RETINI, MICHELE
RETINI, MICHELE
Dipartimento di Scienze Biomolecolari (DISB)
Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties
2022-01-01 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
Boosting GSH Using the Co-Drug Approach: I-152, a Conjugate of N-acetyl-cysteine and β-mercaptoethylamine
2019-01-01 Crinelli, Rita; Zara, Carolina; Smietana, Michaël; Retini, Michele; Magnani, Mauro; Fraternale, Alessandra
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology
2020-01-01 Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni
Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma
2021-01-01 Castelli, Riccardo; Taranto, Sara; Furiassi, Lucia; Bozza, Nicole; Marseglia, Giuseppe; Ferlenghi, Francesca; Rivara, Silvia; Retini, Michele; Bedini, Annalida; Spadoni, Gilberto; Matarazzo, Sara; Ronca, Roberto; Presta, Marco; Mor, Marco; Giacomini, Arianna
Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin
2019-01-01 Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Mari, Michele; Piersanti, Giovanni
Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone
2021-01-01 Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni
General synthesis of unnatural 4-, 5-, 6-, and 7-bromo-d-tryptophans by means of a regioselective indole alkylation
2020-01-01 Bartoccini, Francesca; Fanini, Fabiola; Retini, Michele; Piersanti, Giovanni
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign
2020-01-01 Linciano, Pasquale; Cullia, Gregorio; Borsari, Chiara; Santucci, Matteo; Ferrari, Stefania; Witt, Gesa; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Santarém, Nuno; Cordeiro da Silva, Anabela; Conti, Paola; Bolognesi, Maria Laura; Roberti, Marinella; Prati, Federica; Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni; Cavalli, Andrea; Goldoni, Luca; Bertozzi, Sine Mandrup; Bertozzi, Fabio; Brambilla, Enzo; Rizzo, Vincenzo; Piomelli, Daniele; Pinto, Andrea; Bandiera, Tiziano; Costi, Maria Paola
Intracellular Redox-Modulated Pathways as Targets for Effective Approaches in the Treatment of Viral Infection
2021-01-01 Fraternale, Alessandra; Zara, Carolina; De Angelis, Marta; Nencioni, Lucia; Palamara, Anna Teresa; Retini, Michele; Di Mambro, Tomas; Magnani, Mauro; Crinelli, Rita
Large-Scale Preparation of N-Butanoyl-l-glutathione (C4-GSH)
2019-01-01 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Fraternale, Alessandra; Piersanti, Giovanni
Novel, Chiral, and Enantiopure C2‐Symmetric Thioureas Promote Asymmetric Protio‐Pictet‐Spengler Reactions by Anion‐Binding Catalysis
2021-01-01 Retini, Michele; Bartoccini, Francesca; Zappia, Giovanni; Piersanti, Giovanni
Organocatalytic Aza-Friedel-Crafts/Lactonization Domino Reaction of Naphthols and Phenols with 2-Acetamidoacrylate to Naphtho- and Benzofuranones Bearing a Quaternary Center at the C3 Position
2018-01-01 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Bartolucci, Silvia; Piersanti, Giovanni
Single‐Step Synthesis of Dehydroalanine Derivatives via a Brønsted Acid‐Catalyzed Multicomponent Reaction
2020-01-01 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Galarini, Roberta; Bartolucci, Silvia; Piersanti, Giovanni
Total Synthesis of (-)-Clavicipitic Acid via γ,γ-Dimethylallyltryptophan (DMAT) and Chemoselective C-H Hydroxylation
2019-01-01 Bartoccini, Francesca; Venturi, Silvia; Retini, Michele; Mari, Michele; Piersanti, Giovanni
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties | 1-gen-2022 | Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni | |
Boosting GSH Using the Co-Drug Approach: I-152, a Conjugate of N-acetyl-cysteine and β-mercaptoethylamine | 1-gen-2019 | Crinelli, Rita; Zara, Carolina; Smietana, Michaël; Retini, Michele; Magnani, Mauro; Fraternale, Alessandra | |
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology | 1-gen-2020 | Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni | |
Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma | 1-gen-2021 | Castelli, Riccardo; Taranto, Sara; Furiassi, Lucia; Bozza, Nicole; Marseglia, Giuseppe; Ferlenghi, Francesca; Rivara, Silvia; Retini, Michele; Bedini, Annalida; Spadoni, Gilberto; Matarazzo, Sara; Ronca, Roberto; Presta, Marco; Mor, Marco; Giacomini, Arianna | |
Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin | 1-gen-2019 | Retini, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Mari, Michele; Piersanti, Giovanni | |
Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone | 1-gen-2021 | Bartoccini, Francesca; Regni, Alessio; Retini, Michele; Piersanti, Giovanni | |
General synthesis of unnatural 4-, 5-, 6-, and 7-bromo-d-tryptophans by means of a regioselective indole alkylation | 1-gen-2020 | Bartoccini, Francesca; Fanini, Fabiola; Retini, Michele; Piersanti, Giovanni | |
Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign | 1-gen-2020 | Linciano, Pasquale; Cullia, Gregorio; Borsari, Chiara; Santucci, Matteo; Ferrari, Stefania; Witt, Gesa; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Santarém, Nuno; Cordeiro da Silva, Anabela; Conti, Paola; Bolognesi, Maria Laura; Roberti, Marinella; Prati, Federica; Bartoccini, Francesca; Retini, Michele; Piersanti, Giovanni; Cavalli, Andrea; Goldoni, Luca; Bertozzi, Sine Mandrup; Bertozzi, Fabio; Brambilla, Enzo; Rizzo, Vincenzo; Piomelli, Daniele; Pinto, Andrea; Bandiera, Tiziano; Costi, Maria Paola | |
Intracellular Redox-Modulated Pathways as Targets for Effective Approaches in the Treatment of Viral Infection | 1-gen-2021 | Fraternale, Alessandra; Zara, Carolina; De Angelis, Marta; Nencioni, Lucia; Palamara, Anna Teresa; Retini, Michele; Di Mambro, Tomas; Magnani, Mauro; Crinelli, Rita | |
Large-Scale Preparation of N-Butanoyl-l-glutathione (C4-GSH) | 1-gen-2019 | Bartoccini, Francesca; Mari, Michele; Retini, Michele; Fraternale, Alessandra; Piersanti, Giovanni | |
Novel, Chiral, and Enantiopure C2‐Symmetric Thioureas Promote Asymmetric Protio‐Pictet‐Spengler Reactions by Anion‐Binding Catalysis | 1-gen-2021 | Retini, Michele; Bartoccini, Francesca; Zappia, Giovanni; Piersanti, Giovanni | |
Organocatalytic Aza-Friedel-Crafts/Lactonization Domino Reaction of Naphthols and Phenols with 2-Acetamidoacrylate to Naphtho- and Benzofuranones Bearing a Quaternary Center at the C3 Position | 1-gen-2018 | Bartoccini, Francesca; Mari, Michele; Retini, Michele; Bartolucci, Silvia; Piersanti, Giovanni | |
Single‐Step Synthesis of Dehydroalanine Derivatives via a Brønsted Acid‐Catalyzed Multicomponent Reaction | 1-gen-2020 | Bartoccini, Francesca; Mari, Michele; Retini, Michele; Galarini, Roberta; Bartolucci, Silvia; Piersanti, Giovanni | |
Total Synthesis of (-)-Clavicipitic Acid via γ,γ-Dimethylallyltryptophan (DMAT) and Chemoselective C-H Hydroxylation | 1-gen-2019 | Bartoccini, Francesca; Venturi, Silvia; Retini, Michele; Mari, Michele; Piersanti, Giovanni |