IRIS
TARZIA, GIORGIO
 Distribuzione geografica
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Continente #
NA - Nord America 21.267
EU - Europa 15.269
AS - Asia 6.484
Continente sconosciuto - Info sul continente non disponibili 83
AF - Africa 56
SA - Sud America 36
OC - Oceania 30
AN - Antartide 1
Totale 43.226
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Nazione #
US - Stati Uniti d'America 21.147
GB - Regno Unito 6.100
CN - Cina 4.324
UA - Ucraina 2.750
IT - Italia 1.642
SE - Svezia 1.606
TR - Turchia 1.105
DE - Germania 866
FI - Finlandia 839
SG - Singapore 648
IE - Irlanda 590
FR - Francia 249
RU - Federazione Russa 191
CA - Canada 108
IN - India 107
BE - Belgio 105
JP - Giappone 91
EU - Europa 80
NL - Olanda 77
VN - Vietnam 64
KR - Corea 54
PL - Polonia 50
RO - Romania 41
AT - Austria 33
KE - Kenya 30
AU - Australia 25
CH - Svizzera 24
ES - Italia 24
HK - Hong Kong 20
IR - Iran 16
TG - Togo 16
BR - Brasile 12
ID - Indonesia 10
CL - Cile 9
HU - Ungheria 9
AL - Albania 8
MX - Messico 8
GR - Grecia 7
SA - Arabia Saudita 7
DK - Danimarca 6
PE - Perù 6
EE - Estonia 5
HR - Croazia 5
LU - Lussemburgo 5
NZ - Nuova Zelanda 5
AM - Armenia 4
BD - Bangladesh 4
BG - Bulgaria 4
IQ - Iraq 4
LA - Repubblica Popolare Democratica del Laos 4
MA - Marocco 4
PK - Pakistan 4
PT - Portogallo 4
RS - Serbia 4
SI - Slovenia 4
TW - Taiwan 4
A2 - ???statistics.table.value.countryCode.A2??? 3
CO - Colombia 3
CZ - Repubblica Ceca 3
IL - Israele 3
JM - Giamaica 3
LB - Libano 3
LT - Lituania 3
PH - Filippine 3
SK - Slovacchia (Repubblica Slovacca) 3
ZA - Sudafrica 3
AR - Argentina 2
BO - Bolivia 2
BY - Bielorussia 2
FK - Isole Falkland (Malvinas) 2
LV - Lettonia 2
MD - Moldavia 2
NO - Norvegia 2
SL - Sierra Leone 2
AE - Emirati Arabi Uniti 1
GS - Georgia del Sud e Isole Sandwich Australi 1
IM - Isola di Man 1
IS - Islanda 1
KW - Kuwait 1
LK - Sri Lanka 1
ME - Montenegro 1
MO - Macao, regione amministrativa speciale della Cina 1
MY - Malesia 1
PA - Panama 1
SC - Seychelles 1
SM - San Marino 1
Totale 43.226
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Città #
Southend 5.676
Woodbridge 3.099
Ann Arbor 2.232
Jacksonville 2.211
Houston 2.108
Chandler 1.869
Fairfield 1.852
Nanjing 1.220
Ashburn 1.026
Cambridge 895
Izmir 876
Wilmington 826
Seattle 709
Dublin 532
Boardman 492
Singapore 484
Nanchang 465
San Mateo 345
Beijing 320
Princeton 317
Helsinki 316
Hebei 249
Shenyang 242
Düsseldorf 226
Tianjin 210
Changsha 193
New York 192
Jiaxing 185
Kunming 162
Istanbul 145
Velikiy Novgorod 125
Brussels 103
Shanghai 97
Mülheim 93
San Diego 84
Des Moines 83
Bremen 81
Urbino 81
Jinan 75
Munich 73
Hangzhou 71
San Francisco 70
Toronto 69
Santa Clara 62
Orciano Di Pesaro 61
Guangzhou 59
Lanzhou 59
Venice 56
Amsterdam 55
Changchun 54
Dong Ket 54
Milan 54
Zhengzhou 54
Ningbo 53
Menlo Park 48
Seongnam 45
Dearborn 41
Kraków 40
London 37
Norwalk 37
Haikou 35
Vienna 33
Los Angeles 30
Rome 30
Shenzhen 28
Taizhou 26
Wuppertal 26
Auburn Hills 25
Fuzhou 22
Leawood 21
Parma 21
West Jordan 20
Ancona 19
Redwood City 19
