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Methods, Compositions, and Other Compounds for Modulation of Monoacylglycerol Lipase Pain, and Stress-related Disorders 1-gen-2006 Piomelli, D; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Hohmann, A.
Identification of a Bioactive Impurity Present in a Sample of URB754 1-gen-2006 Antonietti, Francesca; Duranti, Andrea; Tontini, Andrea; Mor, M; Rivara, S; Traldi, P; Astarita, G; King, A; Clapper, J; Piomelli, D; Tarzia, Giorgio
Pharmacological Profile of the Selective FAAH Inhibitor KDS-4103 (URB597) 1-gen-2006 Piomelli, D; Tarzia, Giorgio; Duranti, Andrea; Tontini, Andrea; Mor, M; Compton, Tr; Dasse, O; Monaghan, Ep; Parrot, Ja; Putman, D.
The fatty-acid amide hydrolase inhibitor URB597 does not affect triacylglycerol hydrolysis in rat tissues 1-gen-2006 Clapper, Jr; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Piomelli, D.
Synthesis and Structure–Activity Relationships of FAAH Inhibitors: Cyclohexylcarbamic Acid Biphenyl Esters with Chemical Modulation at the Proximal Phenyl Ring 1-gen-2006 Tarzia, Giorgio; Duranti, Andrea; Gatti, G; Piersanti, Giovanni; Tontini, Andrea; Rivara, S; Lodola, A; Plazzi, Pv; Mor, M; Kathuria, S; Piomelli, D.
Selective inhibition of 2 - AG hydrolysis enhances endocannabinoid signaling in the hippocampus 1-gen-2005 Makara, Jk; Mor, M; Fegley, D; King, A; Szabo, Si; Kathuria, S; Astarita, G; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Rivara, S; Freund, Tf; Piomelli, D.
3D-QSAR study of carbamic acid aryl ester inhibitors of fatty acid amide hydrolase 1-gen-2005 Lodola, A; Mor, M; Rivara, S; Lorenzi, S; Plazzi, Pv; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Piomelli, D.
2 - Arachidonoylglycerol and anandamide are endocannabinoid mediators of stress - induced analgesia 1-gen-2005 Hohmann, Ag; SUPLITA RL, Ii; Bolton, Nm; Makara, Jk; Fegley, D; Mangieri, R; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Piomelli, D.
An endocannabinoid mechanism for stress-induced analgesia 1-gen-2005 Hohmann, Ag; SUPLITA RL, Ii; Bolton, Nm; Neely, Mh; Fegley, D; Mangieri, R; Krey, Jf; Walker, Jm; Holmes, Pv; Crystal, Jd; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Piomelli, D.
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors 1-gen-2005 Mor, M; Rivara, S; Lodola, A; Lorenzi, S; Bordi, F; Plazzi, Pv; Spadoni, Gilberto; Bedini, Annalida; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio
Antidepressant-like activity and modulation of brain monoaminergic transmission by blockade of anandamide hydrolysis 1-gen-2005 Gobbi, G; Bambico, Fr; Mangieri, R; Bortolato, M; Campolongo, P; Solinas, M; Cassano, T; Morgese, Mp; Debonnel, G; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Mor, M; Trezza, V; Goldberg, Sr; Cuomo, V; Piomelli, D.
Characterization of the Fatty Acid Amide Hydrolase Inhibitor Cyclohexyl Carbamic Acid 3'-Carbamoyl-biphenyl-3-yl Ester (URB597): Effects on Anandamide and Oleoylethanolamide Deactivation 1-gen-2005 Fegley, D; Gaetani, S; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio; Piomelli, D.
Selective inhibition of 2-AG hydrolysis enhances endocannabinoid signaling in hippocampus 1-gen-2005 Makara, Jk; Mor, M; Fegley, D; Szabó, Si; Kathuria, S; Astarita, G; Duranti, Andrea; Tontini, Andrea; Tarzia, Giorgio; Rivara, S; Freund, Tf; Piomelli, D.
Anthranilic acid based CCK1 antagonists: the 2-indole moiety may represent a "needle" according to the recent homonymous concept 1-gen-2004 Varnavas, A.; Lassiani, L.; Valenta, V.; Berti, F.; Tontini, Andrea; Mennuni, L.; Makovec, F.
Modulation of Anxiety Through Blockade of Anandamide Hydrolysis 1-gen-2004 Piomelli, D; Duranti, Andrea; Tontini, Andrea; Mor, M; Tarzia, Giorgio
Structure-Activity Relationships of Alkylcarbamic Acid Aryl Esters, as Fatty Acid Amide Hydrolase Inhibitors 1-gen-2004 Tarzia, Giorgio; Mor, M; Rivara, S; Lodola, A; Plazzi, Pv; Duranti, Andrea; Tontini, Andrea; Piersanti, Giovanni; Kathuria, S; Piomelli, D.
A linear relationship between MS/MS data and FAAH inhibitory activity of some carbamates 1-gen-2004 Basso, E; Duranti, Andrea; Mor, M; Piomelli, D; Tontini, Andrea; Tanzia, G; Traldi, P; Tarzia, Giorgio
Inhibition of intracellular anandamide hydrolysis enhances noradrenergic trasmission 1-gen-2004 Bambico, F; Cassano, T; Cuomo, V; Tarzia, Giorgio; Mor, M; Duranti, Andrea; Tontini, Andrea; Piomelli, D; Gobbi, G.
N-alchil-O-arilcarbammati come inibitori delle idrolasi delle ammidi degli acidi grassi (FAAH): aspetti meccanicistici 1-gen-2004 Tarzia, Giorgio; Mor, M; Traldi, P; Duranti, Andrea; Piersanti, Giovanni; Tontini, Andrea; Rivara, S; Lodola, A; Plazzi, Pv; Basso, E; Kathuria, S; Piomelli, D.
Characterization of the fatty acid amide hydrolase inhibitor URB597 1-gen-2004 Fegley, D; Gaetani, S; Tarzia, Giorgio; Mor, M; Duranti, Andrea; Tontini, Andrea; Piomelli, D.
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