Sfoglia per Autore
Composition and Methods of Inhibiting N-Acylethanolamine-hydrolyzing Acid Amidase
2009 Piomelli, D; Tarzia, Giorgio; Mor, M; Duranti, Andrea; Tontini, Andrea
Synthesis and Structure-Activity/Stability Relationships of Carbamate Inhibitors of the FAAH Enzyme
2009 Sanchini, Silvano; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Vacondio, F; Fioni, A; Lodola, A; Rivara, S; Mor, M; Clapper, J; Piomelli, D.
Derivatives of triazoly-imidazopyridine useful as ligands of the adenosine A2a receptor ant their use as medicaments
2009 Tarzia, Giorgio; Piersanti, Giovanni; Giorgi, Luca; Patrizia, Minetti; MARIA A., DI CESARE; Grazia, Gallo; Fabrizio, Giorgi
Rapid and transient stimulation of intracellular reactive oxygen species by melatonin in normal tumor leukocytes, Toxicology and apllied Pharmacology, 239(1), 37-45 (2009)
2009 Radogna, F; Paternoster, L; DE NICOLA, M; Cerella, C; Ammendola, S; Bedini, Annalida; Tarzia, Giorgio; Aquilano, K; Ciriolo, M; Ghibelli, L.
The collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity
2009 Valitutti, G; Duranti, Andrea; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P.
A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo
2009 Clapper, Jr; Vacondio, F; King, Ar; Duranti, Andrea; Tontini, Andrea; Silva, C; Sanchini, Silvano; Tarzia, Giorgio; Mor, M; Piomelli, D.
Structure–Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors: Chemical and Biological Stability
2009 Vacondio, F; Silva, C; Lodola, A; Fioni, A; Rivara, S; Duranti, Andrea; Tontini, Andrea; Sanchini, Silvano; Clapper, J; Piomelli, D; Mor, M; Tarzia, Giorgio
Endocannabinoids in the Treatment of Mood Disorders: Evidence from Animal Models
2009 Bambico, Fr; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Gobbi, G.
N-(Anilinoethyl)amides: design and synthesis of metabolically stable, selective melatonin receptor ligands.
2009 Rivara, S; Vacondio, F; Fioni, A; Silva, C; Carmi, C; Mor, M; Lucini, V; Pannacci, M; Caronno, A; Scaglione, F; Gobbi, G; Spadoni, Gilberto; Bedini, Annalida; Orlando, ; Lucarini, Simone; Tarzia, Giorgio
Selective N-acylethanolamine-hydrolyzing acid amidase inhibition reveals a key role for endogenous palmitoylethanolamide in inflammation
2009 Solorzano, C; Zhu, C; Battista, N; Astarita, G; Lodola, A; Rivara, S; Mor, M; Russo, R; Maccarrone, M; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Cuzzocrea, S; Tarzia, Giorgio; Piomelli, D.
Synthesis and characterization of a peripherally restricted CB1 cannabinoid antagonist, URB447, that reduces feeding and body-weight gain in mice
2009 Loverme, J; Duranti, Andrea; Tontini, Andrea; Spadoni, Gilberto; Mor, M; Rivara, S; Stella, N; Xu, C; Tarzia, Giorgio; Piomelli, D.
Medicinal chemistry: defining itself
2008 Metternich, R; Tarzia, Giorgio
Identification of productive inhibitor binding orientation in fatty acid amide hydrolase (FAAH) by QM/MM mechanistic modeling
2008 Lodola, A; Mor, M; Rivara, S; Christov, C; Tarzia, Giorgio; Piomelli, D; Mulholland, A. J.
Synthesis and pharmacological characterization of URB447, a new cannabinoid receptor neutral antagonist
2008 Tontini, Andrea; Duranti, Andrea; Spadoni, Gilberto; Tarzia, Giorgio; Mor, M; Rivara, S; Loverme, J; Piomelli, D.
Synthesis, QSAR and Pharmacological Evaluation of Alkylcarbamic Acid Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: A Novel Approach to Antianxiety and Analgesic Agents
2008 Tarzia, Giorgio; Duranti, Andrea; Tontini, Andrea; Rivara, S; Mor, M; Piomelli, D.
Sintesi e studi di relazione struttura-attività/stabilità di carbammati inibitori dell’enzima FAAH
2008 Sanchini, Silvano; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Vacondio, F; Fioni, A; Lodola, A; Rivara, S; Mor, M; Clapper, J; Piomelli, D.
Novel carbamate-based fatty-acid amide hydrolase inhibitors with enhanced stability and selectivity
2008 Clapper, Jr; Vacondio, F; King, Ar; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Piomelli, D.
Inhibitors of lysosomal lipid amidase NAAA
2008 Zhu, C; Solorzano, C; Battista, N; Lodola, A; Rivara, S; Mor, M; Russo, R; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Cuzzocrea, S; Tarzia, Giorgio; Piomelli, D.
The Collisional Behavior of ESI-Generated Protonated Molecules of Some Carbamate Bioisosters and its Relationship with their Biological Activity
2008 Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P.
