| Nome |
# |
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Synthesis and Evaluation of Saccharide-Based Aliphatic and Aromatic Esters as Antimicrobial and Antibiofilm Agents, file e18b865c-f896-1ee6-e053-3a05fe0ae544
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137
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Marine Alkaloid 2,2-Bis(6-bromo-3-indolyl) Ethylamine and Its Synthetic Derivatives Inhibit Microbial Biofilms Formation and Disaggregate Developed Biofilms, file e18b865c-be9f-1ee6-e053-3a05fe0ae544
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113
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Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines, file e18b865d-51fd-1ee6-e053-3a05fe0ae544
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97
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Lactose oleate as new biocompatible surfactant for pharmaceutical applications, file e18b865d-5a9d-1ee6-e053-3a05fe0ae544
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89
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|
Synthesis of 2-substituted tryptophans via a C3- to C2-alkyl migration, file e18b865b-8cda-1ee6-e053-3a05fe0ae544
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86
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|
Identification and quantification of new isomers of isopropyl-malic acid in wine by LC-IT and LC-Q-Orbitrap, file e18b865d-55e8-1ee6-e053-3a05fe0ae544
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82
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Palladium(II)-Catalyzed Intramolecular Oxidative C−H/C−H Cross-Coupling Reaction of C3,N-linked Biheterocycles: Rapid Access to Polycyclic Nitrogen Heterocycles, file e18b865d-5a17-1ee6-e053-3a05fe0ae544
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70
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Polycyclic Indolines by Acid-Mediated Intramolecular Dearomative Strategy: Reversing Indole Reactivity in the Pictet‒Spengler-Type Reaction, file e18b865d-8621-1ee6-e053-3a05fe0ae544
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59
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Synthesis, Structure-Activity Relationships and In Vitro Toxicity Profile of Lactose-Based Fatty Acid Monoesters as Possible Drug Permeability Enhancers, file e18b865c-9acd-1ee6-e053-3a05fe0ae544
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57
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A combination of sugar esters and chitosan to promote in vivo wound care, file e18b865d-ae86-1ee6-e053-3a05fe0ae544
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54
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Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives, file e18b865d-5444-1ee6-e053-3a05fe0ae544
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50
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Unsaturated fatty acids lactose esters: cytotoxicity, permeability enhancement and antimicrobial activity, file e18b865d-5aa3-1ee6-e053-3a05fe0ae544
|
40
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Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands, file e18b865d-5f08-1ee6-e053-3a05fe0ae544
|
40
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SYNTHESIS AND EVALUATION OF SUGAR-BASED ALIPHATIC AND AROMATIC FATTY ACID ESTERS AS ANTIMICROBIAL AND ANTIBIOFILM AGENTS, file e18b865c-e4b4-1ee6-e053-3a05fe0ae544
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39
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One-Pot Synthesis of Biheterocycles Based on Indole and Azole Scaffolds Using Tryptamines and 1,2-Diaza-1,3-dienes as Building Blocks, file e18b865d-5418-1ee6-e053-3a05fe0ae544
|
28
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A recent update on new synthetic chiral compounds with antileishmanial activity, file c3d0ff7c-388c-417c-8f99-e1649dcbae6b
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22
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A Fluorinated Analogue of Marine Bisindole Alkaloid 2,2-Bis(6-bromo-1H-indol-3-yl)ethanamine as Potential Anti-Biofilm Agent and Antibiotic Adjuvant Against Staphylococcus aureus, file e18b865d-25ce-1ee6-e053-3a05fe0ae544
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22
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Phenotype Screening of an Azole-bisindole Chemical Library Identifies URB1483 as a New Antileishmanial Agent Devoid of Toxicity on Human Cells, file e18b865d-a367-1ee6-e053-3a05fe0ae544
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14
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Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives, file e18b865b-879e-1ee6-e053-3a05fe0ae544
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10
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|
Synthesis and Biological Evaluation of Metabolites of 2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), A Potent Antagonist of the A2AAdenosine Receptor for the Treatment of Parkinson’s Disease, file e18b865b-87fe-1ee6-e053-3a05fe0ae544
