Sfoglia per Autore
Synthesis, QSAR and Pharmacological Evaluation of Alkylcarbamic Acid Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: A Novel Approach to Antianxiety and Analgesic Agents
2008 Tarzia, Giorgio; Duranti, Andrea; Tontini, Andrea; Rivara, S; Mor, M; Piomelli, D.
Quantitative Structure-Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors
2008 Fioni, A; Vacondio, F; Mor, M; Silva, C; Lodola, A; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Piomelli, D.
Design and structure-activity relationships of subtype selective melatonin receptor ligands.
2008 Rivara, S; Mor, M; Lodola, A; Spadoni, Gilberto; Bedini, Annalida; Tarzia, Giorgio; Lucini, V; Gobbi, G.
Selective increase of Slow Wave Sleep (SWS) by melatonin 2 receptors.
2008 OCHOA SANCHEZ, R; Spadoni, Gilberto; Bedini, Annalida; Mor, M; Rivara, S; Fraschini, F; Tarzia, Giorgio; Gobbi, G.
Sintesi e studi di relazione struttura-attività/stabilità di carbammati inibitori dell’enzima FAAH
2008 Sanchini, Silvano; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Vacondio, F; Fioni, A; Lodola, A; Rivara, S; Mor, M; Clapper, J; Piomelli, D.
Gordon Conference
2008 Bedini, Annalida; Spadoni, Gilberto; Tarzia, Giorgio; Gobbi, G; Mor, M; Rivara, S.
Inibitori dell’enzima NAAA (N-Acylethanolamine-Hydrolizing Acid Amidase) come nuovi agenti antinfiammatori
2008 Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Lodola, A; Rivara, S; Mor, M; Zhu, C; Solorzano, C; Piomelli, D.
Differences between direct cannabinoid agonists and FAAH inhibitors on antidepressant-like behavioural and serotonin-modulatory activity
2008 Bambico, Fr; Hattan, Pr; Katz, N; Labonte, B; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Walker, Cd; Gobbi, G.
Novel carbamate-based fatty-acid amide hydrolase inhibitors with enhanced stability and selectivity
2008 Clapper, Jr; Vacondio, F; King, Ar; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Piomelli, D.
MELATONIN RECEPTOR AGONISTS: SAR AND APPLICATIONS TO THE TREATMENT OF SLEEP-WAKE DISORDERS
2008 Rivara, S; Mor, M; Bedini, Annalida; Spadoni, Gilberto; Tarzia, Giorgio
Synthesis and Quantitative Structure–Activity Relationship of Fatty Acid Amide Hydrolase Inhibitors: Modulation at the N-Portion of Biphenyl-3-yl Alkylcarbamates
2008 Mor, M; Lodola, A; Rivara, S; Vacondio, F; Duranti, Andrea; Tontini, Andrea; Sanchini, S; Piersanti, Giovanni; Tarzia, Giorgio; Clapper, Jr; King, Ar; Piomelli, D.
A novel melatonin partial agonist with sleep-promoting properties
2007 OCHOA SANCHEZ, R; Karam, F; Bambico, F. R.; Katz, N; Spadoni, Gilberto; Bedini, Annalida; Mor, M; Rivara, S; Fraschini, F; Tarzia, Giorgio; Gobbi, G.
The Fatty Acid Amide Hydrolase Inhibitor URB597 (Cyclohexylcarbamic Acid 3’-Carbamoylbiphenyl-3-yl Ester) Reduces Neuropathic Pain after Oral Administration in Mice
2007 Russo, R; Loverme, J; LA RANA, G; Compton, Tr; Parrott, J; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Calignano, A; Piomelli, D.
Characterization of monoacylglycerol lipase (MGL) inhibitor URB602
2007 King, Ar; Rosengarth, A; Clapper, J; Duranti, Andrea; Tontini, Andrea; Mor, M; Rivara, S; Tarzia, Giorgio; Piomelli, D.
