Sfoglia per Autore
New cinnamic acid sugar esters as potential UVB filters: Synthesis, cytotoxicity, and physicochemical properties
2025 Olivieri, Diego; Verboni, Michele; Benedetti, Serena; Paderni, Daniele; Carfagna, Carla; Duranti, Andrea; Lucarini, Simone
Efficient and Rapid Arylation of NH₂‐Unprotected Bromobisindole Ethanamines via Suzuki‐Miyaura Coupling: Generating New Leads Against Leishmania
2025 Buono, Alessandro; Diotallevi, Aurora; Maestrini, Sara; Verboni, Michele; Kiuru, Paula; Galluzzi, Luca; Duranti, Andrea; Olivieri, Diego; Lucarini, Simone
Unveiling the Interactions between Amino Acids-Based Surfactants and Lipid Bilayers: A Small Angle Neutron Scattering and Reflectivity Study
2025 Perinelli, Diego R.; Verboni, Michele; Tiboni, Mattia; Doutch, James; Pisani, Michela; Domenici, Fabio; Bonacucina, Giulia; Cespi, Marco; Lucarini, Simone; Duranti, Andrea; Palmieri, Giovanni Filippo; Campana, Mario; Casettari, Luca
Characterization of the symmetrical benzimidazole twin drug TL1228: the role as viral entry inhibitor for fighting COVID-19
2024 Murdocca, Michela; Andrade Santos-Filho, Osvaldo; De Masi, Claudia; dos Santos Rodrigues, Edivaldo; Campos de Souza, Claudia Valeria; De Santis, Riccardo; Amatore, Donatella; Latini, Andrea; Schipani, Rossella; di Rienzo Businco, Lino; Brandimarte, Bruno; Grilli, Giorgia; Huang, Tien L; Mayence, Annie S; Lista, Florigio; Duranti, Andrea; Sangiuolo, Federica; Vanden Eynde, Jean Jacques; Novelli, Giuseppe
Endocannabinoid Degradation Enzyme Inhibitors as Potential Antipsychotics: A Medicinal Chemistry Perspective
2023 Mangiatordi, Giuseppe Felice; Cavalluzzi, Maria Maddalena; Delre, Pietro; Lamanna, Giuseppe; Lomuscio, Maria Cristina; Saviano, Michele; Majoral, Jean-Pierre; Mignani, Serge; Duranti, Andrea; Lentini, Giovanni
Synthesis and Biological Evaluation of 6-O-Sucrose Monoester Glycolipids as Possible New Antifungal Agents
2023 Verboni, Michele; Sisti, Maurizio; Campana, Raffaella; Benedetti, Serena; Palma, Francesco; Potenza, Lucia; Lucarini, Simone; Duranti, Andrea
Synthetic Methodologies and Therapeutic Potential of Indole-3-Carbinol (I3C) and Its Derivatives
2023 Centofanti, Federica; Buono, Alessandro; Verboni, Michele; Tomino, Carlo; Lucarini, Simone; Duranti, Andrea; Pandolfi, Pier Paolo; Novelli, Giuseppe
Sugar-Based Monoester Surfactants: Synthetic Methodologies, Properties, and Biological Activities
2023 Verboni, Michele; Romano Perinelli, Diego; Buono, Alessandro; Campana, Raffaella; Sisti, Maurizio; Duranti, Andrea; Lucarini, Simone
The influence of mannose-based esters on the mesophase behaviour of lyotropic liquid crystalline nanosystems as drug delivery vectors
2023 Tiboni, Mattia; Astolfi, Paola; Verboni, Michele; Benedetti, Serena; Giorgini, Elisabetta; Notarstefano, Valentina; Vita, Francesco; Ranieri, Simone; Duranti, Andrea; Lucarini, Simone; Casettari, Luca; Pisani, Michela
An Investigation on the Relationships between Mass Spectrometric Collisional Data and Biological Activity/Stability of Some N-Acylethanolamine Acid Amidase (NAAA) β-Lactone Inhibitors