Augusta 18
Florence 18
Nairobi 18
Timisoara 18
Frankfurt am Main 17
Lomé 16
Borås 15
Edinburgh 14
Hefei 14
Mcallen 14
Orange 14
Cava De' Tirreni 13
Focsani 13
Melbourne 13
Palermo 13
Portland 13
Mumbai 12
Dormagen 11
Napoli 11
Nuremberg 11
Padova 11
Wuhan 11
Wuxi 11
Ardabil 10
Chicago 10
Hanoi 10
Totale 32.352
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Nome #
Inibitori dell’enzima NAAA (N-Acylethanolamine-Hydrolizing Acid Amidase) come nuovi agenti antinfiammatori 768
1,5-BENZODIAZEPINE-2,4-DIONE GASTRIN AND CHOLECYSTOKININ-B-RECEPTOR ANTAGONISTS 336
1-(2-Alkylamidoethyl)-6-methoxyindole Derivatives: A New Class of Potent Indole Melatonin Analogues. 334
1-AMINOCYCLOPROPANE-1-CARBOXYLIC ACID DERIVATIVES AS LIGANDS AT THE GLYCINE-BINDING SITE OF THE N-METHYL-D-ASPARTATE RECEPTOR 329
1,7-DIHYDROPYRROLO[3,4-e][1,4]DIAZEPIN-2(3H)-ONE DERIVATIVES, AND THEIR USE AS ANTICONVULSANT AND ANTIANXIETY AGENTS 318
1-Aminocyclopropane-1-carboxylic acid derivatives as ligands at the glicine-site of the NMDA receptor. 317
ORGANIC REACTIONS OF FLUOROXY COMPOUNDS: ADDITION REACTIONS OF UNACTIVATED AND DEACTIVATED UNSATURATED LINKAGES OF STEROIDS 255
Scoperta del primo inibitore dell’enzima idrolasi delle ammidi degli acidi grassi (FAAH) ad azione periferica 247
ENOLATES OF 17,20:20,21-BISMETHYLENEDIOXYPREDNISONE 242
Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moieties 239
Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions 235
Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands 233
Tricyclic Alkylamides as Melatonin Receptor Ligands with Antagonist or Inverse Agonist Activity 227
Synthesis of benzo[1,2-d;3,4-d’]diimidazole and 1H-pyrazolo[4,3-b]pyridine as putative A2A receptor antagonists 223
Structure–Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors: Chemical and Biological Stability 223
2-n-Butyl- 9-methyl-8-(1,2,3)triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological Characterization 218
A new melatonin receptor ligand with mt1-agonist and MT2-antagonist properties 215
Synthesis and Biological Evaluation of Metabolites of 2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), A Potent Antagonist of the A2AAdenosine Receptor for the Treatment of Parkinson’s Disease 213
Alkyl 2 (Diphenyl-methyleneamino) acrylates in the Synthesis of α-Amino Acids 211
Biphenyl-3-yl alkylcarbamates as fatty acid amide hydrolase (FAAH) inhibitors: Steric effects of N-alkyl chain on rat plasma and liver stability 210
Synthesis and Biological Activity of new melatonin dimeric derivatives. 209
Antidepressant-like Activity of the Fatty Acid Amide Hydrolase Inhibitor URB597 in a Rat Model of Chronic Mild Stress 209
(E)-3-(2-(N-phenylcarbamoyl)vinyl)pyrrole-2-carboxylic acid derivatives. A novel class of glycine site antagonists. 205
Modulation of Anxiety Through Blockade of Anandamide Hydrolysis 205
Sintesi e studi di relazione struttura-attività/stabilità di carbammati inibitori dell’enzima FAAH 204
A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo 204