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10
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Organocatalytic synthesis of α-quaternary amino acid derivatives via aza-Friedel–Crafts alkylation of indoles with simple α-amidoacrylates, file e18b865b-850d-1ee6-e053-3a05fe0ae544
|
7
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Synthesis and Properties of Sucrose- and Lactose-Based Aromatic Ester Surfactants as Potential Drugs Permeability Enhancers, file 30ba7e6e-5b93-438c-8cec-97e8096ccf1b
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6
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Design and synthesis of N-[3,3-diphenyl-propenyl]alkanamides as a novel class of potent MT2-selective Melatonin receptor ligands, file e18b865b-7d49-1ee6-e053-3a05fe0ae544
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6
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Permeability-enhancing effects of three laurate-disaccharide monoesters across isolated rat intestinal mucosae, file e18b865d-9763-1ee6-e053-3a05fe0ae544
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6
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2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors, file d961becf-cd0a-41bf-947d-dde7ba57c160
|
5
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A macrocyclic ligand able to bind gallium(III) by preorganized pendant arms; coordination and kinetic studies., file e18b865b-79b8-1ee6-e053-3a05fe0ae544
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5
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A combination of sugar esters and chitosan to promote in vivo wound care, file e18b865d-ae87-1ee6-e053-3a05fe0ae544
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5
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New Ligand bearing preorganized binding side-arms interacting with ammonium cations: Synthesis, conformational studies and crystal structure, file e18b865b-7b3b-1ee6-e053-3a05fe0ae544
|
4
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The indole-3-carbinol tetrameric derivative CTet inhibits cell proliferation via overexpression of p21/CDKN1A in both estrogen receptor-positive and triple-negative breast cancer cell lines, file e18b865b-85ac-1ee6-e053-3a05fe0ae544
|
4
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Organocatalyzed coupling of indoles with dehydroalanine esters: synthesis of bis(indolyl)propanoates and indolacrylates, file e18b865b-88e3-1ee6-e053-3a05fe0ae544
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4
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|
Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands, file e18b865b-a73f-1ee6-e053-3a05fe0ae544
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4
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Palladium(II)-Catalyzed Intramolecular Oxidative C−H/C−H Cross-Coupling Reaction of C3,N-linked Biheterocycles: Rapid Access to Polycyclic Nitrogen Heterocycles, file e18b865c-0f3b-1ee6-e053-3a05fe0ae544
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4
|
|
Synthesis and Biological Evaluation of a γ-Cyclodextrin-based Formulation of the Anticancer Agent 5,6,11,12,17,18,23,24-Octahydrocyclododeca[1,2-b:4,5-b’:7,8-b’’:10,11-b’’’]tetraindole (CTet), file e18b865c-5ac7-1ee6-e053-3a05fe0ae544
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4
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Determination of coeluted isomers in wine samples by application of MS/MS deconvolution analysis, file e18b865d-256a-1ee6-e053-3a05fe0ae544
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4
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Synthesis and Biological Characterization of the New Glycolipid Lactose Undecylenate (URB1418), file e18b865d-c2fa-1ee6-e053-3a05fe0ae544
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4
|
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Versatile stereoselective oxidative alkoxycarbonylation of styrenes at room-temperature, file 46d154bc-70f2-4721-a525-402ee5b4a9cc
|
3
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Sugar-Based Monoester Surfactants: Synthetic Methodologies, Properties, and Biological Activities, file 4c2fd4ba-2a0d-44c1-9a4c-ff3ce860ce16
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3
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Macrocyclic ligands bearing two 3-(Hydroxy)-2-pyridinone moieties as side-arms. Conformational studies, synthesis, crystal structure, and alkali and alkaline earth complex formation., file e18b865b-7ca5-1ee6-e053-3a05fe0ae544
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3
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Inhibition of Testosterone Aromatization by the Indole-3-carbinol Derivative CTet in CYP19A1-overexpressing MCF-7 Breast Cancer Cells, file e18b865b-ab13-1ee6-e053-3a05fe0ae544
|
3
|
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Total Synthesis of Natural Disaccharide Sambubiose, file e18b865d-273e-1ee6-e053-3a05fe0ae544
