| Nome |
# |
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Observations concerning the synthesis of tryptamine homologues and branched tryptamine derivatives via the borrowing hydrogen process: synthesis of psilocin, bufotenin, and serotonin, file e18b865c-f087-1ee6-e053-3a05fe0ae544
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442
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Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents, file e18b865c-f506-1ee6-e053-3a05fe0ae544
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239
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Dithiol Based on L-Cysteine and Cysteamine as a Disulfide-Reducing Agent, file 8c19afb0-8874-4774-aea6-1ec5415d84bd
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205
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A simple, modular synthesis of C4-substituted tryptophan derivatives, file e18b865d-51ff-1ee6-e053-3a05fe0ae544
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174
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|
Organocatalytic Aza-Friedel-Crafts/Lactonization Domino Reaction of Naphthols and Phenols with 2-Acetamidoacrylate to Naphtho- and Benzofuranones Bearing a Quaternary Center at the C3 Position, file e18b865d-80e2-1ee6-e053-3a05fe0ae544
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104
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Synthesis of 2-substituted tryptophans via a C3- to C2-alkyl migration, file e18b865b-8cda-1ee6-e053-3a05fe0ae544
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86
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Asymmetric Alkylation of Cyclic Ketones with Dehydroalanine via H-Bond-Directing Enamine Catalysis: Straightforward Access to Enantiopure Unnatural α-Amino Acids, file 37fcc113-3e16-4afb-b0a0-8cfc6843609f
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85
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Palladium(II)-Catalyzed Cross-Dehydrogenative Coupling (CDC) of N-Phthaloyl Dehydroalanine Esters with Simple Arenes: Stereoselective Synthesis of Z-Dehydrophenylalanine Derivatives, file e18b865d-8673-1ee6-e053-3a05fe0ae544
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83
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Palladium(II)-Catalyzed Intramolecular Oxidative C−H/C−H Cross-Coupling Reaction of C3,N-linked Biheterocycles: Rapid Access to Polycyclic Nitrogen Heterocycles, file e18b865d-5a17-1ee6-e053-3a05fe0ae544
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70
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Total Synthesis of (-)-Clavicipitic Acid via γ,γ-Dimethylallyltryptophan (DMAT) and Chemoselective C-H Hydroxylation, file e18b865d-6c38-1ee6-e053-3a05fe0ae544
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69
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Synthesis of Tryptamine Derivatives via a Direct, One-Pot Reductive Alkylation of Indoles, file e18b865b-8a98-1ee6-e053-3a05fe0ae544
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65
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Polycyclic Indolines by Acid-Mediated Intramolecular Dearomative Strategy: Reversing Indole Reactivity in the Pictet‒Spengler-Type Reaction, file e18b865d-8621-1ee6-e053-3a05fe0ae544
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59
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Iron-Catalyzed Direct C3-Benzylation of Indoles with Benzyl Alcohols through Borrowing Hydrogen, file e18b865d-6984-1ee6-e053-3a05fe0ae544
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54
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Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives, file e18b865d-5444-1ee6-e053-3a05fe0ae544
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50
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Novel, Chiral, and Enantiopure C2‐Symmetric Thioureas Promote Asymmetric Protio‐Pictet‐Spengler Reactions by Anion‐Binding Catalysis, file e18b865d-761f-1ee6-e053-3a05fe0ae544
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38
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Asymmetric Total Synthesis of All Rugulovasine Stereoisomers and Preliminary Evaluation of Their Biological Properties, file f4b030c7-440c-4196-aa78-af49f0a8efc4
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30
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One-Pot Synthesis of Biheterocycles Based on Indole and Azole Scaffolds Using Tryptamines and 1,2-Diaza-1,3-dienes as Building Blocks, file e18b865d-5418-1ee6-e053-3a05fe0ae544
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28
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Synthesis of (−)-Epi-Indolactam V by an Intramolecular Buchwald–Hartwig C–N Coupling Cyclization Reaction, file e18b865b-8800-1ee6-e053-3a05fe0ae544
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15
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Direct, One-Pot Reductive Alkylation of Anilines with Functionalized Acetals Mediated by Triethylsilane and TFA. Straightforward Route for Unsymmetrically Substituted Ethylenediamine, file e18b865b-846c-1ee6-e053-3a05fe0ae544
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11
