Observations concerning the synthesis of substituted tryptamine derivatives starting from indoles and 1,n-amino alcohols via the borrowing hydrogen process are discussed. This catalytic, single-step, and modular approach to tryptamines and homotryptamines allows the synthesis of branched and non branched tryptamines as well as tryptamine-based natural products such as psilocin, bufotenin, and serotonin.

Observations concerning the synthesis of tryptamine homologues and branched tryptamine derivatives via the borrowing hydrogen process: synthesis of psilocin, bufotenin, and serotonin

BARTOLUCCI, SILVIA;MARI, MICHELE;DI GREGORIO, GIOVANNI;PIERSANTI, GIOVANNI
2016-01-01

Abstract

Observations concerning the synthesis of substituted tryptamine derivatives starting from indoles and 1,n-amino alcohols via the borrowing hydrogen process are discussed. This catalytic, single-step, and modular approach to tryptamines and homotryptamines allows the synthesis of branched and non branched tryptamines as well as tryptamine-based natural products such as psilocin, bufotenin, and serotonin.
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Utilizza questo identificativo per citare o creare un link a questo documento: https://hdl.handle.net/11576/2634471
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