2023 Isak, Ilena; Duranti, Andrea; Traldi, Pietro
Characterization of URB Series Synthetic Cannabinoids by HRMS and UHPLC–MS/MS
2023 Agostini, Marco; Favretto, Donata; Renzoni, Caterina; Vogliardi, Susanna; Duranti, Andrea
The Endocannabinoid System as a Target for Neuroprotection/Neuroregeneration in Perinatal Hypoxic–Ischemic Brain Injury
2023 Duranti, Andrea; Beldarrain, Gorane; Álvarez, Antonia; Sbriscia, Matilde; Carloni, Silvia; Balduini, Walter; Alonso-Alconada, Daniel
Synthesis and Properties of Sucrose- and Lactose-Based Aromatic Ester Surfactants as Potential Drugs Permeability Enhancers
2023 Verboni, Michele; Perinelli, Diego Romano; Qiu, Carol Yingshan; Tiboni, Mattia; Aluigi, Annalisa; Lucarini, Simone; Lam, Jenny K. W.; Duranti, Andrea
Characterization and Preliminary In Vitro Antioxidant Activity of a New Multidrug Formulation Based on the Co-Encapsulation of Rutin and the α-Acylamino-β-Lactone NAAA Inhibitor URB894 within PLGA Nanoparticles
2023 Gagliardi, Agnese; Voci, Silvia; Ambrosio, Nicola; Fresta, Massimo; Duranti, Andrea; Cosco, Donato
Inhibition of Fatty Acid Amide Hydrolase (FAAH) Regulates NF-kb Pathways Reducing Bleomycin-Induced Chronic Lung Inflammation and Pulmonary Fibrosis
2023 Genovese, Tiziana; Duranti, Andrea; Monaco, Francesco; Siracusa, Rosalba; Fusco, Roberta; Impellizzeri, Daniela; D'Amico, Ramona; Cordaro, Marika; Cuzzocrea, Salvatore; Di Paola, Rosanna
Synthesis and Biological Characterization of the New Glycolipid Lactose Undecylenate (URB1418)
2022 Verboni, Michele; Benedetti, Serena; Campana, Raffaella; Palma, Francesco; Potenza, Lucia; Sisti, Maurizio; Duranti, Andrea; Lucarini, Simone
A combination of sugar esters and chitosan to promote in vivo wound care
2022 Tiboni, Mattia; Elmowafy, Enas; El-Derany, Marwa O; Benedetti, Serena; Campana, Raffaella; Verboni, Michele; Potenza, Lucia; Palma, Francesco; Citterio, Barbara; Sisti, Maurizio; Duranti, Andrea; Lucarini, Simone; Soliman, Mahmoud E; Casettari, Luca
The Synthetic Cannabinoid URB447 Exerts Antitumor and Antimetastatic Effect in Melanoma and Colon Cancer
2022 Benedicto, Aitor; Arteta, Beatriz; Duranti, Andrea; Alonso-Alconada, Daniel
Indole-3-carbinol in vitro antiviral activity against SARS-Cov-2 virus and in vivo toxicity
2022 Centofanti, Federica; Alonzi, Tonino; Latini, Andrea; Spitalieri, Paola; Murdocca, Michela; Chen, Xiaodong; Cui, Weibo; Shang, Qianwen; Goletti, Delia; Shi, Yufang; Duranti, Andrea; Tomino, Carlo; Biancolella, Michela; Sangiuolo, Federica; Capobianchi, Maria Rosaria; Jain, Suresh; Novelli, Giuseppe; Pandolfi, Pier Paolo
Fatty Acid Amide Hydrolase (FAAH) Inhibition Plays a Key Role in Counteracting Acute Lung Injury
2022 Genovese, Tiziana; Duranti, Andrea; D'Amico, Ramona; Fusco, Roberta; Impellizzeri, Daniela; Peritore, Alessio Filippo; Crupi, Rosalia; Gugliandolo, Enrico; Cuzzocrea, Salvatore; Di Paola, Rosanna; Siracusa, Rosalba; Cordaro, Marika
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| New cinnamic acid sugar esters as potential UVB filters: Synthesis, cytotoxicity, and physicochemical properties | 1-gen-2025 | Olivieri, Diego; Verboni, Michele; Benedetti, Serena; Paderni, Daniele; Carfagna, Carla; Duranti, Andrea; Lucarini, Simone | |