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Direct, Regioselective, and Chemoselective Preparation of Novel Boronated Tryptophans by Friedel–Crafts Alkylation, file e18b865b-860f-1ee6-e053-3a05fe0ae544
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11
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Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives, file e18b865b-879e-1ee6-e053-3a05fe0ae544
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10
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Synthesis and Biological Evaluation of Metabolites of 2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), A Potent Antagonist of the A2AAdenosine Receptor for the Treatment of Parkinson’s Disease, file e18b865b-87fe-1ee6-e053-3a05fe0ae544
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10
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Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign, file 0e81fcb5-1a04-4a3e-89e2-f677dea37cb4
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7
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Targeting SARS-CoV-2 by synthetic dual-acting thiol compounds that inhibit Spike/ACE2 interaction and viral protein production, file b7655352-b690-4009-8f5c-941be50fcb29
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7
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Organocatalytic synthesis of α-quaternary amino acid derivatives via aza-Friedel–Crafts alkylation of indoles with simple α-amidoacrylates, file e18b865b-850d-1ee6-e053-3a05fe0ae544
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7
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Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions, file e18b865b-8cc8-1ee6-e053-3a05fe0ae544
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7
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An efficient, economical synthesis of hydroxytyrosol and its protected forms via Baeyer–Villiger oxidation, file e18b865b-850c-1ee6-e053-3a05fe0ae544
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6
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Synthesis of (E)-8-(3-Chlorostyryl)caffeine Analogues Leading to 9-Deazaxanthine Derivatives as Dual A2AAntagonists/MAO-B Inhibitors, file e18b865b-8cf9-1ee6-e053-3a05fe0ae544
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6
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Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin, file e18b865c-fa2a-1ee6-e053-3a05fe0ae544
|
6
|
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Enantioselective organocatalytic strategies to noncanonical α‐amino acids, file 0cbf48bc-9ed0-4bcd-941b-2e212b9db10a
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5
|
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Photoredox catalysis enabling decarboxylative radical cyclization of γ,γ-dimethylallyltryptophan (DMAT) derivatives: formal synthesis of 6,7-secoagroclavine, file da208138-83b8-4b5e-afa0-050a983cca95
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5
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Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone, file e18b865d-965c-1ee6-e053-3a05fe0ae544
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5
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Synthesis and Fluorescence Properties of 4-Cyano and 4-Formyl Melatonin as Putative Melatoninergic Ligands, file 9770aeb4-e395-4df3-9424-ca9f0cf79b82
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4
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Organocatalyzed coupling of indoles with dehydroalanine esters: synthesis of bis(indolyl)propanoates and indolacrylates, file e18b865b-88e3-1ee6-e053-3a05fe0ae544
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4
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Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands, file e18b865b-a73f-1ee6-e053-3a05fe0ae544
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4
|
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Palladium(II)-Catalyzed Intramolecular Oxidative C−H/C−H Cross-Coupling Reaction of C3,N-linked Biheterocycles: Rapid Access to Polycyclic Nitrogen Heterocycles, file e18b865c-0f3b-1ee6-e053-3a05fe0ae544
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4
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General Access to Clavine Alkaloids via a Rhodium(I)‐Catalyzed Diastereoselective Hayashi‐Miyaura Reaction, file ad8d6969-feaf-4923-85f3-d65fcbbb9b0e
|
3
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Iron-Catalyzed Direct C3-Benzylation of Indoles with Benzyl Alcohols through Borrowing Hydrogen, file e18b865c-353e-1ee6-e053-3a05fe0ae544
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3
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A Short Synthesis of (−)‐6,7‐Secoagroclavine via Metal‐Free Reductive Coupling, file e763ee38-25a4-4584-a457-d71cfb8e0832
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3
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Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign, file 1441af39-77d0-42ab-88d6-41793dfb17c6
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2
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Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin, file 9ea59d34-f973-4949-9da8-12176721df48
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2
