BARTOCCINI, FRANCESCA
BARTOCCINI, FRANCESCA
Dipartimento di Scienze Biomolecolari (DISB)
2-n-Butyl- 9-methyl-8-(1,2,3)triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological Characterization
2005-01-01 Minetti, P; TINTI M., O; Carminati, P; Castorina, M; DI CESARE M., A; DI SERIO, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, Luca; Piersanti, Giovanni; Bartoccini, Francesca; Tarzia, Giorgio
2-n-butyl-9-methyl-8-(1,2,3)triazol-2yl-9H-purin-6-yl-amine (ST 1535) and analogs as A2a Adenosine receptor antagonists. Design, synthesis and pharmacological characterization
2003-01-01 Bartoccini, Francesca; Castorina, M.; DI CESARE, M. A.; Gallo, G; Ghirardi, O.; Giorgi, F. GIORGI L.; Minetti, P.; Piersanti, Giovanni; Tarzia, Giorgio; Tinti, M. O.
Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties
2022-01-01 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology
2020-01-01 Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni
Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin
2019-01-01 Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Mari, Michele; Piersanti, Giovanni
Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone
2021-01-01 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Development of a practical and sustainable strategy for the synthesis of ST1535 by an iron-catalyzed Kumada cross-coupling reaction
2014-01-01 Bartoccini, Francesca; Piersanti, Giovanni; Silvia, Armaroli; Alberto, Cerri; Walter, Cabri
Direct B-alkyl Suzuki-Miyaura cross-coupling of 2-halopurines. Practical synthesis os ST1535, a potent adenosine A2A receptor antagonist
2010-01-01 Bartoccini, Francesca; Cabri, W; Celona, D; Minetti, P; Piersanti, Giovanni; G., Tarzia
Direct, Regioselective, and Chemoselective Preparation of Novel Boronated Tryptophans by Friedel–Crafts Alkylation
2012-01-01 Bartolucci, Silvia; Bartoccini, Francesca; Righi, M.; Piersanti, Giovanni
Divergent reactions of oxindoles with amino alcohols via the borrowing hydrogen process: oxindole ring opening vs. C3 alkylation
2018-01-01 Di Gregorio, Giovanni; Mari, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni
Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions
2012-01-01 Bartoccini, Francesca; Piersanti, Giovanni; Marco, Mor; Tarzia, Giorgio; Patrizia, Minetti; Walter, Cabri
General synthesis of unnatural 4-, 5-, 6-, and 7-bromo-d-tryptophans by means of a regioselective indole alkylation
2020-01-01 Bartoccini, Francesca; Fanini, Fabiola; Retini, Michele; Piersanti, Giovanni
I-152, a supplier of N-acetyl-cysteine and cysteamine, inhibits immunoglobulin secretion and plasma cell maturation in LP-BM5 murine leukemia retrovirus-infected mice by affecting the unfolded protein response
2020-01-01 Fraternale, Alessandra; Zara, Carolina; Di Mambro, Tomas; Manuali, Elisabetta; Genovese, Domenica Anna; Galluzzi, Luca; Diotallevi, Aurora; Pompa, Andrea; De Marchis, Francesca; Ambrogini, Patrizia; Cesarini, Erica; Luchetti, Francesca; Smietana, Michaël; Green, Kathy; Bartoccini, Francesca; Magnani, Mauro; Crinelli, Rita
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign
2020-01-01 Linciano, Pasquale; Cullia, Gregorio; Borsari, Chiara; Santucci, Matteo; Ferrari, Stefania; Witt, Gesa; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Santarém, Nuno; Cordeiro da Silva, Anabela; Conti, Paola; Bolognesi, Maria Laura; Roberti, Marinella; Prati, Federica; Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni; Cavalli, Andrea; Goldoni, Luca; Bertozzi, Sine Mandrup; Bertozzi, Fabio; Brambilla, Enzo; Rizzo, Vincenzo; Piomelli, Daniele; Pinto, Andrea; Bandiera, Tiziano; Costi, Maria Paola
Improved Synthesis of gamma-nitro-alfa-Amino ester and Acid Derivatives
2005-01-01 Ballini, R; Balsamini, Cesarino; Bartoccini, Francesca; Gianotti, M.; Martinelli, C.; Savoretti, N.