Identification of a Bioactive Impurity in a Commercial Sample of 6-Methyl-2-p-tolylaminobenzo[d][1,3]oxazin-4-one (URB754) 202
POSITIVE ION-MASS SPECTRA AND COLLISION-INDUCED DISSOCIATION OF SOME 2,3-DIDEHYDRO AMINO ACIDS 201
4,5-Dihydroisoxazole and 4,5-dihydro-1,2,4-oxadiazole derivatives from cycloaddition reactions of nitrile oxides to alkyl N-(diphenylmethylene)-α ,β -dehydroamino acids 198
An improved route to cycloalka[b]pyrrole 2-carboxylates 195
3-(2-Carbamoylvinyl)-4,5-dimethylpyrrole-2-carboxylic acids as ligands at the NMDA glycine-binding site: a study on the 2-carbamoylvinyl chain modification 195
Cyclohexylcarbamic Acid 3’-or 4’-Substituted Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: Synthesis Quantitative Structure–Activity Relationships, and Molecular Modeling Studies 195
TEICOPLANIN HYDRAZIDES AS ANTIBACTERIALS 191
10-(1-HYDROXYMETHYL)-11-OXO-1-AZATRICYCLOUNDEC-2-ENE-2-CARBOXYLIC ACID ESTERS USEFUL AS ANTIBACTERIAL AND PROCESS FOR THEIR PREPARATION 189
Toward the Definition of Stereochemical Requirements for MT(2)-Selective Antagonists and Partial Agonists by Studying 4-Phenyl-2-propionamidotetralin Derivatives 189
3,6-DISUBSTITUTED TRIAZOLO[3,4-a]PHTHALAZINE DERIVATIVES 188
2,4,5-TRISUBSTITUTED OXAZOLES 186
N-(Anilinoethyl)amides: design and synthesis of metabolically stable, selective melatonin receptor ligands. 185
Synthesis and Structure–Activity Relationships of a Series of Pyrrole Cannabinoid Receptor Agonists 184
Selective N-acylethanolamine-hydrolyzing acid amidase inhibition reveals a key role for endogenous palmitoylethanolamide in inflammation 184
N (Diphenylmethylene)-α,β−didehydroamino Acid Esters. Thermal and Lewis Acid Induced Dimerizations 182
Endocannabinoids in the Treatment of Mood Disorders: Evidence from Animal Models 181
Differentiation between isomeric 1-aminocyclopropane-1-carboxylic acid derivatives by means of chemical ionisation and mass selected collision induced dissociation 179
Plant-derived phenolic compounds prevent the DNA single-strand breakage and cytotoxicity induced by tert-butylhydroperoxide via an iron-chelating mechanism. 179
"Hot spots" in Medicinal Chemistry 179
SULLA MICELIANAMMIDE 178
Promotion of non-rapid eye movement sleep and activation of reticular thalamic neurons by a novel MT2 melatonin receptor ligand 178
Synthesis of (E)-8-(3-Chlorostyryl)caffeine Analogues Leading to 9-Deazaxanthine Derivatives as Dual A2AAntagonists/MAO-B Inhibitors 178
Peripherally Restricted FAAH Inhibitors 178
GENERALISED ELECTROPHILIC FLUORINATION BY FLUOROXY COMPOUNDS 178
Antidepressant-like activity and modulation of brain monoaminergic transmission by blockade of anandamide hydrolysis 177
X-RAY STRUCTURE DETERMINATION OF MEXIPROSTIL, A NEW GASTROPROTECTIVE 16-METHOXY-16METHYL-PGE1 ANALOGUE 176
Mechanisms of action and antiproliferative properties of URB631 in human breast cancer 176
5-(2-Ethyl-phenyl)-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole (DL-111-IT ) and related compounds induce morphological apoptotic patterns in cultures of human tumor cell lines 175