| Efficient and Rapid Arylation of NH₂‐Unprotected Bromobisindole Ethanamines via Suzuki‐Miyaura Coupling: Generating New Leads Against Leishmania | 1-gen-2025 | Buono, Alessandro; Diotallevi, Aurora; Maestrini, Sara; Verboni, Michele; Kiuru, Paula; Galluzzi, Luca; Duranti, Andrea; Olivieri, Diego; Lucarini, Simone | |
| Unveiling the Interactions between Amino Acids-Based Surfactants and Lipid Bilayers: A Small Angle Neutron Scattering and Reflectivity Study | 1-gen-2025 | Perinelli, Diego R.; Verboni, Michele; Tiboni, Mattia; Doutch, James; Pisani, Michela; Domenici, Fabio; Bonacucina, Giulia; Cespi, Marco; Lucarini, Simone; Duranti, Andrea; Palmieri, Giovanni Filippo; Campana, Mario; Casettari, Luca | |
| Characterization of the symmetrical benzimidazole twin drug TL1228: the role as viral entry inhibitor for fighting COVID-19 | 1-gen-2024 | Murdocca, Michela; Andrade Santos-Filho, Osvaldo; De Masi, Claudia; dos Santos Rodrigues, Edivaldo; Campos de Souza, Claudia Valeria; De Santis, Riccardo; Amatore, Donatella; Latini, Andrea; Schipani, Rossella; di Rienzo Businco, Lino; Brandimarte, Bruno; Grilli, Giorgia; Huang, Tien L; Mayence, Annie S; Lista, Florigio; Duranti, Andrea; Sangiuolo, Federica; Vanden Eynde, Jean Jacques; Novelli, Giuseppe | |
| Endocannabinoid Degradation Enzyme Inhibitors as Potential Antipsychotics: A Medicinal Chemistry Perspective | 1-gen-2023 | Mangiatordi, Giuseppe Felice; Cavalluzzi, Maria Maddalena; Delre, Pietro; Lamanna, Giuseppe; Lomuscio, Maria Cristina; Saviano, Michele; Majoral, Jean-Pierre; Mignani, Serge; Duranti, Andrea; Lentini, Giovanni | |
| Synthesis and Biological Evaluation of 6-O-Sucrose Monoester Glycolipids as Possible New Antifungal Agents | 1-gen-2023 | Verboni, Michele; Sisti, Maurizio; Campana, Raffaella; Benedetti, Serena; Palma, Francesco; Potenza, Lucia; Lucarini, Simone; Duranti, Andrea | |
| Synthetic Methodologies and Therapeutic Potential of Indole-3-Carbinol (I3C) and Its Derivatives | 1-gen-2023 | Centofanti, Federica; Buono, Alessandro; Verboni, Michele; Tomino, Carlo; Lucarini, Simone; Duranti, Andrea; Pandolfi, Pier Paolo; Novelli, Giuseppe | |
| Sugar-Based Monoester Surfactants: Synthetic Methodologies, Properties, and Biological Activities | 1-gen-2023 | Verboni, Michele; Romano Perinelli, Diego; Buono, Alessandro; Campana, Raffaella; Sisti, Maurizio; Duranti, Andrea; Lucarini, Simone | |
| The influence of mannose-based esters on the mesophase behaviour of lyotropic liquid crystalline nanosystems as drug delivery vectors | 1-gen-2023 | Tiboni, Mattia; Astolfi, Paola; Verboni, Michele; Benedetti, Serena; Giorgini, Elisabetta; Notarstefano, Valentina; Vita, Francesco; Ranieri, Simone; Duranti, Andrea; Lucarini, Simone; Casettari, Luca; Pisani, Michela | |
| An Investigation on the Relationships between Mass Spectrometric Collisional Data and Biological Activity/Stability of Some N-Acylethanolamine Acid Amidase (NAAA) β-Lactone Inhibitors | 1-gen-2023 | Isak, Ilena; Duranti, Andrea; Traldi, Pietro | |