QSAR and molecular modelling investigations of a new series of alkyl carbamic acid aryl ester inhibitors of fatty acid amide hydrolase
2007 Lodola, A; Rivara, S; Mor, M; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Piomelli, D.
Synthesis of benzo[1,2-d;3,4-d’]diimidazole and 1H-pyrazolo[4,3-b]pyridine as putative A2A receptor antagonists
2007 Piersanti, Giovanni; Giorgi, Luca; Bartoccini, Francesca; Tarzia, Giorgio; P., Minetti; G., Gallo; F., Giorgi; M., Castorina; O., Ghirardi; P., Carminati
N-(anilinoethyl)acylamides: new melatonin receptor ligands with sleep inducing properties.
2007 Spadoni, Gilberto; Bedini, Annalida; Tarzia, Giorgio; Mor, M; Rivara, S; Lucini, V; Fraschini, F; Gobbi, G.
Conformational effects in enzyme catalysis: reaction via a high energy conformation in faty acid amide hydrolase
2007 Lodola, A; Mor, M; Zurek, J; Tarzia, Giorgio; Piomelli, D; Harvey, J; Mulholland, A. J.
Synthesis, Enantiomeric Resolution and Structure-Activity Relationship Study for a Series of 10,11-Dihydro-5H-dibenzo[a,d]cycloheptene MT2 Receptor Antagonists.
2007 Spadoni, Gilberto; Bedini, Annalida; Diamantini, Giuseppe; Tarzia, Giorgio; Rivara, S; Lorenzi, S; Lodola, A; Mor, M; Lucini, V; Pannacci, M; Caronno, A; Fraschini, F.
Melatonin antagonizes apoptosis via receptor interaction in U937 monocytic cell
2007 F., Radogna; Paternoster, Laura; Albertini, MARIA CRISTINA; C., Cerella; Accorsi, Augusto; Bucchini, ANAHI ELENA ADA; Spadoni, Gilberto; Diamantini, Giuseppe; Tarzia, Giorgio; M., DE NICOLA; M., D'Alessio; L., Ghibelli
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis, QSAR and Pharmacological Evaluation of Alkylcarbamic Acid Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: A Novel Approach to Antianxiety and Analgesic Agents | 1-gen-2008 | Tarzia, Giorgio; Duranti, Andrea; Tontini, Andrea; Rivara, S; Mor, M; Piomelli, D. | |
Quantitative Structure-Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors | 1-gen-2008 | Fioni, A; Vacondio, F; Mor, M; Silva, C; Lodola, A; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Piomelli, D. | |
Design and structure-activity relationships of subtype selective melatonin receptor ligands. | 1-gen-2008 | Rivara, S; Mor, M; Lodola, A; Spadoni, Gilberto; Bedini, Annalida; Tarzia, Giorgio; Lucini, V; Gobbi, G. | |
Selective increase of Slow Wave Sleep (SWS) by melatonin 2 receptors. | 1-gen-2008 | OCHOA SANCHEZ, R; Spadoni, Gilberto; Bedini, Annalida; Mor, M; Rivara, S; Fraschini, F; Tarzia, Giorgio; Gobbi, G. | |
Sintesi e studi di relazione struttura-attività/stabilità di carbammati inibitori dell’enzima FAAH | 1-gen-2008 | Sanchini, Silvano; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Vacondio, F; Fioni, A; Lodola, A; Rivara, S; Mor, M; Clapper, J; Piomelli, D. | |
Gordon Conference | 1-gen-2008 | Bedini, Annalida; Spadoni, Gilberto; Tarzia, Giorgio; Gobbi, G; Mor, M; Rivara, S. | |
Inibitori dell’enzima NAAA (N-Acylethanolamine-Hydrolizing Acid Amidase) come nuovi agenti antinfiammatori | 1-gen-2008 | Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Lodola, A; Rivara, S; Mor, M; Zhu, C; Solorzano, C; Piomelli, D. | |
Differences between direct cannabinoid agonists and FAAH inhibitors on antidepressant-like behavioural and serotonin-modulatory activity | 1-gen-2008 | Bambico, Fr; Hattan, Pr; Katz, N; Labonte, B; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Walker, Cd; Gobbi, G. | |