Synthesis and Structure–Activity Relationship (SAR) of 2-Methyl-4-oxo-3-oxetanyl Carbamic Acid Esters, a Class of Potent N-Acylethanolamine Acid Amidase (NAAA) Inhibitors 175
Synthesis and Quantitative Structure–Activity Relationship of Fatty Acid Amide Hydrolase Inhibitors: Modulation at the N-Portion of Biphenyl-3-yl Alkylcarbamates 174
Composition and Methods of Inhibiting N-Acylethanolamine-hydrolyzing Acid Amidase 173
Design, Synthesis and Structure–Activity Relationships of Alkylcarbamic Acid Aryl Esters, a New Class of Fatty Acid Amide Hydrolase Inhibitors 171
Synthesis, Enantiomeric Resolution and Structure-Activity Relationship Study for a Series of 10,11-Dihydro-5H-dibenzo[a,d]cycloheptene MT2 Receptor Antagonists. 170
Structural determinants of peripheral O-arylcarbamate FAAH inhibitors render them dual substrates for Abcb1 and Abcg2 and restrict their access to the brain 170
SYNTHESIS AND BIOLOGICAL PROPERTIES OF N63-CARBOXAMIDES OF TEICOPLANIN ANTIBIOTICS. STRUCTURE-ACTIVITY RELATIONSHIPS. 169
MELATONIN RECEPTOR AGONISTS: SAR AND APPLICATIONS TO THE TREATMENT OF SLEEP-WAKE DISORDERS 168
5-halo-tryptamine derivatives used as ligands of the 5-ht6 and/or 5-ht7 serotonin receptors, preparation, and therapeutic use.. 168
UNIVERSITY EDUCATION OF MEDICINAL CHEMISTS: COMPARISON OF EIGHT COUNTRIES 166
Synthesis and Structure–Activity Relationships of FAAH Inhibitors: Cyclohexylcarbamic Acid Biphenyl Esters with Chemical Modulation at the Proximal Phenyl Ring 166
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors 166
The Fatty Acid Amide Hydrolase Inhibitor URB597 (Cyclohexylcarbamic Acid 3’-Carbamoylbiphenyl-3-yl Ester) Reduces Neuropathic Pain after Oral Administration in Mice 165
URB602 Inhibits Monoacylglycerol Lipase and Selectively Blocks 2-Arachidonoylglycerol Degradation in Intact Brain Slices 164
ANGIOTENSIN CONVERTING ENZYME INHIBITORS AS ANTIHYPERTENSIVE AGENTS: 1-[´2-MERCAPTOCYCLOALKYL`CARBONYL]-L-PROLINES 162
Selective inhibition of 2-AG hydrolysis enhances endocannabinoid signaling in hippocampus 162
2,3-Dehydroamino acid derivatives as intermediates in the synthesis of heterocyclic compounds. 162
Reassessing the melatonin pharmacophore: enantiomeric resolution, pharmacological activity, structure analysis, and molecular modeling of a constrained chiral melatonin analogue. 162
The collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity 162
6-(ALKYLAMINO)-3-ARYL-1,2,4-TRIAZOLO[3,4-A]PHTHALAZINES. A NEW CLASS OF BENZODIAZEPINE RECEPTOR LIGANDS 161
Design and synthesis of N-[3,3-diphenyl-propenyl]alkanamides as a novel class of potent MT2-selective Melatonin receptor ligands 160
DEAMINOTEICOPLANIN AND ITS DERIVATIVES. SYNTHESIS, ANTIBACTERIAL ACTIVITY, AND BINDING STRENGTH TO Ac-D-ALA-D-ALA 160
The fatty-acid amide hydrolase inhibitor URB597 does not affect triacylglycerol hydrolysis in rat tissues 160
O-Biphenyl-3-yl Carbamates as Peripheral FAAH Inhibitors: Synthesis and Structure–Activity (SAR) Relationship Studies 159