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One-Pot Synthesis of Biheterocycles Based on Indole and Azole Scaffolds Using Tryptamines and 1,2-Diaza-1,3-dienes as Building Blocks, file e18b865b-d305-1ee6-e053-3a05fe0ae544
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2
|
|
Observations concerning the synthesis of tryptamine homologues and branched tryptamine derivatives via the borrowing hydrogen process: synthesis of psilocin, bufotenin, and serotonin, file e18b865b-d4da-1ee6-e053-3a05fe0ae544
|
2
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|
Palladium(II)-Catalyzed Cross-Dehydrogenative Coupling (CDC) of N-Phthaloyl Dehydroalanine Esters with Simple Arenes: Stereoselective Synthesis of Z-Dehydrophenylalanine Derivatives, file e18b865b-d635-1ee6-e053-3a05fe0ae544
|
2
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|
A simple, modular synthesis of C4-substituted tryptophan derivatives, file e18b865b-dfdb-1ee6-e053-3a05fe0ae544
|
2
|
|
Synthesis of Tetrahydropyridazine Amino Acid Derivatives by a Formal [4+2| Cycloaddition Reaction of 1,2-Diaza-1,3-dienes with Dehydroalanine Esters, file e18b865c-23e9-1ee6-e053-3a05fe0ae544
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2
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Large-Scale Preparation of N-Butanoyl-l-glutathione (C4-GSH), file e18b865c-fa27-1ee6-e053-3a05fe0ae544
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2
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Novel, Chiral, and Enantiopure C2‐Symmetric Thioureas Promote Asymmetric Protio‐Pictet‐Spengler Reactions by Anion‐Binding Catalysis, file e18b865d-761e-1ee6-e053-3a05fe0ae544
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2
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Synthesis and Reactivity of Uhle’s Ketone and Its Derivatives, file e18b865d-95da-1ee6-e053-3a05fe0ae544
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2
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2-n-Butyl- 9-methyl-8-(1,2,3)triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological Characterization, file e18b865b-7d43-1ee6-e053-3a05fe0ae544
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1
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Enantioselective Total Synthesis of (−)-Acylfulvene and (−)-Irofulven, file e18b865b-808c-1ee6-e053-3a05fe0ae544
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1
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Direct preparation of unsymmetrical difunctionalized cyclen derivatives by an Ugi multicomponent reaction, file e18b865b-81c1-1ee6-e053-3a05fe0ae544
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1
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Synthesis and Configuration Determination of All Enantiopure Stereoisomers of the Melatonin Receptor Ligand 4-Phenyl-2-propionamidotetralin using an Expedient Optical Resolution of 4-Phenyl-2-tetralone, file e18b865b-8544-1ee6-e053-3a05fe0ae544
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1
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Synthesis of (±)-cis-Clavicipitic Acid by a Rh(I)-Catalyzed Intramolecular Imine Reaction, file e18b865b-89f1-1ee6-e053-3a05fe0ae544
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1
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Brønsted Acid-Catalyzed Bisindolization of α-amido acetals: Synthesis and Anticancer activity of bis(indolyl)ethanamino derivatives, file e18b865b-89f5-1ee6-e053-3a05fe0ae544
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1
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Diastereo- and enantioselective hydrogenation of a challenging enamide derived from 4-phenyl-2-tetralone: an appealing shortcut towards enantiopure cis-2-aminotetraline derivatives, file e18b865b-a711-1ee6-e053-3a05fe0ae544
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1
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An improved synthesis of cis-4-phenyl-2-propionamidotetralin (4-P-PDOT): a selective MT2 melatonin receptor antagonist., file e18b865b-aa4e-1ee6-e053-3a05fe0ae544
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1
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Neutral urea-based receptors for phosphates: synthesis and spectrophotometric studies, file e18b865b-dfd9-1ee6-e053-3a05fe0ae544
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1
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DERIVATIVES OF TRIAZOLYL-IMIDAZOPYRIDINE AND OF THE TRIAZOLYLPURINES USEFUL AS LIGANDS OF THE ADENOSINE A2a RECEPTOR AND THEIR USE AS MEDICAMENTS., file e18b865b-e2fd-1ee6-e053-3a05fe0ae544
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1
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Divergent reactions of oxindoles with amino alcohols via the borrowing hydrogen process: oxindole ring opening vs. C3 alkylation, file e18b865c-a2ba-1ee6-e053-3a05fe0ae544
|
1
|
|
Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents, file e18b865c-f09a-1ee6-e053-3a05fe0ae544
|
1
|
|
C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology, file e18b865d-18ca-1ee6-e053-3a05fe0ae544
|
1
|
|
Polycyclic Indolines by Acid-Mediated Intramolecular Dearomative Strategy: Reversing Indole Reactivity in the Pictet‒Spengler-Type Reaction, file e18b865d-8620-1ee6-e053-3a05fe0ae544
|
1
|
| Totale |
2.058 |