| Characterization of URB Series Synthetic Cannabinoids by HRMS and UHPLC–MS/MS | 1-gen-2023 | Agostini, Marco; Favretto, Donata; Renzoni, Caterina; Vogliardi, Susanna; Duranti, Andrea | |
| The Endocannabinoid System as a Target for Neuroprotection/Neuroregeneration in Perinatal Hypoxic–Ischemic Brain Injury | 1-gen-2023 | Duranti, Andrea; Beldarrain, Gorane; Álvarez, Antonia; Sbriscia, Matilde; Carloni, Silvia; Balduini, Walter; Alonso-Alconada, Daniel | |
| Synthesis and Properties of Sucrose- and Lactose-Based Aromatic Ester Surfactants as Potential Drugs Permeability Enhancers | 1-gen-2023 | Verboni, Michele; Perinelli, Diego Romano; Qiu, Carol Yingshan; Tiboni, Mattia; Aluigi, Annalisa; Lucarini, Simone; Lam, Jenny K. W.; Duranti, Andrea | |
| Characterization and Preliminary In Vitro Antioxidant Activity of a New Multidrug Formulation Based on the Co-Encapsulation of Rutin and the α-Acylamino-β-Lactone NAAA Inhibitor URB894 within PLGA Nanoparticles | 1-gen-2023 | Gagliardi, Agnese; Voci, Silvia; Ambrosio, Nicola; Fresta, Massimo; Duranti, Andrea; Cosco, Donato | |
| Inhibition of Fatty Acid Amide Hydrolase (FAAH) Regulates NF-kb Pathways Reducing Bleomycin-Induced Chronic Lung Inflammation and Pulmonary Fibrosis | 1-gen-2023 | Genovese, Tiziana; Duranti, Andrea; Monaco, Francesco; Siracusa, Rosalba; Fusco, Roberta; Impellizzeri, Daniela; D'Amico, Ramona; Cordaro, Marika; Cuzzocrea, Salvatore; Di Paola, Rosanna | |
| Synthesis and Biological Characterization of the New Glycolipid Lactose Undecylenate (URB1418) | 1-gen-2022 | Verboni, Michele; Benedetti, Serena; Campana, Raffaella; Palma, Francesco; Potenza, Lucia; Sisti, Maurizio; Duranti, Andrea; Lucarini, Simone | |
| A combination of sugar esters and chitosan to promote in vivo wound care | 1-gen-2022 | Tiboni, Mattia; Elmowafy, Enas; El-Derany, Marwa O; Benedetti, Serena; Campana, Raffaella; Verboni, Michele; Potenza, Lucia; Palma, Francesco; Citterio, Barbara; Sisti, Maurizio; Duranti, Andrea; Lucarini, Simone; Soliman, Mahmoud E; Casettari, Luca | |
| The Synthetic Cannabinoid URB447 Exerts Antitumor and Antimetastatic Effect in Melanoma and Colon Cancer | 1-gen-2022 | Benedicto, Aitor; Arteta, Beatriz; Duranti, Andrea; Alonso-Alconada, Daniel | |
| Indole-3-carbinol in vitro antiviral activity against SARS-Cov-2 virus and in vivo toxicity | 1-gen-2022 | Centofanti, Federica; Alonzi, Tonino; Latini, Andrea; Spitalieri, Paola; Murdocca, Michela; Chen, Xiaodong; Cui, Weibo; Shang, Qianwen; Goletti, Delia; Shi, Yufang; Duranti, Andrea; Tomino, Carlo; Biancolella, Michela; Sangiuolo, Federica; Capobianchi, Maria Rosaria; Jain, Suresh; Novelli, Giuseppe; Pandolfi, Pier Paolo | |
| Fatty Acid Amide Hydrolase (FAAH) Inhibition Plays a Key Role in Counteracting Acute Lung Injury | 1-gen-2022 | Genovese, Tiziana; Duranti, Andrea; D'Amico, Ramona; Fusco, Roberta; Impellizzeri, Daniela; Peritore, Alessio Filippo; Crupi, Rosalia; Gugliandolo, Enrico; Cuzzocrea, Salvatore; Di Paola, Rosanna; Siracusa, Rosalba; Cordaro, Marika |
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