Iron-Catalyzed Direct C3-Benzylation of Indoles with Benzyl Alcohols through Borrowing Hydrogen
2017-01-01 DI GREGORIO, Giovanni; Mari, Michele; Bartoccini, Francesca; Piersanti, Giovanni
Large-Scale Preparation of N-Butanoyl-l-glutathione (C4-GSH)
2019-01-01 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Fraternale, Alessandra; Piersanti, Giovanni
Metodo di sintesi di derivati del glutatione [Method for the synthesis of glutathione derivatives]
2017-01-01 Bartoccini, Francesca; Fraternale, Alessandra; Piersanti, Giovanni
A Novel One-Pot Approach of Hexahydropyrrolo[2,3-b]indole Nucleus by a cascade addition/cyclization strategy: Synthesis of (±)-Esermethole
2010-01-01 Lucarini, Simone; Bartoccini, Francesca; Battistoni, F; Diamantini, Giuseppe; Piersanti, Giovanni; Righi, M; Spadoni, Gilberto
Novel, Chiral, and Enantiopure C2‐Symmetric Thioureas Promote Asymmetric Protio‐Pictet‐Spengler Reactions by Anion‐Binding Catalysis
2021-01-01 Retini, Michele; Bartoccini, Francesca; Zappia, Giovanni; Piersanti, Giovanni
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 2-n-Butyl- 9-methyl-8-(1,2,3)triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological Characterization | 1-gen-2005 | Minetti, P; TINTI M., O; Carminati, P; Castorina, M; DI CESARE M., A; DI SERIO, S; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, Luca; Piersanti, Giovanni; Bartoccini, Francesca; Tarzia, Giorgio | |
| 2-n-butyl-9-methyl-8-(1,2,3)triazol-2yl-9H-purin-6-yl-amine (ST 1535) and analogs as A2a Adenosine receptor antagonists. Design, synthesis and pharmacological characterization | 1-gen-2003 | Bartoccini, Francesca; Castorina, M.; DI CESARE, M. A.; Gallo, G; Ghirardi, O.; Giorgi, F. GIORGI L.; Minetti, P.; Piersanti, Giovanni; Tarzia, Giorgio; Tinti, M. O. | |
| Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties | 1-gen-2022 | Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni | |
| C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology | 1-gen-2020 | Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni | |
| Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin | 1-gen-2019 | Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Mari, Michele; Piersanti, Giovanni | |
| Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone | 1-gen-2021 | Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni | |
| Development of a practical and sustainable strategy for the synthesis of ST1535 by an iron-catalyzed Kumada cross-coupling reaction | 1-gen-2014 | Bartoccini, Francesca; Piersanti, Giovanni; Silvia, Armaroli; Alberto, Cerri; Walter, Cabri | |
| Direct B-alkyl Suzuki-Miyaura cross-coupling of 2-halopurines. Practical synthesis os ST1535, a potent adenosine A2A receptor antagonist | 1-gen-2010 | Bartoccini, Francesca; Cabri, W; Celona, D; Minetti, P; Piersanti, Giovanni; G., Tarzia | |
| Direct, Regioselective, and Chemoselective Preparation of Novel Boronated Tryptophans by Friedel–Crafts Alkylation | 1-gen-2012 | Bartolucci, Silvia; Bartoccini, Francesca; Righi, M.; Piersanti, Giovanni | |
| Divergent reactions of oxindoles with amino alcohols via the borrowing hydrogen process: oxindole ring opening vs. C3 alkylation | 1-gen-2018 | Di Gregorio, Giovanni; Mari, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni | |
| Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions | 1-gen-2012 | Bartoccini, Francesca; Piersanti, Giovanni; Marco, Mor; Tarzia, Giorgio; Patrizia, Minetti; Walter, Cabri | |
| General synthesis of unnatural 4-, 5-, 6-, and 7-bromo-d-tryptophans by means of a regioselective indole alkylation | 1-gen-2020 | Bartoccini, Francesca; Fanini, Fabiola; Retini, Michele; Piersanti, Giovanni | |
| I-152, a supplier of N-acetyl-cysteine and cysteamine, inhibits immunoglobulin secretion and plasma cell maturation in LP-BM5 murine leukemia retrovirus-infected mice by affecting the unfolded protein response | 1-gen-2020 | Fraternale, Alessandra; Zara, Carolina; Di Mambro, Tomas; Manuali, Elisabetta; Genovese, Domenica Anna; Galluzzi, Luca; Diotallevi, Aurora; Pompa, Andrea; De Marchis, Francesca; Ambrogini, Patrizia; Cesarini, Erica; Luchetti, Francesca; Smietana, Michaël; Green, Kathy; Bartoccini, Francesca; Magnani, Mauro; Crinelli, Rita | |
| Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign | 1-gen-2020 | Linciano, Pasquale; Cullia, Gregorio; Borsari, Chiara; Santucci, Matteo; Ferrari, Stefania; Witt, Gesa; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Santarém, Nuno; Cordeiro da Silva, Anabela; Conti, Paola; Bolognesi, Maria Laura; Roberti, Marinella; Prati, Federica; Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni; Cavalli, Andrea; Goldoni, Luca; Bertozzi, Sine Mandrup; Bertozzi, Fabio; Brambilla, Enzo; Rizzo, Vincenzo; Piomelli, Daniele; Pinto, Andrea; Bandiera, Tiziano; Costi, Maria Paola | |
| Improved Synthesis of gamma-nitro-alfa-Amino ester and Acid Derivatives | 1-gen-2005 | Ballini, R; Balsamini, Cesarino; Bartoccini, Francesca; Gianotti, M.; Martinelli, C.; Savoretti, N. | |
| Iron-Catalyzed Direct C3-Benzylation of Indoles with Benzyl Alcohols through Borrowing Hydrogen | 1-gen-2017 | DI GREGORIO, Giovanni; Mari, Michele; Bartoccini, Francesca; Piersanti, Giovanni | |
| Large-Scale Preparation of N-Butanoyl-l-glutathione (C4-GSH) | 1-gen-2019 | Bartoccini, Francesca; Mari, Michele; Retini, Michele; Fraternale, Alessandra; Piersanti, Giovanni | |
| Metodo di sintesi di derivati del glutatione [Method for the synthesis of glutathione derivatives] | 1-gen-2017 | Bartoccini, Francesca; Fraternale, Alessandra; Piersanti, Giovanni | |
| A Novel One-Pot Approach of Hexahydropyrrolo[2,3-b]indole Nucleus by a cascade addition/cyclization strategy: Synthesis of (±)-Esermethole | 1-gen-2010 | Lucarini, Simone; Bartoccini, Francesca; Battistoni, F; Diamantini, Giuseppe; Piersanti, Giovanni; Righi, M; Spadoni, Gilberto | |
| Novel, Chiral, and Enantiopure C2‐Symmetric Thioureas Promote Asymmetric Protio‐Pictet‐Spengler Reactions by Anion‐Binding Catalysis | 1-gen-2021 | Retini, Michele; Bartoccini, Francesca; Zappia, Giovanni; Piersanti, Giovanni |