Novel carbamate-based fatty-acid amide hydrolase inhibitors with enhanced stability and selectivity | 1-gen-2008 | Clapper, Jr; Vacondio, F; King, Ar; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Piomelli, D. | |
MELATONIN RECEPTOR AGONISTS: SAR AND APPLICATIONS TO THE TREATMENT OF SLEEP-WAKE DISORDERS | 1-gen-2008 | Rivara, S; Mor, M; Bedini, Annalida; Spadoni, Gilberto; Tarzia, Giorgio | |
Synthesis and Quantitative Structure–Activity Relationship of Fatty Acid Amide Hydrolase Inhibitors: Modulation at the N-Portion of Biphenyl-3-yl Alkylcarbamates | 1-gen-2008 | Mor, M; Lodola, A; Rivara, S; Vacondio, F; Duranti, Andrea; Tontini, Andrea; Sanchini, S; Piersanti, Giovanni; Tarzia, Giorgio; Clapper, Jr; King, Ar; Piomelli, D. | |
A novel melatonin partial agonist with sleep-promoting properties | 1-gen-2007 | OCHOA SANCHEZ, R; Karam, F; Bambico, F. R.; Katz, N; Spadoni, Gilberto; Bedini, Annalida; Mor, M; Rivara, S; Fraschini, F; Tarzia, Giorgio; Gobbi, G. | |
The Fatty Acid Amide Hydrolase Inhibitor URB597 (Cyclohexylcarbamic Acid 3’-Carbamoylbiphenyl-3-yl Ester) Reduces Neuropathic Pain after Oral Administration in Mice | 1-gen-2007 | Russo, R; Loverme, J; LA RANA, G; Compton, Tr; Parrott, J; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Calignano, A; Piomelli, D. | |
Characterization of monoacylglycerol lipase (MGL) inhibitor URB602 | 1-gen-2007 | King, Ar; Rosengarth, A; Clapper, J; Duranti, Andrea; Tontini, Andrea; Mor, M; Rivara, S; Tarzia, Giorgio; Piomelli, D. | |
QSAR and molecular modelling investigations of a new series of alkyl carbamic acid aryl ester inhibitors of fatty acid amide hydrolase | 1-gen-2007 | Lodola, A; Rivara, S; Mor, M; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Piomelli, D. | |
Synthesis of benzo[1,2-d;3,4-d’]diimidazole and 1H-pyrazolo[4,3-b]pyridine as putative A2A receptor antagonists | 1-gen-2007 | Piersanti, Giovanni; Giorgi, Luca; Bartoccini, Francesca; Tarzia, Giorgio; P., Minetti; G., Gallo; F., Giorgi; M., Castorina; O., Ghirardi; P., Carminati | |
N-(anilinoethyl)acylamides: new melatonin receptor ligands with sleep inducing properties. | 1-gen-2007 | Spadoni, Gilberto; Bedini, Annalida; Tarzia, Giorgio; Mor, M; Rivara, S; Lucini, V; Fraschini, F; Gobbi, G. | |
Conformational effects in enzyme catalysis: reaction via a high energy conformation in faty acid amide hydrolase | 1-gen-2007 | Lodola, A; Mor, M; Zurek, J; Tarzia, Giorgio; Piomelli, D; Harvey, J; Mulholland, A. J. | |
Synthesis, Enantiomeric Resolution and Structure-Activity Relationship Study for a Series of 10,11-Dihydro-5H-dibenzo[a,d]cycloheptene MT2 Receptor Antagonists. | 1-gen-2007 | Spadoni, Gilberto; Bedini, Annalida; Diamantini, Giuseppe; Tarzia, Giorgio; Rivara, S; Lorenzi, S; Lodola, A; Mor, M; Lucini, V; Pannacci, M; Caronno, A; Fraschini, F. | |
Melatonin antagonizes apoptosis via receptor interaction in U937 monocytic cell | 1-gen-2007 | F., Radogna; Paternoster, Laura; Albertini, MARIA CRISTINA; C., Cerella; Accorsi, Augusto; Bucchini, ANAHI ELENA ADA; Spadoni, Gilberto; Diamantini, Giuseppe; Tarzia, Giorgio; M., DE NICOLA; M., D'Alessio; L., Ghibelli |
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