N-(DIPHENYLMETHYLENE)-ALPHA,BETA-DIDEHYDROAMINO ACID ESTERS. THERMAL AND LEWIS ACID INDUCED DIMERIZATIONS 158
SUITABILITY OF FAST-ION BOMBARDMENT MASS SPECTROMETRY FOR THE INVESTIGATION OF 11,4-DIHYDROPYRIDINE DERIVATIVES 158
Conformationally Restrained Melatonin Analogs: Synthesis, Binding Affinity for the Melatonin Receptor, Evaluation of the Biological Activity, and Molecular Modeling Study 158
Bivalent Ligand Approach on N-[2-[(3-methoxyphenyl)methylamino]ethyl]acetamide. Synthesis, Binding Affinity and Intrinsic Acivity for MT(1) and MT(2) melatonin Receptors. 158
Modulation of anxiety through blockade of anandamide hydrolysis 157
2-[N-Acylamino(C1-C3)alkyl]indoles as MT1 melatonin receptor partial agonists, antagonists, and putative inverse agonists 157
Electron Impact Ionization and Fast Atom Bombardment Mass Spectrometry of Some 3,3-Dimethyl-1-(Isoxazol-3-yl)-triazenes. A New Class of Potential Anticancer Agents. 156
STRUCTURE-AFFINITY RELATIONSHIPS OF INDOLE-BASED MELATONIN ANALOGS 156
Melatonin prevents apoptosis induced by UV-B treatment in U937 cell line. 155
METABOLIC PATHWAYS OF THE ANTIHYPERTENSIVE AGENT, N-(2,5-DIMETHYL-1H-PYRROL-1-YL)-6-(4-MORPHOLINYL)-3-PYRIDAZINAMINE HYDROCHLORIDE. II.STUDIES IN THE DOG 155
An endocannabinoid mechanism for stress-induced analgesia 155
Sintesi e studi biologici preliminari su analoghi di URB937, il primo inibitore ad azione periferica dell'enzima FAAH 155
Synthesis and characterization of a peripherally restricted CB1 cannabinoid antagonist, URB447, that reduces feeding and body-weight gain in mice 154
PYRROLOPYRIDINE ANALOGS OF NALIDIXIC ACID. 2. PYRROLO[3,4-b]PYRIDINES 154
Metastable ion studies in the characterization melatonin isomers 153
Recent advances in the development of melatonin MT1 and MT2 receptor agonists 153
SYNTHESIS OF BETA-AMINOPYRROLES 152
N-Acyl-5- and -2,5-substituted tryptamines: synthesis, activity and affinity for human mt1 and MT2 melatonin receptors 152
Application of a non-electrophysiological method to study binding affinity and efficacy of glicine analogs to the glicine site of the NMDA receptor-ion channel complex. 152
Derivati 2-Acilamminoalchilindolici come Antagonisti/Agonisti Parziali della Melatonina 152
Melatonin receptor ligands: synthesis of new melatonin derivatives and comprehensive comparative molecular field analysis (CoMFA) study. 150
Alchilammidi tricicliche: legandi selettivi dei recettori melatoninergici MT1 e MT2 150
Totale 19.380
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Categoria #
all - tutte 131.767
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 131.767
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/20203.290 0 0 0 0 0 626 562 616 315 522 255 394
2020/20214.711 133 401 155 592 237 371 263 371 700 425 743 320
2021/20223.235 188 375 398 514 74 84 111 202 219 136 41 893
2022/20235.271 613 291 153 643 460 1.157 15 428 868 137 354 152
2023/20241.271 165 132 78 157 81 294 65 80 19 88 22 90
2024/20252.034 285 248 1.123 275 98 5 0 0 0 0 0 0
Totale 43.509