalida; Spadoni, Gilberto
Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moieties 1-gen-2014 Spadoni, Gilberto; Bedini, Annalida; Bartolucci, Silvia; Pala, D.; Mor, M.; Riccioni, T.; Borsini, F.; Cabri, W.; Celona, D.; Marzi, M.; Tarzia, Giorgio; Rivara, S.; Minetti, P.
Melatonin, non-selective MT1/MT2 and selective MT2 receptor agonists: differential effects on the 24-hr vigilance states 1-gen-2014 Ochoa Sanchez, R.; Comai, S.; Spadoni, Gilberto; Bedini, Annalida; Tarzia, Giorgio; Gobbi, G.
Synthesis and Characterization of New Bivalent Agents as Melatonin- and Histamine H3-Ligands 1-gen-2014 Pala, D.; Scalvini, L.; Lodola, A.; Mor, M.; Flammini, L.; Barocelli, E.; Lucini, V.; Scaglione, F.; Bartolucci, Silvia; Bedini, Annalida; Rivara, S.; Spadoni, Gilberto
Homology models of melatonin receptors: challenges and recent advances 1-gen-2013 D., Pala; A., Lodola; Bedini, Annalida; Spadoni, Gilberto; S., Rivara
Synthesis and Configuration Determination of All Enantiopure Stereoisomers of the Melatonin Receptor Ligand 4-Phenyl-2-propionamidotetralin using an Expedient Optical Resolution of 4-Phenyl-2-tetralone 1-gen-2012 Lucarini, Simone; Bartolucci, Silvia; Bedini, Annalida; Gatti, G.; Orlando, Pierfrancesco; Piersanti, Giovanni; Spadoni, Gilberto
Synthesis of Tryptamine Derivatives via a Direct, One-Pot Reductive Alkylation of Indoles 1-gen-2012 Marika, Righi; Francesca, Topi; Bartolucci, Silvia; Bedini, Annalida; Piersanti, Giovanni; Spadoni, Gilberto
MT1-Selective Melatonin Receptor Ligands: Synthesis, Pharmacological Evaluation, and Molecular Dynamics Investigation of N-{[(3-O-Substituted)anilino]alkyl}amides 1-gen-2012 Rivara, S.; Pala, D.; Lodola, A.; Mor, M.; Lucini, V.; Dugnani, S.; Scaglione, F.; Bedini, Annalida; Lucarini, Simone; Tarzia, Giorgio; Spadoni, Gilberto
Anxiolytic effects of the melatonin MT2 receptor partial agonist UCM765: Comparison with melatonin and diazepam 1-gen-2012 Ochoa Sanchez, R.; Rainer, Q.; Comai, S.; Spadoni, Gilberto; Bedini, Annalida; Rivara, S.; Fraschini, F.; Mor, M.; Tarzia, Giorgio; Gobbi, G.
Toward the Definition of Stereochemical Requirements for MT(2)-Selective Antagonists and Partial Agonists by Studying 4-Phenyl-2-propionamidotetralin Derivatives 1-gen-2011 Bedini, Annalida; Lucarini, Simone; Spadoni, Gilberto; Tarzia, Giorgio; Scaglione, F; Dugnani, S; Pannacci, M; Lucini, V; Carmi, C; Pala, D; Rivara, S; Mor, M.
Direct, One-Pot Reductive Alkylation of Anilines with Functionalized Acetals Mediated by Triethylsilane and TFA. Straightforward Route for Unsymmetrically Substituted Ethylenediamine 1-gen-2011 M., Righi; Bedini, Annalida; Piersanti, Giovanni; F., Romagnoli; Spadoni, Gilberto
Bivalent Ligand Approach on N-[2-[(3-methoxyphenyl)methylamino]ethyl]acetamide. Synthesis, Binding Affinity and Intrinsic Acivity for MT(1) and MT(2) melatonin Receptors. 1-gen-2011 Spadoni, Gilberto; Bedini, Annalida; Orlando, Pierfrancesco; Lucarini, Simone; Tarzia, Giorgio; Mor, M.; Rivara, S.; Lucini, V.; Pannacci, M.; Scaglione, F.
Promotion of non-rapid eye movement sleep and activation of reticular thalamic neurons by a novel MT2 melatonin receptor ligand 1-gen-2011 Ochoa Sanchez, R; Comai, S; Lacoste, B; Bambico, Fr; Dominguez Lopez, S; Spadoni, Gilberto; Rivara, S; Bedini, Annalida; Angeloni, D; Fraschini, F; Mor, M; Tarzia, Giorgio; Descarries, L; Gobbi, G.
Melatonin receptor agonists: new options for insomnia and depression treatment 1-gen-2011 Spadoni, Gilberto; Bedini, Annalida; Rivara, S; Mor, M.
Diastereo- and enantioselective hydrogenation of a challenging enamide derived from 4-phenyl-2-tetralone: an appealing shortcut towards enantiopure cis-2-aminotetraline derivatives 1-gen-2010 Lucarini, Simone; Alessi, M; Bedini, Annalida; Giorgini, G; Piersanti, Giovanni; Spadoni, Gilberto
Recent advances in the development of melatonin MT1 and MT2 receptor agonists 1-gen-2010 Mor, M; Rivara, S; Pala, D; Bedini, Annalida; Spadoni, Gilberto; Tarzia, Giorgio
N-(Anilinoethyl)amides: design and synthesis of metabolically stable, selective melatonin receptor ligands. 1-gen-2009 Rivara, S; Vacondio, F; Fioni, A; Silva, C; Carmi, C; Mor, M; Lucini, V; Pannacci, M; Caronno, A; Scaglione, F; Gobbi, G; Spadoni, Gilberto; Bedini, Annalida; Orlando, ; Lucarini, Simone; Tarzia, Giorgio
Rapid and transient stimulation of intracellular reactive oxygen species by melatonin in normal tumor leukocytes, Toxicology and apllied Pharmacology, 239(1), 37-45 (2009) 1-gen-2009 Radogna, F; Paternoster, L; DE NICOLA, M; Cerella, C; Ammendola, S; Bedini, Annalida; Tarzia, Giorgio; Aquilano, K; Ciriolo, M; Ghibelli, L.
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