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Synthesis of 2-substituted tryptophans via a C3- to C2-alkyl migration 1-gen-2014 Mari, Michele; Lucarini, Simone; Bartoccini, Francesca; Piersanti, Giovanni; Spadoni, Gilberto
Synthesis and Characterization of New Bivalent Agents as Melatonin- and Histamine H3-Ligands 1-gen-2014 Pala, D.; Scalvini, L.; Lodola, A.; Mor, M.; Flammini, L.; Barocelli, E.; Lucini, V.; Scaglione, F.; Bartolucci, Silvia; Bedini, Annalida; Rivara, S.; Spadoni, Gilberto
Brønsted Acid-Catalyzed Bisindolization of α-amido acetals: Synthesis and Anticancer activity of bis(indolyl)ethanamino derivatives 1-gen-2014 Mari, Michele; Aurora, Tassoni; Lucarini, Simone; Fanelli, Mirco; Piersanti, Giovanni; Spadoni, Gilberto
Homology models of melatonin receptors: challenges and recent advances 1-gen-2013 D., Pala; A., Lodola; Bedini, Annalida; Spadoni, Gilberto; S., Rivara
Organocatalyzed coupling of indoles with dehydroalanine esters: synthesis of bis(indolyl)propanoates and indolacrylates 1-gen-2013 Lucarini, Simone; Mari, Michele; Piersanti, Giovanni; Spadoni, Gilberto
A Versatile Biomimetic Approach to Diindolylmethane Derivatives as Potential Anticancer Agents 1-gen-2012 Lucarini, Simone; Piersanti, Giovanni; Duranti, Andrea; Spadoni, Gilberto
Description of the constitutive activity of cloned human melatonin receptors hMT1 and hMT2 and discovery of inverse agonists 1-gen-2012 Devavry, S; Legros, C; Brasseur, C; Delagrange, P; Spadoni, Gilberto; Cohen, W; Malpaux, B; Boutin, Ja; Nosjean,
Synthesis of Tryptamine Derivatives via a Direct, One-Pot Reductive Alkylation of Indoles 1-gen-2012 Marika, Righi; Francesca, Topi; Bartolucci, Silvia; Bedini, Annalida; Piersanti, Giovanni; Spadoni, Gilberto
MT1-Selective Melatonin Receptor Ligands: Synthesis, Pharmacological Evaluation, and Molecular Dynamics Investigation of N-{[(3-O-Substituted)anilino]alkyl}amides 1-gen-2012 Rivara, S.; Pala, D.; Lodola, A.; Mor, M.; Lucini, V.; Dugnani, S.; Scaglione, F.; Bedini, Annalida; Lucarini, Simone; Tarzia, Giorgio; Spadoni, Gilberto
Anxiolytic effects of the melatonin MT2 receptor partial agonist UCM765: Comparison with melatonin and diazepam 1-gen-2012 Ochoa Sanchez, R.; Rainer, Q.; Comai, S.; Spadoni, Gilberto; Bedini, Annalida; Rivara, S.; Fraschini, F.; Mor, M.; Tarzia, Giorgio; Gobbi, G.
Synthesis and Configuration Determination of All Enantiopure Stereoisomers of the Melatonin Receptor Ligand 4-Phenyl-2-propionamidotetralin using an Expedient Optical Resolution of 4-Phenyl-2-tetralone 1-gen-2012 Lucarini, Simone; Bartolucci, Silvia; Bedini, Annalida; Gatti, G.; Orlando, Pierfrancesco; Piersanti, Giovanni; Spadoni, Gilberto
Promotion of non-rapid eye movement sleep and activation of reticular thalamic neurons by a novel MT2 melatonin receptor ligand 1-gen-2011 Ochoa Sanchez, R; Comai, S; Lacoste, B; Bambico, Fr; Dominguez Lopez, S; Spadoni, Gilberto; Rivara, S; Bedini, Annalida; Angeloni, D; Fraschini, F; Mor, M; Tarzia, Giorgio; Descarries, L; Gobbi, G.
Toward the Definition of Stereochemical Requirements for MT(2)-Selective Antagonists and Partial Agonists by Studying 4-Phenyl-2-propionamidotetralin Derivatives 1-gen-2011 Bedini, Annalida; Lucarini, Simone; Spadoni, Gilberto; Tarzia, Giorgio; Scaglione, F; Dugnani, S; Pannacci, M; Lucini, V; Carmi, C; Pala, D; Rivara, S; Mor, M.
ST1936 stimulates cAMP, Ca2+, ERK1/2 and Fyn Kinase through a full activation of cloned hman 5-HT6 receptors 1-gen-2011 Riccioni, T.; Bordi, F.; Minetti, P.; Spadoni, Gilberto; Yun, H. M.; Im, B. H.; Tarzia, Giorgio; Rhim, H.; Borsini, F.
Direct, One-Pot Reductive Alkylation of Anilines with Functionalized Acetals Mediated by Triethylsilane and TFA. Straightforward Route for Unsymmetrically Substituted Ethylenediamine 1-gen-2011 M., Righi; Bedini, Annalida; Piersanti, Giovanni; F., Romagnoli; Spadoni, Gilberto
Bivalent Ligand Approach on N-[2-[(3-methoxyphenyl)methylamino]ethyl]acetamide. Synthesis, Binding Affinity and Intrinsic Acivity for MT(1) and MT(2) melatonin Receptors. 1-gen-2011 Spadoni, Gilberto; Bedini, Annalida; Orlando, Pierfrancesco; Lucarini, Simone; Tarzia, Giorgio; Mor, M.; Rivara, S.; Lucini, V.; Pannacci, M.; Scaglione, F.
Melatonin receptor agonists: new options for insomnia and depression treatment 1-gen-2011 Spadoni, Gilberto; Bedini, Annalida; Rivara, S; Mor, M.
A Novel One-Pot Approach of Hexahydropyrrolo[2,3-b]indole Nucleus by a cascade addition/cyclization strategy: Synthesis of (±)-Esermethole 1-gen-2010 Lucarini, Simone; Bartoccini, Francesca; Battistoni, F; Diamantini, Giuseppe; Piersanti, Giovanni; Righi, M; Spadoni, Gilberto
Diastereo- and enantioselective hydrogenation of a challenging enamide derived from 4-phenyl-2-tetralone: an appealing shortcut towards enantiopure cis-2-aminotetraline derivatives 1-gen-2010 Lucarini, Simone; Alessi, M; Bedini, Annalida; Giorgini, G; Piersanti, Giovanni; Spadoni, Gilberto
Recent advances in the development of melatonin MT1 and MT2 receptor agonists 1-gen-2010 Mor, M; Rivara, S; Pala, D; Bedini, Annalida; Spadoni, Gilberto; Tarzia, Giorgio
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