Sfoglia per Autore
Divergent reactions of oxindoles with amino alcohols via the borrowing hydrogen process: oxindole ring opening vs. C3 alkylation
2018 Di Gregorio, Giovanni; Mari, Michele; Bartolucci, Silvia; Bartoccini, Francesca; Piersanti, Giovanni
Organocatalytic Aza-Friedel-Crafts/Lactonization Domino Reaction of Naphthols and Phenols with 2-Acetamidoacrylate to Naphtho- and Benzofuranones Bearing a Quaternary Center at the C3 Position
2018 Bartoccini, Francesca; Mari, Michele; Retini, Michele; Bartolucci, Silvia; Piersanti, Giovanni
Polycyclic Indolines by Acid-Mediated Intramolecular Dearomative Strategy: Reversing Indole Reactivity in the Pictet‒Spengler-Type Reaction
2018 Ciccolini, Cecilia; Mari, Michele; Lucarini, Simone; Mantellini, Fabio; Piersanti, Giovanni; Favi, Gianfranco
Metodo di sintesi di derivati del glutatione [Method for the synthesis of glutathione derivatives]
2017 Bartoccini, Francesca; Fraternale, Alessandra; Piersanti, Giovanni
Iron-Catalyzed Direct C3-Benzylation of Indoles with Benzyl Alcohols through Borrowing Hydrogen
2017 DI GREGORIO, Giovanni; Mari, Michele; Bartoccini, Francesca; Piersanti, Giovanni
Palladium(II)-Catalyzed Intramolecular Oxidative C−H/C−H Cross-Coupling Reaction of C3,N-linked Biheterocycles: Rapid Access to Polycyclic Nitrogen Heterocycles
2017 Mantenuto, Serena; Ciccolini, Cecilia; Lucarini, Simone; Piersanti, Giovanni; Favi, Gianfranco; Mantellini, Fabio
Palladium(II)-Catalyzed Cross-Dehydrogenative Coupling (CDC) of N-Phthaloyl Dehydroalanine Esters with Simple Arenes: Stereoselective Synthesis of Z-Dehydrophenylalanine Derivatives
2016 Bartoccini, Francesca; Cannas, Diego Maria; Fini, Francesco; Piersanti, Giovanni
One-Pot Synthesis of Biheterocycles Based on Indole and Azole Scaffolds Using Tryptamines and 1,2-Diaza-1,3-dienes as Building Blocks
2016 Mantenuto, Serena; Lucarini, Simone; DE SANTI, Mauro; Piersanti, Giovanni; Brandi, Giorgio; Favi, Gianfranco; Mantellini, Fabio
Neutral urea-based receptors for phosphates: synthesis and spectrophotometric studies
2016 Formica, Mauro; Fusi, Vieri; Giorgi, Luca; Piersanti, Giovanni; Michele, Retini; Zappia, Giovanni
A simple, modular synthesis of C4-substituted tryptophan derivatives
2016 Bartoccini, Francesca; Bartolucci, Silvia; Mari, Michele; Piersanti, Giovanni
Observations concerning the synthesis of tryptamine homologues and branched tryptamine derivatives via the borrowing hydrogen process: synthesis of psilocin, bufotenin, and serotonin
2016 Bartolucci, Silvia; Mari, Michele; DI GREGORIO, Giovanni; Piersanti, Giovanni
Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands
2015 Pace, Silvia; Brogin, Giandomenico; Stasi, Maria Antonietta; Riccioni, Teresa; Borsini, Franco; Capocasa, Francesca; Manera, Francesco; Tallarico, Carlo; Grossi, Pietro; Vacondio, Federica; Bassi, Michele; Bartoccini, Francesca; Lucarini, Simone; Piersanti, Giovanni; Tarzia, Giorgio; Cabri, Walter; Minetti, Patrizia
Synthesis of Boron- and Silicon-Containing Amino Acids through Copper-Catalysed Conjugate Additions to Dehydroalanine Derivatives
2015 Bartoccini, Francesca; Bartolucci, Silvia; Lucarini, Simone; Piersanti, Giovanni
Iridium-Catalyzed Direct Synthesis of Tryptamine Derivatives from Indoles: Exploiting N-Protected β-Amino Alcohols as Alkylating Agents
2015 Bartolucci, Silvia; Mari, Michele; Bedini, Annalida; Piersanti, Giovanni; Spadoni, Gilberto
Derivatizzazione one-pot di indoli per la sintesi di triptofani, pirroloindoline, bis-indoli & co
2014 Lucarini, Simone; Piersanti, Giovanni; Duranti, Andrea; Spadoni, Gilberto
Brønsted Acid-Catalyzed Bisindolization of α-amido acetals: Synthesis and Anticancer activity of bis(indolyl)ethanamino derivatives
2014 Mari, Michele; Aurora, Tassoni; Lucarini, Simone; Fanelli, Mirco; Piersanti, Giovanni; Spadoni, Gilberto
Development of a practical and sustainable strategy for the synthesis of ST1535 by an iron-catalyzed Kumada cross-coupling reaction
2014 Bartoccini, Francesca; Piersanti, Giovanni; Silvia, Armaroli; Alberto, Cerri; Walter, Cabri
Synthesis of (±)-cis-Clavicipitic Acid by a Rh(I)-Catalyzed Intramolecular Imine Reaction
2014 Bartoccini, Francesca; Mariangela, Casoli; Mari, Michele; Piersanti, Giovanni
Synthesis of 2-substituted tryptophans via a C3- to C2-alkyl migration
2014 Mari, Michele; Lucarini, Simone; Bartoccini, Francesca; Piersanti, Giovanni; Spadoni, Gilberto
Synthesis of Tetrahydropyridazine Amino Acid Derivatives by a Formal [4+2| Cycloaddition Reaction of 1,2-Diaza-1,3-dienes with Dehydroalanine Esters
2013 Attanasi, ORAZIO ANTONIO; Favi, Gianfranco; G., Giorgi; Mantellini, Fabio; Moscatelli, Giada; Piersanti, Giovanni
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