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3
|
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6'-O-Lactose Ester Surfactants as an Innovative Opportunity in the Pharmaceutical Field: From Synthetic Methods to Biological Applications, file e18b865d-a369-1ee6-e053-3a05fe0ae544
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3
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Single-Walled Carbon Nanotubes Functionalization for the Delivery of the Water Insoluble Anticancer Agent Indole-3-carbinol Cyclic Tetrameric Derivative CTet, file e18b865b-878b-1ee6-e053-3a05fe0ae544
|
2
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One-Pot Synthesis of Biheterocycles Based on Indole and Azole Scaffolds Using Tryptamines and 1,2-Diaza-1,3-dienes as Building Blocks, file e18b865b-d305-1ee6-e053-3a05fe0ae544
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2
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Marine bisindole alkaloid: A potential apoptotic inducer in human cancer cells, file e18b865c-9a57-1ee6-e053-3a05fe0ae544
|
2
|
|
Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands, file e18b865c-9b02-1ee6-e053-3a05fe0ae544
|
2
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The influence of mannose-based esters on the mesophase behaviour of lyotropic liquid crystalline nanosystems as drug delivery vectors, file 77956484-db05-4dea-9b38-fdc90775c07c
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1
|
|
Synthesis and Biological Evaluation of 6-O-Sucrose Monoester Glycolipids as Possible New Antifungal Agents, file 9b13e5c1-9400-4584-905f-829cdcb8a638
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1
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Synthetic Methodologies and Therapeutic Potential of Indole-3-Carbinol (I3C) and Its Derivatives, file c5c83cfa-7b4b-4faa-9d2f-a1e4ef52c695
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1
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Synthesis and Configuration Determination of All Enantiopure Stereoisomers of the Melatonin Receptor Ligand 4-Phenyl-2-propionamidotetralin using an Expedient Optical Resolution of 4-Phenyl-2-tetralone, file e18b865b-8544-1ee6-e053-3a05fe0ae544
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1
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Brønsted Acid-Catalyzed Bisindolization of α-amido acetals: Synthesis and Anticancer activity of bis(indolyl)ethanamino derivatives, file e18b865b-89f5-1ee6-e053-3a05fe0ae544
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1
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|
Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines, file e18b865b-a413-1ee6-e053-3a05fe0ae544
|
1
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|
Diastereo- and enantioselective hydrogenation of a challenging enamide derived from 4-phenyl-2-tetralone: an appealing shortcut towards enantiopure cis-2-aminotetraline derivatives, file e18b865b-a711-1ee6-e053-3a05fe0ae544
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1
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A practical and expeditious method for the preparation of the anticancer agent 5,6,11,12,17,18,23,24-octahydrocyclododeca[1,2-b:4,5-b’:7,8-b’’:10,11-b’’’]tetraindole (CTet), file e18b865b-aa04-1ee6-e053-3a05fe0ae544
|
1
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An improved synthesis of cis-4-phenyl-2-propionamidotetralin (4-P-PDOT): a selective MT2 melatonin receptor antagonist., file e18b865b-aa4e-1ee6-e053-3a05fe0ae544
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1
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Bivalent Ligand Approach on N-[2-[(3-methoxyphenyl)methylamino]ethyl]acetamide. Synthesis, Binding Affinity and Intrinsic Acivity for MT(1) and MT(2) melatonin Receptors., file e18b865b-ad36-1ee6-e053-3a05fe0ae544
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1
|
|
Pharmacokinetic and pharmacodynamic evaluation of ramelteon : an insomnia therapy, file e18b865b-ad39-1ee6-e053-3a05fe0ae544
|
1
|
|
MT1-Selective Melatonin Receptor Ligands: Synthesis, Pharmacological Evaluation, and Molecular Dynamics Investigation of N-{[(3-O-Substituted)anilino]alkyl}amides, file e18b865b-afd4-1ee6-e053-3a05fe0ae544
|
1
|
|
Lactose oleate as new biocompatible surfactant for pharmaceutical applications, file e18b865c-6c5e-1ee6-e053-3a05fe0ae544
|
1
|
|
Antitumoral activity of indole-3-carbinol cyclic tri- and tetrameric derivatives mixture in human breast cancer cells: in vitro and in vivo studies, file e18b865c-878f-1ee6-e053-3a05fe0ae544
|
1
|
|
Unsaturated fatty acids lactose esters: cytotoxicity, permeability enhancement and antimicrobial activity, file e18b865c-f39d-1ee6-e053-3a05fe0ae544
|
1
|
|
Polycyclic Indolines by Acid-Mediated Intramolecular Dearomative Strategy: Reversing Indole Reactivity in the Pictet‒Spengler-Type Reaction, file e18b865d-8620-1ee6-e053-3a05fe0ae544
|
1
|
|
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors, file eda2b55a-93da-457f-8131-b1087d062aae
|
1
|
| Totale |
1.234 |