Cannabinoids Modify Hippocampal Serotonergic Transmission
2008 Hattan, P; Bambico, F; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Walker, Cd; Gobbi, G.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Composition and Methods of Inhibiting N-Acylethanolamine-hydrolyzing Acid Amidase | 1-gen-2009 | Piomelli, D; Tarzia, Giorgio; Mor, M; Duranti, Andrea; Tontini, Andrea | |
Synthesis and Structure-Activity/Stability Relationships of Carbamate Inhibitors of the FAAH Enzyme | 1-gen-2009 | Sanchini, Silvano; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Vacondio, F; Fioni, A; Lodola, A; Rivara, S; Mor, M; Clapper, J; Piomelli, D. | |
Derivatives of triazoly-imidazopyridine useful as ligands of the adenosine A2a receptor ant their use as medicaments | 1-gen-2009 | Tarzia, Giorgio; Piersanti, Giovanni; Giorgi, Luca; Patrizia, Minetti; MARIA A., DI CESARE; Grazia, Gallo; Fabrizio, Giorgi | |
Rapid and transient stimulation of intracellular reactive oxygen species by melatonin in normal tumor leukocytes, Toxicology and apllied Pharmacology, 239(1), 37-45 (2009) | 1-gen-2009 | Radogna, F; Paternoster, L; DE NICOLA, M; Cerella, C; Ammendola, S; Bedini, Annalida; Tarzia, Giorgio; Aquilano, K; Ciriolo, M; Ghibelli, L. | |
The collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity | 1-gen-2009 | Valitutti, G; Duranti, Andrea; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P. | |
A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo | 1-gen-2009 | Clapper, Jr; Vacondio, F; King, Ar; Duranti, Andrea; Tontini, Andrea; Silva, C; Sanchini, Silvano; Tarzia, Giorgio; Mor, M; Piomelli, D. | |
Structure–Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors: Chemical and Biological Stability | 1-gen-2009 | Vacondio, F; Silva, C; Lodola, A; Fioni, A; Rivara, S; Duranti, Andrea; Tontini, Andrea; Sanchini, Silvano; Clapper, J; Piomelli, D; Mor, M; Tarzia, Giorgio | |
Endocannabinoids in the Treatment of Mood Disorders: Evidence from Animal Models | 1-gen-2009 | Bambico, Fr; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Gobbi, G. | |
N-(Anilinoethyl)amides: design and synthesis of metabolically stable, selective melatonin receptor ligands. | 1-gen-2009 | Rivara, S; Vacondio, F; Fioni, A; Silva, C; Carmi, C; Mor, M; Lucini, V; Pannacci, M; Caronno, A; Scaglione, F; Gobbi, G; Spadoni, Gilberto; Bedini, Annalida; Orlando, ; Lucarini, Simone; Tarzia, Giorgio | |
Selective N-acylethanolamine-hydrolyzing acid amidase inhibition reveals a key role for endogenous palmitoylethanolamide in inflammation | 1-gen-2009 | Solorzano, C; Zhu, C; Battista, N; Astarita, G; Lodola, A; Rivara, S; Mor, M; Russo, R; Maccarrone, M; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Cuzzocrea, S; Tarzia, Giorgio; Piomelli, D. | |
Synthesis and characterization of a peripherally restricted CB1 cannabinoid antagonist, URB447, that reduces feeding and body-weight gain in mice | 1-gen-2009 | Loverme, J; Duranti, Andrea; Tontini, Andrea; Spadoni, Gilberto; Mor, M; Rivara, S; Stella, N; Xu, C; Tarzia, Giorgio; Piomelli, D. | |
Medicinal chemistry: defining itself | 1-gen-2008 | Metternich, R; Tarzia, Giorgio | |
Identification of productive inhibitor binding orientation in fatty acid amide hydrolase (FAAH) by QM/MM mechanistic modeling | 1-gen-2008 | Lodola, A; Mor, M; Rivara, S; Christov, C; Tarzia, Giorgio; Piomelli, D; Mulholland, A. J. | |
Synthesis and pharmacological characterization of URB447, a new cannabinoid receptor neutral antagonist | 1-gen-2008 | Tontini, Andrea; Duranti, Andrea; Spadoni, Gilberto; Tarzia, Giorgio; Mor, M; Rivara, S; Loverme, J; Piomelli, D. | |
Synthesis, QSAR and Pharmacological Evaluation of Alkylcarbamic Acid Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: A Novel Approach to Antianxiety and Analgesic Agents | 1-gen-2008 | Tarzia, Giorgio; Duranti, Andrea; Tontini, Andrea; Rivara, S; Mor, M; Piomelli, D. | |
Sintesi e studi di relazione struttura-attività/stabilità di carbammati inibitori dell’enzima FAAH | 1-gen-2008 | Sanchini, Silvano; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Vacondio, F; Fioni, A; Lodola, A; Rivara, S; Mor, M; Clapper, J; Piomelli, D. | |
Novel carbamate-based fatty-acid amide hydrolase inhibitors with enhanced stability and selectivity | 1-gen-2008 | Clapper, Jr; Vacondio, F; King, Ar; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Piomelli, D. | |
Inhibitors of lysosomal lipid amidase NAAA | 1-gen-2008 | Zhu, C; Solorzano, C; Battista, N; Lodola, A; Rivara, S; Mor, M; Russo, R; Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Cuzzocrea, S; Tarzia, Giorgio; Piomelli, D. | |
The Collisional Behavior of ESI-Generated Protonated Molecules of Some Carbamate Bioisosters and its Relationship with their Biological Activity | 1-gen-2008 | Valitutti, G; Duranti, Andrea; Lodola, A; Mor, M; Piersanti, Giovanni; Piomelli, D; Rivara, S; Tontini, Andrea; Tarzia, Giorgio; Traldi, P. | |
Cannabinoids Modify Hippocampal Serotonergic Transmission | 1-gen-2008 | Hattan, P; Bambico, F; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Walker, Cd; Gobbi, G. |
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